Compile Data Set for Download or QSAR
Report error Found 9 Enz. Inhib. hit(s) with all data for entry = 50016376
TargetLysophosphatidic acid receptor 2(Human)
Universidad Complutense De Madrid

Curated by ChEMBL
LigandPNGBDBM50594511(CHEMBL5182278)
Affinity DataKd:  1.30nMAssay Description:Binding affinity to LPA2 receptor (unknown origin) by free solution assay-compensated interferometric reader (FSA-CIR) techniqueMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details
PubMed
TargetLysophosphatidic acid receptor 1(Human)
Universidad Complutense De Madrid

Curated by ChEMBL
LigandPNGBDBM50170859(3-(4-(4-((1-(2-chlorophenyl)ethoxy)carbonylamino)-...)
Affinity DataIC50: 800nMAssay Description:Antagonist activity at LPA1 receptor (unknown origin) expressed in cells assessed as blockade of LPA-induced calcium mobilization measured after 120 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details
PubMed
TargetLysophosphatidic acid receptor 2(Human)
Universidad Complutense De Madrid

Curated by ChEMBL
LigandPNGBDBM50170859(3-(4-(4-((1-(2-chlorophenyl)ethoxy)carbonylamino)-...)
Affinity DataIC50: 1.20E+3nMAssay Description:Antagonist activity at LPA2 receptor (unknown origin) expressed in cells assessed as blockade of LPA-induced calcium mobilization measured after 120 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details
PubMed
TargetLysophosphatidic acid receptor 3(Human)
Universidad Complutense De Madrid

Curated by ChEMBL
LigandPNGBDBM50170859(3-(4-(4-((1-(2-chlorophenyl)ethoxy)carbonylamino)-...)
Affinity DataIC50: 1.60E+3nMAssay Description:Antagonist activity at LPA3 receptor (unknown origin) expressed in cells assessed as blockade of LPA-induced calcium mobilization measured after 120 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details
PubMed
TargetLysophosphatidic acid receptor 2(Human)
Universidad Complutense De Madrid

Curated by ChEMBL
LigandPNGBDBM50594511(CHEMBL5182278)
Affinity DataIC50: 1.90E+3nMAssay Description:Antagonist activity at LPA2 receptor (unknown origin) expressed in cells assessed as blockade of LPA-induced calcium mobilization measured after 120 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details
PubMed
TargetLysophosphatidic acid receptor 2(Human)
Universidad Complutense De Madrid

Curated by ChEMBL
LigandPNGBDBM50594510(CHEMBL5183786)
Affinity DataIC50: 5.10E+3nMAssay Description:Antagonist activity at LPA2 receptor (unknown origin) expressed in cells assessed as blockade of LPA-induced calcium mobilization measured after 120 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details
PubMed
TargetLysophosphatidic acid receptor 2(Human)
Universidad Complutense De Madrid

Curated by ChEMBL
LigandPNGBDBM50594508(CHEMBL5184934)
Affinity DataIC50: 5.50E+3nMAssay Description:Antagonist activity at LPA2 receptor (unknown origin) expressed in cells assessed as blockade of LPA-induced calcium mobilization measured after 120 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details
PubMed
TargetLysophosphatidic acid receptor 2(Human)
Universidad Complutense De Madrid

Curated by ChEMBL
LigandPNGBDBM50594509(CHEMBL5178032)
Affinity DataIC50: 1.16E+4nMAssay Description:Antagonist activity at LPA2 receptor (unknown origin) expressed in cells assessed as blockade of LPA-induced calcium mobilization measured after 120 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details
PubMed
TargetLysophosphatidic acid receptor 2(Human)
Universidad Complutense De Madrid

Curated by ChEMBL
LigandPNGBDBM50594512(CHEMBL5191342)
Affinity DataIC50: 3.10E+4nMAssay Description:Antagonist activity at LPA2 receptor (unknown origin) expressed in cells assessed as blockade of LPA-induced calcium mobilization measured after 120 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details
PubMed