Compile Data Set for Download or QSAR
Report error Found 95 Enz. Inhib. hit(s) with all data for entry = 50017036
Target5-hydroxytryptamine receptor 2A(Human)
City University of New York

Curated by ChEMBL
LigandPNGBDBM50599264(CHEMBL5204813)
Affinity DataIC50: 137nMAssay Description:Antagonist activity at 5-HT2A receptor (unknown origin) incubated for 60 mins followed by 10 mins incubation in dark at room temperature by FLIPR met...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
Target5-hydroxytryptamine receptor 2C(Human)
City University of New York

Curated by ChEMBL
LigandPNGBDBM50599264(CHEMBL5204813)
Affinity DataIC50: 161nMAssay Description:Antagonist activity at 5-HT2C receptor (unknown origin) incubated for 60 mins followed by 10 mins incubation in dark at room temperature by FLIPR met...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
City University of New York

Curated by ChEMBL
LigandPNGBDBM50599263(CHEMBL5195241)
Affinity DataIC50: 162nMAssay Description:Antagonist activity at 5-HT2A receptor (unknown origin) incubated for 60 mins followed by 10 mins incubation in dark at room temperature by FLIPR met...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
Target5-hydroxytryptamine receptor 2C(Human)
City University of New York

Curated by ChEMBL
LigandPNGBDBM50599263(CHEMBL5195241)
Affinity DataIC50: 436nMAssay Description:Antagonist activity at 5-HT2C receptor (unknown origin) incubated for 60 mins followed by 10 mins incubation in dark at room temperature by FLIPR met...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
Target5-hydroxytryptamine receptor 2B(Human)
City University of New York

Curated by ChEMBL
LigandPNGBDBM50599264(CHEMBL5204813)
Affinity DataIC50: 1.23E+3nMAssay Description:Antagonist activity at 5-HT2B receptor (unknown origin) incubated for 60 mins followed by 10 mins incubation in dark at room temperature by FLIPR met...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
Target5-hydroxytryptamine receptor 2B(Human)
City University of New York

Curated by ChEMBL
LigandPNGBDBM50599263(CHEMBL5195241)
Affinity DataIC50: 3.00E+3nMAssay Description:Antagonist activity at 5-HT2B receptor (unknown origin) incubated for 60 mins followed by 10 mins incubation in dark at room temperature by FLIPR met...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
Target5-hydroxytryptamine receptor 2C(Human)
City University of New York

Curated by ChEMBL
LigandPNGBDBM50001775(cid_5074 | Ritanserine | 6-(2-{4-[Bis-(4-fluoro-ph...)
Affinity DataKi:  0.800nMAssay Description:Displacement of [3H]Mesulergine from 5-HT2C receptor (unknown origin) assessed as inhibition constant incubated for 90 mins by MicroBeta scintillatio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
Target5-hydroxytryptamine receptor 2C(Human)
City University of New York

Curated by ChEMBL
LigandPNGBDBM50599264(CHEMBL5204813)
Affinity DataKi:  4nMAssay Description:Displacement of [3H]Mesulergine from 5-HT2C receptor (unknown origin) assessed as inhibition constant incubated for 90 mins by MicroBeta scintillatio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
Target5-hydroxytryptamine receptor 2B(Human)
City University of New York

Curated by ChEMBL
LigandPNGBDBM50089979(CHEMBL3581250)
Affinity DataKi:  10nMAssay Description:Displacement of [3H]LSD from 5-HT2B receptor (unknown origin) assessed as inhibition constant incubated for 90 mins by MicroBeta scintillation counti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
Target5-hydroxytryptamine receptor 2B(Human)
City University of New York

Curated by ChEMBL
LigandPNGBDBM50599254(CHEMBL5174366)
Affinity DataKi:  15nMAssay Description:Displacement of [3H]LSD from 5-HT2B receptor (unknown origin) assessed as inhibition constant incubated for 90 mins by MicroBeta scintillation counti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
Target5-hydroxytryptamine receptor 2B(Human)
City University of New York

Curated by ChEMBL
LigandPNGBDBM50599252(CHEMBL5180016)
Affinity DataKi:  16nMAssay Description:Displacement of [3H]LSD from 5-HT2B receptor (unknown origin) assessed as inhibition constant incubated for 90 mins by MicroBeta scintillation counti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
City University of New York

Curated by ChEMBL
LigandPNGBDBM50599263(CHEMBL5195241)
Affinity DataKi:  20nMAssay Description:Displacement of [3H]Ketanserin from 5-HT2A receptor (unknown origin) assessed as inhibition constant incubated for 90 mins by MicroBeta scintillation...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
Target5-hydroxytryptamine receptor 2B(Human)
City University of New York

