Compile Data Set for Download or QSAR
Report error Found 9 Enz. Inhib. hit(s) with all data for entry = 50016169
TargetExcitatory amino acid transporter 2(Human)
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50592916(CHEMBL5206486)
Affinity DataEC50:  11nMAssay Description:Activation of human EAAT2 transfected in COS7 cells assessed as glutamate uptakeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetExcitatory amino acid transporter 2(Human)
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50592918(CHEMBL5187206)
Affinity DataEC50:  20nMAssay Description:Activation of human EAAT2 transfected in COS7 cells assessed as glutamate uptakeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetExcitatory amino acid transporter 2(Human)
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50592916(CHEMBL5206486)
Affinity DataEC50:  25nMAssay Description:Activation of human EAAT2 transfected in Glial cells assessed as glutamate uptakeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetExcitatory amino acid transporter 2(Human)
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50592918(CHEMBL5187206)
Affinity DataEC50:  0.100nMAssay Description:Activation of human EAAT2 transfected in Glial cells assessed as glutamate uptakeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetAlbumin(Human)
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50592916(CHEMBL5206486)
Affinity DataKd:  1.97E+6nMAssay Description:Binding affinity to human serum albumin assessed as dissociation constant by LC/MS analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetSynaptic vesicle glycoprotein 2A(Human)
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50592916(CHEMBL5206486)
Affinity DataKi: >2.50E+5nMAssay Description:Binding affinity to human SV2A in presence of levetiracetam by radioligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetSynaptic vesicle glycoprotein 2A(Human)
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50592917(CHEMBL5185567)
Affinity DataKi: >2.50E+5nMAssay Description:Binding affinity to human SV2A in presence of levetiracetam by radioligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetSynaptic vesicle glycoprotein 2A(Mouse)
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50592916(CHEMBL5206486)
Affinity DataKi: >2.50E+5nMAssay Description:Binding affinity to mouse SV2A in presence of levetiracetam by radioligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetSynaptic vesicle glycoprotein 2A(Mouse)
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50592917(CHEMBL5185567)
Affinity DataKi: >2.50E+5nMAssay Description:Binding affinity to mouse SV2A in presence of levetiracetam by radioligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed