Report error Found 60 Enz. Inhib. hit(s) with all data for entry = 50016941
TargetEpidermal growth factor receptor(Human)
College of Pharmacy of Liaoning University
Curated by ChEMBL
College of Pharmacy of Liaoning University
Curated by ChEMBL
Affinity DataIC50: 0.5nMAssay Description:Inhibition of EGFR L858R/T790M mutant (unknown origin) by mobility shift assayMore data for this Ligand-Target Pair
TargetEpidermal growth factor receptor(Human)
College of Pharmacy of Liaoning University
Curated by ChEMBL
College of Pharmacy of Liaoning University
Curated by ChEMBL
Affinity DataIC50: 5nMAssay Description:Inhibition of wild type EGFR (unknown origin) by mobility shift assayMore data for this Ligand-Target Pair
TargetEpidermal growth factor receptor(Human)
College of Pharmacy of Liaoning University
Curated by ChEMBL
College of Pharmacy of Liaoning University
Curated by ChEMBL
Affinity DataIC50: 10nMAssay Description:Inhibition of EGFR L858R/T790M mutant (unknown origin) by mobility shift assayMore data for this Ligand-Target Pair
TargetEpidermal growth factor receptor(Human)
College of Pharmacy of Liaoning University
Curated by ChEMBL
College of Pharmacy of Liaoning University
Curated by ChEMBL
Affinity DataIC50: 17nMAssay Description:Inhibition of EGFR L858R/T790M mutant (unknown origin) by mobility shift assayMore data for this Ligand-Target Pair
TargetEpidermal growth factor receptor(Human)
College of Pharmacy of Liaoning University
Curated by ChEMBL
College of Pharmacy of Liaoning University
Curated by ChEMBL
Affinity DataIC50: 29nMAssay Description:Inhibition of wild type EGFR (unknown origin) by mobility shift assayMore data for this Ligand-Target Pair
TargetEpidermal growth factor receptor(Human)
College of Pharmacy of Liaoning University
Curated by ChEMBL
College of Pharmacy of Liaoning University
Curated by ChEMBL
Affinity DataIC50: 30nMAssay Description:Inhibition of EGFR L858R/T790M mutant (unknown origin) by mobility shift assayMore data for this Ligand-Target Pair
TargetEpidermal growth factor receptor(Human)
College of Pharmacy of Liaoning University
Curated by ChEMBL
College of Pharmacy of Liaoning University
Curated by ChEMBL
Affinity DataIC50: 41nMAssay Description:Inhibition of EGFR L858R/T790M mutant (unknown origin) by mobility shift assayMore data for this Ligand-Target Pair
TargetEpidermal growth factor receptor(Human)
College of Pharmacy of Liaoning University
Curated by ChEMBL
College of Pharmacy of Liaoning University
Curated by ChEMBL
Affinity DataIC50: 42nMAssay Description:Inhibition of EGFR L858R/T790M mutant (unknown origin) by mobility shift assayMore data for this Ligand-Target Pair
TargetEpidermal growth factor receptor(Human)
College of Pharmacy of Liaoning University
Curated by ChEMBL
College of Pharmacy of Liaoning University
Curated by ChEMBL
Affinity DataIC50: 87nMAssay Description:Inhibition of EGFR L858R/T790M mutant (unknown origin) by mobility shift assayMore data for this Ligand-Target Pair
TargetEpidermal growth factor receptor(Human)
College of Pharmacy of Liaoning University
Curated by ChEMBL
College of Pharmacy of Liaoning University
Curated by ChEMBL
Affinity DataIC50: 100nMAssay Description:Inhibition of EGFR L858R/T790M mutant (unknown origin) by mobility shift assayMore data for this Ligand-Target Pair
TargetEpidermal growth factor receptor(Human)
College of Pharmacy of Liaoning University
Curated by ChEMBL
College of Pharmacy of Liaoning University
Curated by ChEMBL
Affinity DataIC50: 110nMAssay Description:Inhibition of EGFR L858R/T790M mutant (unknown origin) by mobility shift assayMore data for this Ligand-Target Pair
TargetEpidermal growth factor receptor(Human)
College of Pharmacy of Liaoning University
Curated by ChEMBL
College of Pharmacy of Liaoning University
Curated by ChEMBL
Affinity DataIC50: 137nMAssay Description:Inhibition of EGFR L858R/T790M/C797S mutant (unknown origin) by mobility shift assayMore data for this Ligand-Target Pair
TargetEpidermal growth factor receptor(Human)
College of Pharmacy of Liaoning University
Curated by ChEMBL
College of Pharmacy of Liaoning University
Curated by ChEMBL
Affinity DataIC50: 146nMAssay Description:Inhibition of wild type EGFR (unknown origin) by mobility shift assayMore data for this Ligand-Target Pair
TargetEpidermal growth factor receptor(Human)
College of Pharmacy of Liaoning University
Curated by ChEMBL
College of Pharmacy of Liaoning University
Curated by ChEMBL
Affinity DataIC50: 161nMAssay Description:Inhibition of EGFR L858R/T790M/C797S mutant (unknown origin) by mobility shift assayMore data for this Ligand-Target Pair
TargetEpidermal growth factor receptor(Human)
College of Pharmacy of Liaoning University
Curated by ChEMBL
College of Pharmacy of Liaoning University
Curated by ChEMBL
Affinity DataIC50: 224nMAssay Description:Inhibition of wild type EGFR (unknown origin) by mobility shift assayMore data for this Ligand-Target Pair
TargetEpidermal growth factor receptor(Human)
College of Pharmacy of Liaoning University
Curated by ChEMBL
College of Pharmacy of Liaoning University
Curated by ChEMBL
Affinity DataIC50: 242nMAssay Description:Inhibition of EGFR L858R/T790M/C797S mutant (unknown origin) by mobility shift assayMore data for this Ligand-Target Pair
TargetEpidermal growth factor receptor(Human)
College of Pharmacy of Liaoning University
Curated by ChEMBL
College of Pharmacy of Liaoning University
Curated by ChEMBL
Affinity DataIC50: 360nMAssay Description:Inhibition of EGFR L858R/T790M mutant (unknown origin) by mobility shift assayMore data for this Ligand-Target Pair
TargetEpidermal growth factor receptor(Human)
College of Pharmacy of Liaoning University
Curated by ChEMBL
College of Pharmacy of Liaoning University
Curated by ChEMBL
Affinity DataIC50: 360nMAssay Description:Inhibition of wild type EGFR (unknown origin) by mobility shift assayMore data for this Ligand-Target Pair
TargetEpidermal growth factor receptor(Human)
College of Pharmacy of Liaoning University
Curated by ChEMBL
College of Pharmacy of Liaoning University
Curated by ChEMBL
Affinity DataIC50: 391nMAssay Description:Inhibition of EGFR L858R/T790M mutant (unknown origin) by mobility shift assayMore data for this Ligand-Target Pair
TargetEpidermal growth factor receptor(Human)
College of Pharmacy of Liaoning University
Curated by ChEMBL
College of Pharmacy of Liaoning University
Curated by ChEMBL
Affinity DataIC50: 410nMAssay Description:Inhibition of EGFR L858R/T790M/C797S mutant (unknown origin) by mobility shift assayMore data for this Ligand-Target Pair
TargetEpidermal growth factor receptor(Human)
College of Pharmacy of Liaoning University
Curated by ChEMBL
College of Pharmacy of Liaoning University
Curated by ChEMBL
Affinity DataIC50: 420nMAssay Description:Inhibition of EGFR L858R/T790M mutant (unknown origin) by mobility shift assayMore data for this Ligand-Target Pair
TargetEpidermal growth factor receptor(Human)
College of Pharmacy of Liaoning University
Curated by ChEMBL
College of Pharmacy of Liaoning University
Curated by ChEMBL
Affinity DataIC50: 420nMAssay Description:Inhibition of EGFR L858R/T790M/C797S mutant (unknown origin) by mobility shift assayMore data for this Ligand-Target Pair
TargetEpidermal growth factor receptor(Human)
College of Pharmacy of Liaoning University
Curated by ChEMBL
College of Pharmacy of Liaoning University
Curated by ChEMBL
Affinity DataIC50: 500nMAssay Description:Inhibition of EGFR L858R/T790M/C797S mutant (unknown origin) by mobility shift assayMore data for this Ligand-Target Pair
TargetEpidermal growth factor receptor(Human)
College of Pharmacy of Liaoning University
Curated by ChEMBL
College of Pharmacy of Liaoning University
Curated by ChEMBL
Affinity DataIC50: 500nMAssay Description:Inhibition of EGFR L858R/T790M/C797S mutant (unknown origin) by mobility shift assayMore data for this Ligand-Target Pair
TargetEpidermal growth factor receptor(Human)
College of Pharmacy of Liaoning University
Curated by ChEMBL
College of Pharmacy of Liaoning University
Curated by ChEMBL
Affinity DataIC50: 500nMAssay Description:Inhibition of EGFR L858R/T790M/C797S mutant (unknown origin) by mobility shift assayMore data for this Ligand-Target Pair
TargetEpidermal growth factor receptor(Human)
College of Pharmacy of Liaoning University
Curated by ChEMBL
College of Pharmacy of Liaoning University
Curated by ChEMBL
Affinity DataIC50: 500nMAssay Description:Inhibition of EGFR L858R/T790M/C797S mutant (unknown origin) by mobility shift assayMore data for this Ligand-Target Pair
TargetEpidermal growth factor receptor(Human)
College of Pharmacy of Liaoning University
Curated by ChEMBL
College of Pharmacy of Liaoning University
Curated by ChEMBL
Affinity DataIC50: 500nMAssay Description:Inhibition of EGFR L858R/T790M/C797S mutant (unknown origin) by mobility shift assayMore data for this Ligand-Target Pair
TargetEpidermal growth factor receptor(Human)
College of Pharmacy of Liaoning University
Curated by ChEMBL
College of Pharmacy of Liaoning University
Curated by ChEMBL
Affinity DataIC50: 500nMAssay Description:Inhibition of EGFR L858R/T790M/C797S mutant (unknown origin) by mobility shift assayMore data for this Ligand-Target Pair
TargetEpidermal growth factor receptor(Human)
College of Pharmacy of Liaoning University
Curated by ChEMBL
College of Pharmacy of Liaoning University
Curated by ChEMBL
Affinity DataIC50: 500nMAssay Description:Inhibition of EGFR L858R/T790M/C797S mutant (unknown origin) by mobility shift assayMore data for this Ligand-Target Pair
TargetEpidermal growth factor receptor(Human)
College of Pharmacy of Liaoning University
Curated by ChEMBL
College of Pharmacy of Liaoning University
Curated by ChEMBL
Affinity DataIC50: 500nMAssay Description:Inhibition of EGFR L858R/T790M/C797S mutant (unknown origin) by mobility shift assayMore data for this Ligand-Target Pair
TargetEpidermal growth factor receptor(Human)
College of Pharmacy of Liaoning University
Curated by ChEMBL
College of Pharmacy of Liaoning University
Curated by ChEMBL
Affinity DataIC50: 500nMAssay Description:Inhibition of EGFR L858R/T790M/C797S mutant (unknown origin) by mobility shift assayMore data for this Ligand-Target Pair
TargetEpidermal growth factor receptor(Human)
College of Pharmacy of Liaoning University
Curated by ChEMBL
College of Pharmacy of Liaoning University
Curated by ChEMBL
Affinity DataIC50: 500nMAssay Description:Inhibition of wild type EGFR (unknown origin) by mobility shift assayMore data for this Ligand-Target Pair
TargetEpidermal growth factor receptor(Human)
College of Pharmacy of Liaoning University
Curated by ChEMBL
College of Pharmacy of Liaoning University
Curated by ChEMBL
Affinity DataIC50: 500nMAssay Description:Inhibition of EGFR L858R/T790M mutant (unknown origin) by mobility shift assayMore data for this Ligand-Target Pair
TargetEpidermal growth factor receptor(Human)
College of Pharmacy of Liaoning University
Curated by ChEMBL
College of Pharmacy of Liaoning University
Curated by ChEMBL
Affinity DataIC50: 500nMAssay Description:Inhibition of EGFR L858R/T790M/C797S mutant (unknown origin) by mobility shift assayMore data for this Ligand-Target Pair
TargetEpidermal growth factor receptor(Human)
College of Pharmacy of Liaoning University
Curated by ChEMBL
College of Pharmacy of Liaoning University
Curated by ChEMBL
Affinity DataIC50: 500nMAssay Description:Inhibition of wild type EGFR (unknown origin) by mobility shift assayMore data for this Ligand-Target Pair
TargetEpidermal growth factor receptor(Human)
College of Pharmacy of Liaoning University
Curated by ChEMBL
College of Pharmacy of Liaoning University
Curated by ChEMBL
Affinity DataIC50: 500nMAssay Description:Inhibition of wild type EGFR (unknown origin) by mobility shift assayMore data for this Ligand-Target Pair
TargetEpidermal growth factor receptor(Human)
College of Pharmacy of Liaoning University
Curated by ChEMBL
College of Pharmacy of Liaoning University
Curated by ChEMBL
Affinity DataIC50: 500nMAssay Description:Inhibition of wild type EGFR (unknown origin) by mobility shift assayMore data for this Ligand-Target Pair
TargetEpidermal growth factor receptor(Human)