Curated by ChEMBL
LigandPNGBDBM50060417(CHEMBL297784 | SB 206553 | SB-206553 | 5-Methyl-3,...)
Affinity DataKi:  20nMAssay Description:Displacement of [3H]LSD from 5-HT2B receptor (unknown origin) assessed as inhibition constant incubated for 90 mins by MicroBeta scintillation counti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
City University of New York

Curated by ChEMBL
LigandPNGBDBM50599264(CHEMBL5204813)
Affinity DataKi:  22nMAssay Description:Displacement of [3H]Ketanserin from 5-HT2A receptor (unknown origin) assessed as inhibition constant incubated for 90 mins by MicroBeta scintillation...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
Target5-hydroxytryptamine receptor 2B(Human)
City University of New York

Curated by ChEMBL
LigandPNGBDBM50089980(CHEMBL3581249)
Affinity DataKi:  22nMAssay Description:Displacement of [3H]LSD from 5-HT2B receptor (unknown origin) assessed as inhibition constant incubated for 90 mins by MicroBeta scintillation counti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
Target5-hydroxytryptamine receptor 2C(Human)
City University of New York

Curated by ChEMBL
LigandPNGBDBM50599263(CHEMBL5195241)
Affinity DataKi:  23nMAssay Description:Displacement of [3H]Mesulergine from 5-HT2C receptor (unknown origin) assessed as inhibition constant incubated for 90 mins by MicroBeta scintillatio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
City University of New York

Curated by ChEMBL
LigandPNGBDBM50001884(8-Chloro-11-(4-methyl-piperazin-1-yl)-5H-dibenzo[b...)
Affinity DataKi:  24nMAssay Description:Displacement of [3H]Ketanserin from 5-HT2A receptor (unknown origin) assessed as inhibition constant incubated for 90 mins by MicroBeta scintillation...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
Target5-hydroxytryptamine receptor 2B(Human)
City University of New York

Curated by ChEMBL
LigandPNGBDBM50599259(CHEMBL5203303)
Affinity DataKi:  25nMAssay Description:Displacement of [3H]LSD from 5-HT2B receptor (unknown origin) assessed as inhibition constant incubated for 90 mins by MicroBeta scintillation counti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
Target5-hydroxytryptamine receptor 2B(Human)
City University of New York

Curated by ChEMBL
LigandPNGBDBM50089976(CHEMBL3581252)
Affinity DataKi:  29nMAssay Description:Displacement of [3H]LSD from 5-HT2B receptor (unknown origin) assessed as inhibition constant incubated for 90 mins by MicroBeta scintillation counti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
Target5-hydroxytryptamine receptor 2B(Human)
City University of New York

Curated by ChEMBL
LigandPNGBDBM50089977(CHEMBL3581251)
Affinity DataKi:  33nMAssay Description:Displacement of [3H]LSD from 5-HT2B receptor (unknown origin) assessed as inhibition constant incubated for 90 mins by MicroBeta scintillation counti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
Target5-hydroxytryptamine receptor 2C(Human)
City University of New York

Curated by ChEMBL
LigandPNGBDBM50599259(CHEMBL5203303)
Affinity DataKi:  37nMAssay Description:Displacement of [3H]Mesulergine from 5-HT2C receptor (unknown origin) assessed as inhibition constant incubated for 90 mins by MicroBeta scintillatio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
Target5-hydroxytryptamine receptor 2B(Human)
City University of New York

Curated by ChEMBL
LigandPNGBDBM50599261(CHEMBL5185086)
Affinity DataKi:  40nMAssay Description:Displacement of [3H]LSD from 5-HT2B receptor (unknown origin) assessed as inhibition constant incubated for 90 mins by MicroBeta scintillation counti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
Target5-hydroxytryptamine receptor 2C(Human)
City University of New York

Curated by ChEMBL
LigandPNGBDBM50599255(CHEMBL5183799)
Affinity DataKi:  40nMAssay Description:Displacement of [3H]Mesulergine from 5-HT2C receptor (unknown origin) assessed as inhibition constant incubated for 90 mins by MicroBeta scintillatio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
Target5-hydroxytryptamine receptor 2B(Human)
City University of New York

Curated by ChEMBL
LigandPNGBDBM50089972(CHEMBL3581256)
Affinity DataKi:  42nMAssay Description:Displacement of [3H]LSD from 5-HT2B receptor (unknown origin) assessed as inhibition constant incubated for 90 mins by MicroBeta scintillation counti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
Target5-hydroxytryptamine receptor 2B(Human)
City University of New York

Curated by ChEMBL
LigandPNGBDBM50090001(CHEMBL3581248)
Affinity DataKi:  45nMAssay Description:Displacement of [3H]LSD from 5-HT2B receptor (unknown origin) assessed as inhibition constant incubated for 90 mins by MicroBeta scintillation counti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
Target5-hydroxytryptamine receptor 2B(Human)
City University of New York

Curated by ChEMBL
LigandPNGBDBM50599255(CHEMBL5183799)
Affinity DataKi:  47nMAssay Description:Displacement of [3H]LSD from 5-HT2B receptor (unknown origin) assessed as inhibition constant incubated for 90 mins by MicroBeta scintillation counti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
Target5-hydroxytryptamine receptor 2C(Human)
City University of New York

Curated by ChEMBL
LigandPNGBDBM50599254(CHEMBL5174366)
Affinity DataKi:  47nMAssay Description:Displacement of [3H]Mesulergine from 5-HT2C receptor (unknown origin) assessed as inhibition constant incubated for 90 mins by MicroBeta scintillatio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
Target5-hydroxytryptamine receptor 2B(Human)
City University of New York

Curated by ChEMBL
LigandPNGBDBM50090007(CHEMBL3581247)
Affinity DataKi:  48nMAssay Description:Displacement of [3H]LSD from 5-HT2B receptor (unknown origin) assessed as inhibition constant incubated for 90 mins by MicroBeta scintillation counti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
Target5-hydroxytryptamine receptor 2B(Human)
City University of New York

Curated by ChEMBL
LigandPNGBDBM50599264(CHEMBL5204813)
Affinity DataKi:  48nMAssay Description:Displacement of [3H]LSD from 5-HT2B receptor (unknown origin) assessed as inhibition constant incubated for 90 mins by MicroBeta scintillation counti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
Target5-hydroxytryptamine receptor 2C(Human)
City University of New York

Curated by ChEMBL
LigandPNGBDBM50599252(CHEMBL5180016)
Affinity DataKi:  50nMAssay Description:Displacement of [3H]Mesulergine from 5-HT2C receptor (unknown origin) assessed as inhibition constant incubated for 90 mins by MicroBeta scintillatio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
Target5-hydroxytryptamine receptor 2B(Human)
City University of New York

Curated by ChEMBL
LigandPNGBDBM50089975(CHEMBL3581253)
Affinity DataKi:  53nMAssay Description:Displacement of [3H]LSD from 5-HT2B receptor (unknown origin) assessed as inhibition constant incubated for 90 mins by MicroBeta scintillation counti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
Target5-hydroxytryptamine receptor 2B(Human)
City University of New York

Curated by ChEMBL
LigandPNGBDBM50090008(CHEMBL3581246)
Affinity DataKi:  53nMAssay Description:Displacement of [3H]LSD from 5-HT2B receptor (unknown origin) assessed as inhibition constant incubated for 90 mins by MicroBeta scintillation counti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
Target5-hydroxytryptamine receptor 2B(Human)
City University of New York

Curated by ChEMBL
LigandPNGBDBM50089974(CHEMBL3581254)
Affinity DataKi:  55nMAssay Description:Displacement of [3H]LSD from 5-HT2B receptor (unknown origin) assessed as inhibition constant incubated for 90 mins by MicroBeta scintillation counti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
Target5-hydroxytryptamine receptor 2B(Human)
City University of New York

Curated by ChEMBL
LigandPNGBDBM50090078(CHEMBL3581245)
Affinity DataKi:  56nMAssay Description:Displacement of [3H]LSD from 5-HT2B receptor (unknown origin) assessed as inhibition constant incubated for 90 mins by MicroBeta scintillation counti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
Target5-hydroxytryptamine receptor 2B(Human)
City University of New York

Curated by ChEMBL
LigandPNGBDBM50090077(CHEMBL3580670)
Affinity DataKi:  57nMAssay Description:Displacement of [3H]LSD from 5-HT2B receptor (unknown origin) assessed as inhibition constant incubated for 90 mins by MicroBeta scintillation counti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
Target5-hydroxytryptamine receptor 2C(Human)
City University of New York

Curated by ChEMBL
LigandPNGBDBM50599260(CHEMBL5175973)
Affinity DataKi:  72nMAssay Description:Displacement of [3H]Mesulergine from 5-HT2C receptor (unknown origin) assessed as inhibition constant incubated for 90 mins by MicroBeta scintillatio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
Target5-hydroxytryptamine receptor 2B(Human)
City University of New York

Curated by ChEMBL
LigandPNGBDBM50090079(CHEMBL3581244)
Affinity DataKi:  80nMAssay Description:Displacement of [3H]LSD from 5-HT2B receptor (unknown origin) assessed as inhibition constant incubated for 90 mins by MicroBeta scintillation counti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
Target5-hydroxytryptamine receptor 2C(Human)
City University of New York

