Report error Found 100 Enz. Inhib. hit(s) with all data for entry = 50019660
Affinity DataKi: 2.10nMAssay Description:Displacement of [3H]-ditolylguanidine from sigma 2 receptor/TMEM97 in rat PC-12 cells assessed as inhibition constant in the presence of (+)-pentazoc...More data for this Ligand-Target Pair
Ligand InfoSimilars
Affinity DataKi: 2.10nMAssay Description:Displacement of [3H]-ditolylguanidine from sigma 2 receptor/TMEM97 in rat PC-12 cells assessed as inhibition constant in the presence of (+)-pentazoc...More data for this Ligand-Target Pair
Ligand InfoSimilars
Affinity DataKi: 2.70nMAssay Description:Displacement of [3H]-ditolylguanidine from sigma 2 receptor/TMEM97 in rat PC-12 cells assessed as inhibition constant in the presence of (+)-pentazoc...More data for this Ligand-Target Pair
Ligand InfoSimilars
Affinity DataKi: 4.5nMAssay Description:Displacement of [3H]-ditolylguanidine from sigma 2 receptor/TMEM97 in rat PC-12 cells assessed as inhibition constant in the presence of (+)-pentazoc...More data for this Ligand-Target Pair
Ligand InfoSimilars
Affinity DataKi: 4.60nMAssay Description:Displacement of [3H]-ditolylguanidine from sigma 2 receptor/TMEM97 in rat PC-12 cells assessed as inhibition constant in the presence of (+)-pentazoc...More data for this Ligand-Target Pair
Ligand InfoSimilars
Affinity DataKi: 5.10nMAssay Description:Displacement of [3H]-ditolylguanidine from sigma 2 receptor/TMEM97 in rat PC-12 cells assessed as inhibition constant in the presence of (+)-pentazoc...More data for this Ligand-Target Pair
Affinity DataKi: 5.5nMAssay Description:Displacement of [3H]-ditolylguanidine from sigma 2 receptor/TMEM97 in rat PC-12 cells assessed as inhibition constant in the presence of (+)-pentazoc...More data for this Ligand-Target Pair
Ligand InfoSimilars
Affinity DataKi: 7.20nMAssay Description:Displacement of [3H]-ditolylguanidine from sigma 2 receptor/TMEM97 in rat PC-12 cells assessed as inhibition constant in the presence of (+)-pentazoc...More data for this Ligand-Target Pair
Ligand InfoSimilars
Affinity DataKi: 8.30nMAssay Description:Displacement of [3H]-ditolylguanidine from sigma 2 receptor/TMEM97 in rat PC-12 cells assessed as inhibition constant in the presence of (+)-pentazoc...More data for this Ligand-Target Pair
Ligand InfoSimilars
Affinity DataKi: 9.40nMAssay Description:Displacement of [3H]-ditolylguanidine from sigma 2 receptor/TMEM97 in rat PC-12 cells assessed as inhibition constant in the presence of (+)-pentazoc...More data for this Ligand-Target Pair
Ligand InfoSimilars
Affinity DataKi: 9.60nMAssay Description:Displacement of [3H]-ditolylguanidine from human sigma 2 receptor/TMEM97 transfected in HEK293 cells assessed as inhibition constant in the presence ...More data for this Ligand-Target Pair
Ligand InfoSimilars
Affinity DataKi: 12nMAssay Description:Displacement of [3H]-ditolylguanidine from sigma 2 receptor/TMEM97 in rat PC-12 cells assessed as inhibition constant in the presence of (+)-pentazoc...More data for this Ligand-Target Pair
Ligand InfoSimilars
TargetSigma non-opioid intracellular receptor 1(Guinea pig)
The University of Texas At Austin
Curated by ChEMBL
The University of Texas At Austin
Curated by ChEMBL
Affinity DataKi: 12nMAssay Description:Displacement of [3H](+)-pentazocine from sigma 1 receptor in guinea pig brain assessed as inhibition constant by competition binding assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
Affinity DataKi: 13nMAssay Description:Displacement of [3H]-ditolylguanidine from sigma 2 receptor/TMEM97 in rat PC-12 cells assessed as inhibition constant in the presence of (+)-pentazoc...More data for this Ligand-Target Pair
Ligand InfoSimilars
Affinity DataKi: 15nMAssay Description:Displacement of [3H]-ditolylguanidine from human sigma 2 receptor/TMEM97 transfected in HEK293 cells assessed as inhibition constant in the presence ...More data for this Ligand-Target Pair
Ligand InfoSimilars
TargetSigma non-opioid intracellular receptor 1(Guinea pig)
The University of Texas At Austin
Curated by ChEMBL
The University of Texas At Austin
Curated by ChEMBL
Affinity DataKi: 16nMAssay Description:Displacement of [3H](+)-pentazocine from sigma 1 receptor in guinea pig brain assessed as inhibition constant by competition binding assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
Affinity DataKi: 17nMAssay Description:Displacement of [3H]-ditolylguanidine from sigma 2 receptor/TMEM97 in rat PC-12 cells assessed as inhibition constant in the presence of (+)-pentazoc...More data for this Ligand-Target Pair
Ligand InfoSimilars
Affinity DataKi: 17nMAssay Description:Displacement of [3H]-ditolylguanidine from human sigma 2 receptor/TMEM97 transfected in HEK293 cells assessed as inhibition constant in the presence ...More data for this Ligand-Target Pair
Ligand InfoSimilars
Affinity DataKi: 17nMAssay Description:Displacement of [3H]-ditolylguanidine from human sigma 2 receptor/TMEM97 transfected in HEK293 cells assessed as inhibition constant in the presence ...More data for this Ligand-Target Pair
Ligand InfoSimilars
Affinity DataKi: 20nMAssay Description:Displacement of [3H]-ditolylguanidine from sigma 2 receptor/TMEM97 in rat PC-12 cells assessed as inhibition constant in the presence of (+)-pentazoc...More data for this Ligand-Target Pair
Ligand InfoSimilars
Affinity DataKi: 20nMAssay Description:Binding affinity at human Histamine H1 receptor assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand InfoSimilars
TargetSigma non-opioid intracellular receptor 1(Guinea pig)
The University of Texas At Austin
Curated by ChEMBL
The University of Texas At Austin
Curated by ChEMBL
Affinity DataKi: 21nMAssay Description:Displacement of [3H](+)-pentazocine from sigma 1 receptor in guinea pig brain assessed as inhibition constant by competition binding assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
Affinity DataKi: 21nMAssay Description:Displacement of [3H]-ditolylguanidine from sigma 2 receptor/TMEM97 in rat PC-12 cells assessed as inhibition constant in the presence of (+)-pentazoc...More data for this Ligand-Target Pair
Ligand InfoSimilars
Affinity DataKi: 23nMAssay Description:Binding affinity to sigma 2 receptor/TMEM97 (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
Affinity DataKi: 25nMAssay Description:Displacement of [3H]-ditolylguanidine from sigma 2 receptor/TMEM97 in rat PC-12 cells assessed as inhibition constant in the presence of (+)-pentazoc...More data for this Ligand-Target Pair
Ligand InfoSimilars
Affinity DataKi: 26nMAssay Description:Displacement of [3H]-ditolylguanidine from sigma 2 receptor/TMEM97 in rat PC-12 cells assessed as inhibition constant in the presence of (+)-pentazoc...More data for this Ligand-Target Pair
Ligand InfoSimilars
TargetSigma non-opioid intracellular receptor 1(Guinea pig)
The University of Texas At Austin
Curated by ChEMBL
The University of Texas At Austin
Curated by ChEMBL
Affinity DataKi: 33nMAssay Description:Displacement of [3H](+)-pentazocine from sigma 1 receptor in guinea pig brain assessed as inhibition constant by competition binding assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
Affinity DataKi: 33nMAssay Description:Displacement of [3H]-ditolylguanidine from human sigma 2 receptor/TMEM97 transfected in HEK293 cells assessed as inhibition constant in the presence ...More data for this Ligand-Target Pair
Ligand InfoSimilars
Affinity DataKi: 35nMAssay Description:Displacement of [3H]-ditolylguanidine from human sigma 2 receptor/TMEM97 transfected in HEK293 cells assessed as inhibition constant in the presence ...More data for this Ligand-Target Pair
Ligand InfoSimilars
Affinity DataKi: 35nMAssay Description:Displacement of [3H]-ditolylguanidine from sigma 2 receptor/TMEM97 in rat PC-12 cells assessed as inhibition constant in the presence of (+)-pentazoc...More data for this Ligand-Target Pair
Ligand InfoSimilars
TargetSigma non-opioid intracellular receptor 1(Guinea pig)
The University of Texas At Austin
Curated by ChEMBL
The University of Texas At Austin
Curated by ChEMBL
Affinity DataKi: 40nMAssay Description:Displacement of [3H](+)-pentazocine from sigma 1 receptor in guinea pig brain assessed as inhibition constant by competition binding assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
Affinity DataKi: 46nMAssay Description:Displacement of [3H]-ditolylguanidine from sigma 2 receptor/TMEM97 in rat PC-12 cells assessed as inhibition constant in the presence of (+)-pentazoc...More data for this Ligand-Target Pair
Affinity DataKi: 50nMAssay Description:Displacement of [3H]-ditolylguanidine from sigma 2 receptor/TMEM97 in rat PC-12 cells assessed as inhibition constant in the presence of (+)-pentazoc...More data for this Ligand-Target Pair
Ligand InfoSimilars
Affinity DataKi: 53nMAssay Description:Displacement of [3H]-ditolylguanidine from human sigma 2 receptor/TMEM97 transfected in HEK293 cells assessed as inhibition constant in the presence ...More data for this Ligand-Target Pair
Ligand InfoSimilars
TargetSigma non-opioid intracellular receptor 1(Human)
The University of Texas At Austin
Curated by ChEMBL
The University of Texas At Austin
Curated by ChEMBL
Affinity DataKi: 82nMAssay Description:Displacement of [3H](+)-pentazocine from human sigma 1 receptor transfected in HEK293 cells assessed as inhibition constant by competition binding as...More data for this Ligand-Target Pair