College of Pharmacy of Liaoning University
Curated by ChEMBL
College of Pharmacy of Liaoning University
Curated by ChEMBL
Affinity DataIC50: 500nMAssay Description:Inhibition of wild type EGFR (unknown origin) by mobility shift assayMore data for this Ligand-Target Pair
TargetEpidermal growth factor receptor(Human)
College of Pharmacy of Liaoning University
Curated by ChEMBL
College of Pharmacy of Liaoning University
Curated by ChEMBL
Affinity DataIC50: 500nMAssay Description:Inhibition of wild type EGFR (unknown origin) by mobility shift assayMore data for this Ligand-Target Pair
TargetEpidermal growth factor receptor(Human)
College of Pharmacy of Liaoning University
Curated by ChEMBL
College of Pharmacy of Liaoning University
Curated by ChEMBL
Affinity DataIC50: 500nMAssay Description:Inhibition of wild type EGFR (unknown origin) by mobility shift assayMore data for this Ligand-Target Pair
TargetEpidermal growth factor receptor(Human)
College of Pharmacy of Liaoning University
Curated by ChEMBL
College of Pharmacy of Liaoning University
Curated by ChEMBL
Affinity DataIC50: 500nMAssay Description:Inhibition of wild type EGFR (unknown origin) by mobility shift assayMore data for this Ligand-Target Pair
TargetEpidermal growth factor receptor(Human)
College of Pharmacy of Liaoning University
Curated by ChEMBL
College of Pharmacy of Liaoning University
Curated by ChEMBL
Affinity DataIC50: 500nMAssay Description:Inhibition of EGFR L858R/T790M mutant (unknown origin) by mobility shift assayMore data for this Ligand-Target Pair
TargetEpidermal growth factor receptor(Human)
College of Pharmacy of Liaoning University
Curated by ChEMBL
College of Pharmacy of Liaoning University
Curated by ChEMBL
Affinity DataIC50: 500nMAssay Description:Inhibition of EGFR L858R/T790M mutant (unknown origin) by mobility shift assayMore data for this Ligand-Target Pair
TargetEpidermal growth factor receptor(Human)
College of Pharmacy of Liaoning University
Curated by ChEMBL
College of Pharmacy of Liaoning University
Curated by ChEMBL
Affinity DataIC50: 590nMAssay Description:Inhibition of wild type EGFR (unknown origin) by mobility shift assayMore data for this Ligand-Target Pair
TargetEpidermal growth factor receptor(Human)
College of Pharmacy of Liaoning University
Curated by ChEMBL
College of Pharmacy of Liaoning University
Curated by ChEMBL
Affinity DataIC50: 743nMAssay Description:Inhibition of wild type EGFR (unknown origin) by mobility shift assayMore data for this Ligand-Target Pair
TargetHepatocyte growth factor receptor(Human)
College of Pharmacy of Liaoning University
Curated by ChEMBL
College of Pharmacy of Liaoning University
Curated by ChEMBL
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of c-Met (unknown origin) by mobility shift assayMore data for this Ligand-Target Pair
TargetHepatocyte growth factor receptor(Human)
College of Pharmacy of Liaoning University
Curated by ChEMBL
College of Pharmacy of Liaoning University
Curated by ChEMBL
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of c-Met (unknown origin) by mobility shift assayMore data for this Ligand-Target Pair
TargetHepatocyte growth factor receptor(Human)
College of Pharmacy of Liaoning University
Curated by ChEMBL
College of Pharmacy of Liaoning University
Curated by ChEMBL
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of c-Met (unknown origin) by mobility shift assayMore data for this Ligand-Target Pair
TargetHepatocyte growth factor receptor(Human)
College of Pharmacy of Liaoning University
Curated by ChEMBL
College of Pharmacy of Liaoning University
Curated by ChEMBL
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of c-Met (unknown origin) by mobility shift assayMore data for this Ligand-Target Pair
TargetHepatocyte growth factor receptor(Human)
College of Pharmacy of Liaoning University
Curated by ChEMBL
College of Pharmacy of Liaoning University
Curated by ChEMBL
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of c-Met (unknown origin) by mobility shift assayMore data for this Ligand-Target Pair