Curated by ChEMBL
LigandPNGBDBM50599256(CHEMBL5194057)
Affinity DataKi:  82nMAssay Description:Displacement of [3H]Mesulergine from 5-HT2C receptor (unknown origin) assessed as inhibition constant incubated for 90 mins by MicroBeta scintillatio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
Target5-hydroxytryptamine receptor 2B(Human)
City University of New York

Curated by ChEMBL
LigandPNGBDBM50599260(CHEMBL5175973)
Affinity DataKi:  82nMAssay Description:Displacement of [3H]LSD from 5-HT2B receptor (unknown origin) assessed as inhibition constant incubated for 90 mins by MicroBeta scintillation counti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
Target5-hydroxytryptamine receptor 2B(Human)
City University of New York

Curated by ChEMBL
LigandPNGBDBM50599262(CHEMBL5208882)
Affinity DataKi:  92nMAssay Description:Displacement of [3H]LSD from 5-HT2B receptor (unknown origin) assessed as inhibition constant incubated for 90 mins by MicroBeta scintillation counti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
Target5-hydroxytryptamine receptor 2C(Human)
City University of New York

Curated by ChEMBL
LigandPNGBDBM50599258(CHEMBL5188171)
Affinity DataKi:  94nMAssay Description:Displacement of [3H]Mesulergine from 5-HT2C receptor (unknown origin) assessed as inhibition constant incubated for 90 mins by MicroBeta scintillatio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
Target5-hydroxytryptamine receptor 2B(Human)
City University of New York

Curated by ChEMBL
LigandPNGBDBM50599258(CHEMBL5188171)
Affinity DataKi:  96nMAssay Description:Displacement of [3H]LSD from 5-HT2B receptor (unknown origin) assessed as inhibition constant incubated for 90 mins by MicroBeta scintillation counti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
City University of New York

Curated by ChEMBL
LigandPNGBDBM50599252(CHEMBL5180016)
Affinity DataKi:  101nMAssay Description:Displacement of [3H]Ketanserin from 5-HT2A receptor (unknown origin) assessed as inhibition constant incubated for 90 mins by MicroBeta scintillation...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
Target5-hydroxytryptamine receptor 2C(Human)
City University of New York

Curated by ChEMBL
LigandPNGBDBM50599261(CHEMBL5185086)
Affinity DataKi:  104nMAssay Description:Displacement of [3H]Mesulergine from 5-HT2C receptor (unknown origin) assessed as inhibition constant incubated for 90 mins by MicroBeta scintillatio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
Target5-hydroxytryptamine receptor 2B(Human)
City University of New York

Curated by ChEMBL
LigandPNGBDBM50599256(CHEMBL5194057)
Affinity DataKi:  105nMAssay Description:Displacement of [3H]LSD from 5-HT2B receptor (unknown origin) assessed as inhibition constant incubated for 90 mins by MicroBeta scintillation counti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
Target5-hydroxytryptamine receptor 2C(Human)
City University of New York

Curated by ChEMBL
LigandPNGBDBM50599262(CHEMBL5208882)
Affinity DataKi:  113nMAssay Description:Displacement of [3H]Mesulergine from 5-HT2C receptor (unknown origin) assessed as inhibition constant incubated for 90 mins by MicroBeta scintillatio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
Target5-hydroxytryptamine receptor 2B(Human)
City University of New York

Curated by ChEMBL
LigandPNGBDBM50197829(CHEMBL228082 | glaucine fumarate | (S)-1,2,9,10-te...)
Affinity DataKi:  119nMAssay Description:Displacement of [3H]LSD from 5-HT2B receptor (unknown origin) assessed as inhibition constant incubated for 90 mins by MicroBeta scintillation counti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
City University of New York

Curated by ChEMBL
LigandPNGBDBM50599255(CHEMBL5183799)
Affinity DataKi:  138nMAssay Description:Displacement of [3H]Ketanserin from 5-HT2A receptor (unknown origin) assessed as inhibition constant incubated for 90 mins by MicroBeta scintillation...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
Target5-hydroxytryptamine receptor 2B(Human)
City University of New York

Curated by ChEMBL
LigandPNGBDBM50599253(CHEMBL5181312)
Affinity DataKi:  153nMAssay Description:Displacement of [3H]LSD from 5-HT2B receptor (unknown origin) assessed as inhibition constant incubated for 90 mins by MicroBeta scintillation counti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
City University of New York

Curated by ChEMBL
LigandPNGBDBM50599260(CHEMBL5175973)
Affinity DataKi:  155nMAssay Description:Displacement of [3H]Ketanserin from 5-HT2A receptor (unknown origin) assessed as inhibition constant incubated for 90 mins by MicroBeta scintillation...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
Displayed 1 to 50 (of 95 total ) | Next | Last >>
Jump to: