Compile Data Set for Download or QSAR
Report error Found 20 Enz. Inhib. hit(s) with all data for entry = 50015921
Target5-hydroxytryptamine receptor 6(Human)
Hec Research and Development Center

Curated by ChEMBL
LigandPNGBDBM394084(US9974785, Example 3)
Affinity DataKi:  0.430nMAssay Description:Displacement of [3H]-LSD from human 5HT6 receptor expressed in CHO cells assessed as inhibition constant incubated for 120 mins by liquid scintillati...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/19/2023
Entry Details
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Hec Research and Development Center

Curated by ChEMBL
LigandPNGBDBM394083(US9974785, Example 2)
Affinity DataKi:  0.460nMAssay Description:Displacement of [3H]-LSD from human 5HT6 receptor expressed in CHO cells assessed as inhibition constant incubated for 120 mins by liquid scintillati...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/19/2023
Entry Details
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Hec Research and Development Center

Curated by ChEMBL
LigandPNGBDBM50590516(CHEMBL5196479)
Affinity DataKi:  0.510nMAssay Description:Displacement of [3H]-LSD from human 5HT6 receptor expressed in CHO cells assessed as inhibition constant incubated for 120 mins by liquid scintillati...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/19/2023
Entry Details
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Hec Research and Development Center

Curated by ChEMBL
LigandPNGBDBM394086(US9974785, Example 5)
Affinity DataKi:  0.520nMAssay Description:Displacement of [3H]-LSD from human 5HT6 receptor expressed in CHO cells assessed as inhibition constant incubated for 120 mins by liquid scintillati...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/19/2023
Entry Details
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Hec Research and Development Center

Curated by ChEMBL
LigandPNGBDBM394087(US9974785, Example 6)
Affinity DataKi:  0.680nMAssay Description:Displacement of [3H]-LSD from human 5HT6 receptor expressed in CHO cells assessed as inhibition constant incubated for 120 mins by liquid scintillati...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/19/2023
Entry Details
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Hec Research and Development Center

Curated by ChEMBL
LigandPNGBDBM50019754(LU-AE58054 | IDALOPIRDINE)
Affinity DataKi:  0.830nMAssay Description:Displacement of [3H]-LSD from human 5HT6 receptor expressed in CHO cells assessed as inhibition constant incubated for 120 mins by liquid scintillati...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/19/2023
Entry Details
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Hec Research and Development Center

Curated by ChEMBL
LigandPNGBDBM394085(US9974785, Example 4)
Affinity DataKi:  1.10nMAssay Description:Displacement of [3H]-LSD from human 5HT6 receptor expressed in CHO cells assessed as inhibition constant incubated for 120 mins by liquid scintillati...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/19/2023
Entry Details
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Hec Research and Development Center

Curated by ChEMBL
LigandPNGBDBM394082(US9974785, Example 1)
Affinity DataKi:  1.60nMAssay Description:Displacement of [3H]-LSD from human 5HT6 receptor expressed in CHO cells assessed as inhibition constant incubated for 120 mins by liquid scintillati...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/19/2023
Entry Details
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Hec Research and Development Center

Curated by ChEMBL
LigandPNGBDBM394088(US9974785, Example 7)
Affinity DataKi:  6.40nMAssay Description:Displacement of [3H]-LSD from human 5HT6 receptor expressed in CHO cells assessed as inhibition constant incubated for 120 mins by liquid scintillati...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/19/2023
Entry Details
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Hec Research and Development Center

Curated by ChEMBL
LigandPNGBDBM394091(US9974785, Example 11)
Affinity DataKi:  11nMAssay Description:Displacement of [3H]-LSD from human 5HT6 receptor expressed in CHO cells assessed as inhibition constant incubated for 120 mins by liquid scintillati...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/19/2023
Entry Details
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Hec Research and Development Center

Curated by ChEMBL
LigandPNGBDBM394089(US9974785, Example 8)
Affinity DataKi:  12nMAssay Description:Displacement of [3H]-LSD from human 5HT6 receptor expressed in CHO cells assessed as inhibition constant incubated for 120 mins by liquid scintillati...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/19/2023
Entry Details
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Hec Research and Development Center

Curated by ChEMBL
LigandPNGBDBM394099(US9974785, Example 19)
Affinity DataKi:  13nMAssay Description:Displacement of [3H]-LSD from human 5HT6 receptor expressed in CHO cells assessed as inhibition constant incubated for 120 mins by liquid scintillati...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/19/2023
Entry Details
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Hec Research and Development Center

Curated by ChEMBL
LigandPNGBDBM394097(US9974785, Example 17)
Affinity DataKi:  13nMAssay Description:Displacement of [3H]-LSD from human 5HT6 receptor expressed in CHO cells assessed as inhibition constant incubated for 120 mins by liquid scintillati...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/19/2023
Entry Details
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Hec Research and Development Center

Curated by ChEMBL
LigandPNGBDBM394093(US9974785, Example 13)
Affinity DataKi:  13nMAssay Description:Displacement of [3H]-LSD from human 5HT6 receptor expressed in CHO cells assessed as inhibition constant incubated for 120 mins by liquid scintillati...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/19/2023
Entry Details
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Hec Research and Development Center

Curated by ChEMBL
LigandPNGBDBM394098(US9974785, Example 18)
Affinity DataKi:  15nMAssay Description:Displacement of [3H]-LSD from human 5HT6 receptor expressed in CHO cells assessed as inhibition constant incubated for 120 mins by liquid scintillati...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/19/2023
Entry Details
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Hec Research and Development Center

Curated by ChEMBL
LigandPNGBDBM394095(US9974785, Example 15)
Affinity DataKi:  17nMAssay Description:Displacement of [3H]-LSD from human 5HT6 receptor expressed in CHO cells assessed as inhibition constant incubated for 120 mins by liquid scintillati...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/19/2023
Entry Details
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Hec Research and Development Center

Curated by ChEMBL
LigandPNGBDBM394094(US9974785, Example 14)
Affinity DataKi:  20nMAssay Description:Displacement of [3H]-LSD from human 5HT6 receptor expressed in CHO cells assessed as inhibition constant incubated for 120 mins by liquid scintillati...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/19/2023
Entry Details
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Hec Research and Development Center

Curated by ChEMBL
LigandPNGBDBM394092(US9974785, Example 12)
Affinity DataKi:  30nMAssay Description:Displacement of [3H]-LSD from human 5HT6 receptor expressed in CHO cells assessed as inhibition constant incubated for 120 mins by liquid scintillati...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/19/2023
Entry Details
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Hec Research and Development Center

Curated by ChEMBL
LigandPNGBDBM394100(US9974785, Example 20)
Affinity DataKi:  44nMAssay Description:Displacement of [3H]-LSD from human 5HT6 receptor expressed in CHO cells assessed as inhibition constant incubated for 120 mins by liquid scintillati...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/19/2023
Entry Details
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Hec Research and Development Center

Curated by ChEMBL
LigandPNGBDBM394096(US9974785, Example 16)
Affinity DataKi:  67nMAssay Description:Displacement of [3H]-LSD from human 5HT6 receptor expressed in CHO cells assessed as inhibition constant incubated for 120 mins by liquid scintillati...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/19/2023
Entry Details
PubMed