Compile Data Set for Download or QSAR
Report error Found 18 Enz. Inhib. hit(s) with all data for entry = 50015753
TargetIntegrin alpha-V/beta-3(Human)
Hefei Normal University

Curated by ChEMBL
LigandPNGBDBM50235980(CHEMBL429876 | EMD-121974 | cyclo(Arg-Gly-Asp-D-Ph...)
Affinity DataIC50: 110nMAssay Description:Inhibition of alphavbeta3 integrin receptor-mediated cell adhesion to fibrinogen in human HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/18/2023
Entry Details
PubMed
TargetIntegrin alpha-5/beta-1(Human)
Hefei Normal University

Curated by ChEMBL
LigandPNGBDBM50589355(CHEMBL5175534)
Affinity DataIC50: 154nMAssay Description:Inhibition of alpha5beta1 integrin receptor expressed on human surface of adipose tissue-derived stem cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/18/2023
Entry Details
PubMed
TargetIntegrin alpha-5/beta-1(Human)
Hefei Normal University

Curated by ChEMBL
LigandPNGBDBM50589354(CHEMBL5208467)
Affinity DataIC50: 154nMAssay Description:Inhibition of alpha5beta1 integrin receptor expressed on human surface of adipose tissue-derived stem cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/18/2023
Entry Details
PubMed
TargetIntegrin alpha-5/beta-1(Human)
Hefei Normal University

Curated by ChEMBL
LigandPNGBDBM50589353(CHEMBL5203975)
Affinity DataIC50: 154nMAssay Description:Inhibition of alpha5beta1 integrin receptor expressed on human surface of adipose tissue-derived stem cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/18/2023
Entry Details
PubMed
TargetIntegrin alpha-V/beta-3(Human)
Hefei Normal University

Curated by ChEMBL
LigandPNGBDBM50589354(CHEMBL5208467)
Affinity DataIC50: 200nMAssay Description:Inhibition of alphavbeta3 integrin receptor-mediated cell adhesion to fibrinogen in human HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/18/2023
Entry Details
PubMed
TargetIntegrin alpha-V/beta-3(Human)
Hefei Normal University

Curated by ChEMBL
LigandPNGBDBM50235980(CHEMBL429876 | EMD-121974 | cyclo(Arg-Gly-Asp-D-Ph...)
Affinity DataIC50: 220nMAssay Description:Inhibition of alphavbeta3 integrin receptor-mediated cell adhesion to fibrinogen in human SK-OV-3 cells expressing alphavbeta5 integrin receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/18/2023
Entry Details
PubMed
TargetIntegrin alpha-V/beta-5(Human)
Hefei Normal University

Curated by ChEMBL
LigandPNGBDBM50235980(CHEMBL429876 | EMD-121974 | cyclo(Arg-Gly-Asp-D-Ph...)
Affinity DataIC50: 350nMAssay Description:Inhibition of alphavbeta5 integrin receptor-mediated cell adhesion to vitronectin in human HT-29 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/18/2023
Entry Details
PubMed
TargetIntegrin alpha-IIb/beta-3(Human)
Hefei Normal University

Curated by ChEMBL
LigandPNGBDBM50589355(CHEMBL5175534)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of alpha2bbeta3 integrin receptor expressed on human surface of plateletsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/18/2023
Entry Details
PubMed
TargetIntegrin alpha-IIb/beta-3(Human)
Hefei Normal University

Curated by ChEMBL
LigandPNGBDBM50589354(CHEMBL5208467)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of alpha2bbeta3 integrin receptor expressed on human surface of plateletsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/18/2023
Entry Details
PubMed
TargetIntegrin alpha-IIb/beta-3(Human)
Hefei Normal University

Curated by ChEMBL
LigandPNGBDBM50589353(CHEMBL5203975)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of alpha2bbeta3 integrin receptor expressed on human surface of plateletsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/18/2023
Entry Details
PubMed
TargetIntegrin alpha-V/beta-3(Human)
Hefei Normal University

Curated by ChEMBL
LigandPNGBDBM50589353(CHEMBL5203975)
Affinity DataIC50: 1.54E+3nMAssay Description:Inhibition of alphavbeta3 integrin receptor-mediated cell adhesion to fibrinogen in human HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/18/2023
Entry Details
PubMed
TargetIntegrin alpha-V/beta-3(Human)
Hefei Normal University

Curated by ChEMBL
LigandPNGBDBM50589355(CHEMBL5175534)
Affinity DataIC50: 8.43E+3nMAssay Description:Inhibition of alphavbeta3 integrin receptor-mediated cell adhesion to fibrinogen in human HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/18/2023
Entry Details
PubMed
TargetIntegrin alpha-V/beta-3(Human)
Hefei Normal University

Curated by ChEMBL
LigandPNGBDBM50589354(CHEMBL5208467)
Affinity DataIC50: 2.51E+4nMAssay Description:Inhibition of alphavbeta3 integrin receptor-mediated cell adhesion to fibrinogen in human SK-OV-3 cells expressing alphavbeta5 integrin receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/18/2023
Entry Details
PubMed
TargetIntegrin alpha-V/beta-5(Human)
Hefei Normal University

Curated by ChEMBL
LigandPNGBDBM50589354(CHEMBL5208467)
Affinity DataIC50: 3.02E+4nMAssay Description:Inhibition of alphavbeta5 integrin receptor-mediated cell adhesion to vitronectin in human HT-29 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/18/2023
Entry Details
PubMed
TargetIntegrin alpha-V/beta-3(Human)
Hefei Normal University

Curated by ChEMBL
LigandPNGBDBM50589353(CHEMBL5203975)
Affinity DataIC50: 3.02E+4nMAssay Description:Inhibition of alphavbeta3 integrin receptor-mediated cell adhesion to fibrinogen in human SK-OV-3 cells expressing alphavbeta5 integrin receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/18/2023
Entry Details
PubMed
TargetIntegrin alpha-V/beta-3(Human)
Hefei Normal University

Curated by ChEMBL
LigandPNGBDBM50589355(CHEMBL5175534)
Affinity DataIC50: 3.40E+4nMAssay Description:Inhibition of alphavbeta3 integrin receptor-mediated cell adhesion to fibrinogen in human SK-OV-3 cells expressing alphavbeta5 integrin receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/18/2023
Entry Details
PubMed
TargetIntegrin alpha-V/beta-5(Human)
Hefei Normal University

Curated by ChEMBL
LigandPNGBDBM50589353(CHEMBL5203975)
Affinity DataIC50: 6.00E+4nMAssay Description:Inhibition of alphavbeta5 integrin receptor-mediated cell adhesion to vitronectin in human HT-29 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/18/2023
Entry Details
PubMed
TargetIntegrin alpha-V/beta-5(Human)
Hefei Normal University

Curated by ChEMBL
LigandPNGBDBM50589355(CHEMBL5175534)
Affinity DataIC50: 2.08E+5nMAssay Description:Inhibition of alphavbeta5 integrin receptor-mediated cell adhesion to vitronectin in human HT-29 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/18/2023
Entry Details
PubMed