Compile Data Set for Download or QSAR
Report error Found 13 Enz. Inhib. hit(s) with all data for entry = 50016558
TargetMatrilysin(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50042944(cid_638278 | (E)-1-(2,4-Dihydroxy-phenyl)-3-(4-hyd...)
Affinity DataIC50: 8nMAssay Description:Inhibition of MMP7 in human U2OS cells by peptide microarray-based fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
Target72 kDa type IV collagenase(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50063917(CHEMBL279785 | marimastat | cid_119031 | (2S,3R)-N...)
Affinity DataIC50: 8nMAssay Description:Inhibition of MMP2 in human U2OS cells by peptide microarray-based fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetMatrix metalloproteinase-9(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50042944(cid_638278 | (E)-1-(2,4-Dihydroxy-phenyl)-3-(4-hyd...)
Affinity DataIC50: 10nMAssay Description:Inhibition of MMP9 in human U2OS cells by peptide microarray-based fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetMatrilysin(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50063917(CHEMBL279785 | marimastat | cid_119031 | (2S,3R)-N...)
Affinity DataIC50: 10nMAssay Description:Inhibition of MMP7 in human U2OS cells by peptide microarray-based fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
Target72 kDa type IV collagenase(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50042944(cid_638278 | (E)-1-(2,4-Dihydroxy-phenyl)-3-(4-hyd...)
Affinity DataIC50: 10nMAssay Description:Inhibition of MMP2 in human U2OS cells by peptide microarray-based fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetCollagenase 3(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50042944(cid_638278 | (E)-1-(2,4-Dihydroxy-phenyl)-3-(4-hyd...)
Affinity DataIC50: 14nMAssay Description:Inhibition of MMP13 in human U2OS cells by peptide microarray-based fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetInterstitial collagenase(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50042944(cid_638278 | (E)-1-(2,4-Dihydroxy-phenyl)-3-(4-hyd...)
Affinity DataIC50: 16nMAssay Description:Inhibition of MMP1 in human U2OS cells by peptide microarray-based fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetStromelysin-1(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50063917(CHEMBL279785 | marimastat | cid_119031 | (2S,3R)-N...)
Affinity DataIC50: 26nMAssay Description:Inhibition of MMP3 in human U2OS cells by peptide microarray-based fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetStromelysin-1(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50042944(cid_638278 | (E)-1-(2,4-Dihydroxy-phenyl)-3-(4-hyd...)
Affinity DataIC50: 81nMAssay Description:Inhibition of MMP3 in human U2OS cells by peptide microarray-based fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetCollagenase 3(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50063917(CHEMBL279785 | marimastat | cid_119031 | (2S,3R)-N...)
Affinity DataIC50: 128nMAssay Description:Inhibition of MMP13 in human U2OS cells by peptide microarray-based fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetCollagenase 3(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50595721(CHEMBL5204643)
Affinity DataIC50: 250nMAssay Description:Inhibition of MMP13 in human U2OS cells by peptide microarray-based fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetMatrix metalloproteinase-9(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50248691((1S)-1,5-anhydro-1-(1,3,6,7-tetrahydroxy-9-oxo-9H-...)
Affinity DataIC50: 250nMAssay Description:Inhibition of MMP9 in human U2OS cells by peptide microarray-based fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetMatrix metalloproteinase-9(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50063917(CHEMBL279785 | marimastat | cid_119031 | (2S,3R)-N...)
Affinity DataIC50: 795nMAssay Description:Inhibition of MMP9 in human U2OS cells by peptide microarray-based fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed