Compile Data Set for Download or QSAR
Report error Found 16 Enz. Inhib. hit(s) with all data for entry = 50015826
TargetUrokinase-type plasminogen activator(Human)
Texas A&M University

Curated by ChEMBL
LigandPNGBDBM50589990(CHEMBL5169692)
Affinity DataIC50: 2.45E+3nMAssay Description:Inhibition of uPAR/uPA (unknown origin) interaction by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/19/2023
Entry Details
PubMed
TargetUrokinase-type plasminogen activator(Human)
Texas A&M University

Curated by ChEMBL
LigandPNGBDBM50589991(CHEMBL5186118)
Affinity DataIC50: 2.85E+3nMAssay Description:Inhibition of uPAR/uPA (unknown origin) interaction by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/19/2023
Entry Details
PubMed
TargetUrokinase-type plasminogen activator(Human)
Texas A&M University

Curated by ChEMBL
LigandPNGBDBM50589988(CHEMBL5183489)
Affinity DataIC50: 3.06E+3nMAssay Description:Inhibition of uPAR/uPA (unknown origin) interaction by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/19/2023
Entry Details
PubMed
TargetUrokinase-type plasminogen activator(Human)
Texas A&M University

Curated by ChEMBL
LigandPNGBDBM50589994(CHEMBL5199716)
Affinity DataIC50: 3.06E+3nMAssay Description:Inhibition of uPAR/uPA (unknown origin) interaction by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/19/2023
Entry Details
PubMed
TargetUrokinase-type plasminogen activator(Human)
Texas A&M University

Curated by ChEMBL
LigandPNGBDBM50589989(CHEMBL5169901)
Affinity DataIC50: 8.35E+3nMAssay Description:Inhibition of uPAR/uPA (unknown origin) interaction by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/19/2023
Entry Details
PubMed
TargetUrokinase-type plasminogen activator(Human)
Texas A&M University

Curated by ChEMBL
LigandPNGBDBM50589993(CHEMBL5187565)
Affinity DataIC50: 1.47E+4nMAssay Description:Inhibition of uPAR/uPA (unknown origin) interaction by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/19/2023
Entry Details
PubMed
TargetUrokinase-type plasminogen activator(Human)
Texas A&M University

Curated by ChEMBL
LigandPNGBDBM50589992(CHEMBL5182189)
Affinity DataIC50: 1.55E+4nMAssay Description:Inhibition of uPAR/uPA (unknown origin) interaction by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/19/2023
Entry Details
PubMed
TargetUrokinase-type plasminogen activator(Human)
Texas A&M University

Curated by ChEMBL
LigandPNGBDBM222350(IPR-1110 (1))
Affinity DataIC50: 1.84E+4nMAssay Description:Inhibition of uPAR/uPA (unknown origin) interaction by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/19/2023
Entry Details
PubMed
TargetUrokinase-type plasminogen activator(Human)
Texas A&M University

Curated by ChEMBL
LigandPNGBDBM222350(IPR-1110 (1))
Affinity DataKi:  700nMAssay Description:Inhibition of uPAR/uPA (unknown origin) interaction assessed as dissociation constant by fluorescence polarization (FP) assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/19/2023
Entry Details
PubMed
TargetUrokinase-type plasminogen activator(Human)
Texas A&M University

Curated by ChEMBL
LigandPNGBDBM50589990(CHEMBL5169692)
Affinity DataKi:  2.20E+3nMAssay Description:Inhibition of uPAR/uPA (unknown origin) interaction assessed as dissociation constant by fluorescence polarization (FP) assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/19/2023
Entry Details
PubMed
TargetUrokinase-type plasminogen activator(Human)
Texas A&M University

Curated by ChEMBL
LigandPNGBDBM50589992(CHEMBL5182189)
Affinity DataKi:  2.50E+3nMAssay Description:Inhibition of uPAR/uPA (unknown origin) interaction assessed as dissociation constant by fluorescence polarization (FP) assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/19/2023
Entry Details
PubMed
TargetUrokinase-type plasminogen activator(Human)
Texas A&M University

Curated by ChEMBL
LigandPNGBDBM50589991(CHEMBL5186118)
Affinity DataKi:  2.56E+3nMAssay Description:Inhibition of uPAR/uPA (unknown origin) interaction assessed as dissociation constant by fluorescence polarization (FP) assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/19/2023
Entry Details
PubMed
TargetUrokinase-type plasminogen activator(Human)
Texas A&M University

Curated by ChEMBL
LigandPNGBDBM50589988(CHEMBL5183489)
Affinity DataKi:  2.75E+3nMAssay Description:Inhibition of uPAR/uPA (unknown origin) interaction assessed as dissociation constant by fluorescence polarization (FP) assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/19/2023
Entry Details
PubMed
TargetUrokinase-type plasminogen activator(Human)
Texas A&M University

Curated by ChEMBL
LigandPNGBDBM50589994(CHEMBL5199716)
Affinity DataKi:  6.20E+3nMAssay Description:Inhibition of uPAR/uPA (unknown origin) interaction assessed as dissociation constant by fluorescence polarization (FP) assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/19/2023
Entry Details
PubMed
TargetUrokinase-type plasminogen activator(Human)
Texas A&M University

Curated by ChEMBL
LigandPNGBDBM50589989(CHEMBL5169901)
Affinity DataKi:  7.50E+3nMAssay Description:Inhibition of uPAR/uPA (unknown origin) interaction assessed as dissociation constant by fluorescence polarization (FP) assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/19/2023
Entry Details
PubMed
TargetUrokinase-type plasminogen activator(Human)
Texas A&M University

Curated by ChEMBL
LigandPNGBDBM50589993(CHEMBL5187565)
Affinity DataKi:  1.32E+4nMAssay Description:Inhibition of uPAR/uPA (unknown origin) interaction assessed as dissociation constant by fluorescence polarization (FP) assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/19/2023
Entry Details
PubMed