Compile Data Set for Download or QSAR
Report error Found 18 Enz. Inhib. hit(s) with all data for entry = 50019498
TargetSerine/threonine-protein kinase PLK1(Human)
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50240826(AZD-1775 | MK-1775 | US11124518, Example AZD1775 |...)
Affinity DataIC50: 268nMAssay Description:Inhibition of PLK1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2024
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetSerine/threonine-protein kinase PLK1(Human)
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50619739(CHEMBL5403604)
Affinity DataIC50: 516nMAssay Description:Inhibition of PLK1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2024
Entry Details
PubMed
TargetSerine/threonine-protein kinase PLK1(Human)
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50619746(CHEMBL5403903)
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibition of PLK1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2024
Entry Details
PubMed
TargetSerine/threonine-protein kinase PLK1(Human)
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50619749(CHEMBL5432090)
Affinity DataIC50: 2.07E+3nMAssay Description:Inhibition of PLK1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2024
Entry Details
PubMed
TargetSerine/threonine-protein kinase PLK1(Human)
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50619743(CHEMBL5434663)
Affinity DataIC50: 2.09E+3nMAssay Description:Inhibition of PLK1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2024
Entry Details
PubMed
TargetSerine/threonine-protein kinase PLK1(Human)
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50619745(CHEMBL5440440)
Affinity DataIC50: 2.15E+3nMAssay Description:Inhibition of PLK1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2024
Entry Details
PubMed
TargetSerine/threonine-protein kinase PLK1(Human)
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50619738(CHEMBL5440332)
Affinity DataIC50: 2.35E+3nMAssay Description:Inhibition of PLK1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2024
Entry Details
PubMed
TargetSerine/threonine-protein kinase PLK1(Human)
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50619744(CHEMBL5406356)
Affinity DataIC50: 2.43E+3nMAssay Description:Inhibition of PLK1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2024
Entry Details
PubMed
TargetSerine/threonine-protein kinase PLK1(Human)
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50619752(CHEMBL5431802)
Affinity DataIC50: 2.97E+3nMAssay Description:Inhibition of PLK1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2024
Entry Details
PubMed
TargetSerine/threonine-protein kinase PLK1(Human)
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50619750(CHEMBL5427326)
Affinity DataIC50: 3.43E+3nMAssay Description:Inhibition of PLK1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2024
Entry Details
PubMed
TargetSerine/threonine-protein kinase PLK1(Human)
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50619741(CHEMBL5420142)
Affinity DataIC50: 3.77E+3nMAssay Description:Inhibition of PLK1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2024
Entry Details
PubMed
TargetSerine/threonine-protein kinase PLK1(Human)
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50619753(CHEMBL5393910)
Affinity DataIC50: 4.38E+3nMAssay Description:Inhibition of PLK1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2024
Entry Details
PubMed
TargetSerine/threonine-protein kinase PLK1(Human)
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50619747(CHEMBL5414912)
Affinity DataIC50: 5.41E+3nMAssay Description:Inhibition of PLK1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2024
Entry Details
PubMed
TargetSerine/threonine-protein kinase PLK1(Human)
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50619751(CHEMBL5405576)
Affinity DataIC50: 5.54E+3nMAssay Description:Inhibition of PLK1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2024
Entry Details
PubMed
TargetSerine/threonine-protein kinase PLK1(Human)
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50619740(CHEMBL5412194)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of PLK1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2024
Entry Details
PubMed
TargetSerine/threonine-protein kinase PLK1(Human)
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50619742(CHEMBL5425172)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of PLK1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2024
Entry Details
PubMed
TargetSerine/threonine-protein kinase PLK1(Human)
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50619737(CHEMBL5412009)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of PLK1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2024
Entry Details
PubMed
TargetSerine/threonine-protein kinase PLK1(Human)
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50619748(CHEMBL5421561)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of PLK1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2024
Entry Details
PubMed