Ligand InfoSimilars
TargetSigma non-opioid intracellular receptor 1(Guinea pig)
The University of Texas At Austin
Curated by ChEMBL
The University of Texas At Austin
Curated by ChEMBL
Affinity DataKi: 86nMAssay Description:Displacement of [3H](+)-pentazocine from sigma 1 receptor in guinea pig brain assessed as inhibition constant by competition binding assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
Affinity DataKi: 90nMAssay Description:Binding affinity to sigma 2 receptor/TMEM97 (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
Affinity DataKi: 100nMAssay Description:Binding affinity to human 5HT2B receptor assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand InfoSimilars
TargetSigma non-opioid intracellular receptor 1(Guinea pig)
The University of Texas At Austin
Curated by ChEMBL
The University of Texas At Austin
Curated by ChEMBL
Affinity DataKi: 104nMAssay Description:Displacement of [3H](+)-pentazocine from sigma 1 receptor in guinea pig brain assessed as inhibition constant by competition binding assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
Affinity DataKi: 128nMAssay Description:Displacement of [3H]-ditolylguanidine from human sigma 2 receptor/TMEM97 transfected in HEK293 cells assessed as inhibition constant in the presence ...More data for this Ligand-Target Pair
Ligand InfoSimilars
Affinity DataKi: 135nMAssay Description:Binding affinity to human 5HT1D receptor assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand InfoSimilars
Affinity DataKi: 135nMAssay Description:Displacement of [3H]-ditolylguanidine from human sigma 2 receptor/TMEM97 transfected in HEK293 cells assessed as inhibition constant in the presence ...More data for this Ligand-Target Pair
Ligand InfoSimilars
TargetSigma non-opioid intracellular receptor 1(Guinea pig)
The University of Texas At Austin
Curated by ChEMBL
The University of Texas At Austin
Curated by ChEMBL
Affinity DataKi: 140nMAssay Description:Displacement of [3H](+)-pentazocine from sigma 1 receptor in guinea pig brain assessed as inhibition constant by competition binding assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
Affinity DataKi: 156nMAssay Description:Binding affinity to human 5HT1A receptor assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand InfoSimilars
TargetSigma non-opioid intracellular receptor 1(Guinea pig)
The University of Texas At Austin
Curated by ChEMBL
The University of Texas At Austin
Curated by ChEMBL
Affinity DataKi: 187nMAssay Description:Displacement of [3H](+)-pentazocine from sigma 1 receptor in guinea pig brain assessed as inhibition constant by competition binding assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
TargetSigma non-opioid intracellular receptor 1(Human)
The University of Texas At Austin
Curated by ChEMBL
The University of Texas At Austin
Curated by ChEMBL
Affinity DataKi: 188nMAssay Description:Displacement of [3H](+)-pentazocine from human sigma 1 receptor transfected in HEK293 cells assessed as inhibition constant by competition binding as...More data for this Ligand-Target Pair
Ligand InfoSimilars
TargetSigma non-opioid intracellular receptor 1(Human)
The University of Texas At Austin
Curated by ChEMBL
The University of Texas At Austin
Curated by ChEMBL
Affinity DataKi: 196nMAssay Description:Displacement of [3H](+)-pentazocine from human sigma 1 receptor transfected in HEK293 cells assessed as inhibition constant by competition binding as...More data for this Ligand-Target Pair
Ligand InfoSimilars
TargetSigma non-opioid intracellular receptor 1(Guinea pig)
The University of Texas At Austin
Curated by ChEMBL
The University of Texas At Austin
Curated by ChEMBL
Affinity DataKi: 199nMAssay Description:Displacement of [3H](+)-pentazocine from sigma 1 receptor in guinea pig brain assessed as inhibition constant by competition binding assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
TargetSigma non-opioid intracellular receptor 1(Guinea pig)
The University of Texas At Austin
Curated by ChEMBL
The University of Texas At Austin
Curated by ChEMBL
Affinity DataKi: 200nMAssay Description:Displacement of [3H](+)-pentazocine from sigma 1 receptor in guinea pig brain assessed as inhibition constant by competition binding assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
TargetSigma non-opioid intracellular receptor 1(Guinea pig)
The University of Texas At Austin
Curated by ChEMBL
The University of Texas At Austin
Curated by ChEMBL
Affinity DataKi: 223nMAssay Description:Displacement of [3H](+)-pentazocine from sigma 1 receptor in guinea pig brain assessed as inhibition constant by competition binding assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
