Compile Data Set for Download or QSAR
Report error Found 29 Enz. Inhib. hit(s) with all data for entry = 50016484
TargetVascular endothelial growth factor receptor 2(Human)
University of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50595295(CHEMBL5170855)
Affinity DataIC50: 1.40E+5nMAssay Description:Inhibition of VEGFR2 (unknown origin) using poly[Glu:Tyr] (4:1) as substrate incubated for 45 mins by kinase-glo max reagent based luminescence analy...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details
PubMed
TargetCarbonic anhydrase 12(Human)
University of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50595293(CHEMBL5208376)
Affinity DataKi:  3.80E+3nMAssay Description:Inhibition of recombinant human carbonic anhydrase 12 assessed as inhibition constant incubated for 1 hr prior to testing by phenol red based stopped...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details
PubMed
TargetCarbonic anhydrase 9(Human)
University of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50595293(CHEMBL5208376)
Affinity DataKi:  3.80E+3nMAssay Description:Inhibition of recombinant human carbonic anhydrase 9 assessed as inhibition constant incubated for 1 hr prior to testing by phenol red based stopped-...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details
PubMed
TargetCarbonic anhydrase 12(Human)
University of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM10880(Acetazolamide, AAZ | AZA2 | CHEMBL20 | Acetazolami...)
Affinity DataKi:  5.70E+3nMAssay Description:Inhibition of recombinant human carbonic anhydrase 12 assessed as inhibition constant incubated for 1 hr prior to testing by phenol red based stopped...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetCarbonic anhydrase 9(Human)
University of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM10880(Acetazolamide, AAZ | AZA2 | CHEMBL20 | Acetazolami...)
Affinity DataKi:  5.70E+3nMAssay Description:Inhibition of recombinant human carbonic anhydrase 9 assessed as inhibition constant incubated for 1 hr prior to testing by phenol red based stopped-...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details
PubMed
TargetCarbonic anhydrase 2(Human)
University of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50595293(CHEMBL5208376)
Affinity DataKi:  8.80E+3nMAssay Description:Inhibition of recombinant human carbonic anhydrase 2 assessed as inhibition constant incubated for 1 hr prior to testing by phenol red based stopped-...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details
PubMed
TargetCarbonic anhydrase 2(Human)
University of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM10880(Acetazolamide, AAZ | AZA2 | CHEMBL20 | Acetazolami...)
Affinity DataKi:  1.25E+4nMAssay Description:Inhibition of recombinant human carbonic anhydrase 2 assessed as inhibition constant incubated for 1 hr prior to testing by phenol red based stopped-...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetCarbonic anhydrase 1(Human)
University of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50595293(CHEMBL5208376)
Affinity DataKi:  5.01E+4nMAssay Description:Inhibition of recombinant human carbonic anhydrase 1 assessed as inhibition constant incubated for 1 hr prior to testing by phenol red based stopped-...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details
PubMed
TargetCarbonic anhydrase 9(Human)
University of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50595289(CHEMBL5190054)
Affinity DataKi: >1.00E+5nMAssay Description:Inhibition of recombinant human carbonic anhydrase 9 assessed as inhibition constant incubated for 1 hr prior to testing by phenol red based stopped-...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details
PubMed
TargetCarbonic anhydrase 12(Human)
University of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50595294(CHEMBL5177027)
Affinity DataKi: >1.00E+5nMAssay Description:Inhibition of recombinant human carbonic anhydrase 12 assessed as inhibition constant incubated for 1 hr prior to testing by phenol red based stopped...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details
PubMed
TargetCarbonic anhydrase 12(Human)
University of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50595292(CHEMBL5171643)
Affinity DataKi: >1.00E+5nMAssay Description:Inhibition of recombinant human carbonic anhydrase 12 assessed as inhibition constant incubated for 1 hr prior to testing by phenol red based stopped...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details
PubMed
TargetCarbonic anhydrase 12(Human)
University of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50595291(CHEMBL5207251)
Affinity DataKi: >1.00E+5nMAssay Description:Inhibition of recombinant human carbonic anhydrase 12 assessed as inhibition constant incubated for 1 hr prior to testing by phenol red based stopped...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details
PubMed
TargetCarbonic anhydrase 12(Human)
University of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50595290(CHEMBL5185728)
Affinity DataKi: >1.00E+5nMAssay Description:Inhibition of recombinant human carbonic anhydrase 12 assessed as inhibition constant incubated for 1 hr prior to testing by phenol red based stopped...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details
PubMed
TargetCarbonic anhydrase 12(Human)
University of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50595289(CHEMBL5190054)
Affinity DataKi: >1.00E+5nMAssay Description:Inhibition of recombinant human carbonic anhydrase 12 assessed as inhibition constant incubated for 1 hr prior to testing by phenol red based stopped...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details
PubMed
TargetCarbonic anhydrase 9(Human)
University of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50595294(CHEMBL5177027)
Affinity DataKi: >1.00E+5nMAssay Description:Inhibition of recombinant human carbonic anhydrase 9 assessed as inhibition constant incubated for 1 hr prior to testing by phenol red based stopped-...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details
PubMed
TargetCarbonic anhydrase 9(Human)
University of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50595292(CHEMBL5171643)
Affinity DataKi: >1.00E+5nMAssay Description:Inhibition of recombinant human carbonic anhydrase 9 assessed as inhibition constant incubated for 1 hr prior to testing by phenol red based stopped-...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details
PubMed
TargetCarbonic anhydrase 9(Human)
University of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50595291(CHEMBL5207251)
Affinity DataKi: >1.00E+5nMAssay Description:Inhibition of recombinant human carbonic anhydrase 9 assessed as inhibition constant incubated for 1 hr prior to testing by phenol red based stopped-...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details
PubMed
TargetCarbonic anhydrase 9(Human)
University of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50595290(CHEMBL5185728)
Affinity DataKi: >1.00E+5nMAssay Description:Inhibition of recombinant human carbonic anhydrase 9 assessed as inhibition constant incubated for 1 hr prior to testing by phenol red based stopped-...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details
PubMed
TargetCarbonic anhydrase 1(Human)
University of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50595289(CHEMBL5190054)
Affinity DataKi: >1.00E+5nMAssay Description:Inhibition of recombinant human carbonic anhydrase 1 assessed as inhibition constant incubated for 1 hr prior to testing by phenol red based stopped-...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details
PubMed
TargetCarbonic anhydrase 2(Human)
University of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50595294(CHEMBL5177027)
Affinity DataKi: >1.00E+5nMAssay Description:Inhibition of recombinant human carbonic anhydrase 2 assessed as inhibition constant incubated for 1 hr prior to testing by phenol red based stopped-...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details
PubMed
TargetCarbonic anhydrase 2(Human)
University of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50595292(CHEMBL5171643)
Affinity DataKi: >1.00E+5nMAssay Description:Inhibition of recombinant human carbonic anhydrase 2 assessed as inhibition constant incubated for 1 hr prior to testing by phenol red based stopped-...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details
PubMed
TargetCarbonic anhydrase 2(Human)
University of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50595291(CHEMBL5207251)
Affinity DataKi: >1.00E+5nMAssay Description:Inhibition of recombinant human carbonic anhydrase 2 assessed as inhibition constant incubated for 1 hr prior to testing by phenol red based stopped-...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details
PubMed
TargetCarbonic anhydrase 2(Human)
University of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50595290(CHEMBL5185728)
Affinity DataKi: >1.00E+5nMAssay Description:Inhibition of recombinant human carbonic anhydrase 2 assessed as inhibition constant incubated for 1 hr prior to testing by phenol red based stopped-...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details
PubMed
TargetCarbonic anhydrase 2(Human)
University of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50595289(CHEMBL5190054)
Affinity DataKi: >1.00E+5nMAssay Description:Inhibition of recombinant human carbonic anhydrase 2 assessed as inhibition constant incubated for 1 hr prior to testing by phenol red based stopped-...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details
PubMed
TargetCarbonic anhydrase 1(Human)
University of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50595294(CHEMBL5177027)
Affinity DataKi: >1.00E+5nMAssay Description:Inhibition of recombinant human carbonic anhydrase 1 assessed as inhibition constant incubated for 1 hr prior to testing by phenol red based stopped-...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details
PubMed
TargetCarbonic anhydrase 1(Human)
University of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50595292(CHEMBL5171643)
Affinity DataKi: >1.00E+5nMAssay Description:Inhibition of recombinant human carbonic anhydrase 1 assessed as inhibition constant incubated for 1 hr prior to testing by phenol red based stopped-...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details
PubMed
TargetCarbonic anhydrase 1(Human)
University of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50595291(CHEMBL5207251)
Affinity DataKi: >1.00E+5nMAssay Description:Inhibition of recombinant human carbonic anhydrase 1 assessed as inhibition constant incubated for 1 hr prior to testing by phenol red based stopped-...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details
PubMed
TargetCarbonic anhydrase 1(Human)
University of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50595290(CHEMBL5185728)
Affinity DataKi: >1.00E+5nMAssay Description:Inhibition of recombinant human carbonic anhydrase 1 assessed as inhibition constant incubated for 1 hr prior to testing by phenol red based stopped-...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details
PubMed
TargetCarbonic anhydrase 1(Human)
University of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM10880(Acetazolamide, AAZ | AZA2 | CHEMBL20 | Acetazolami...)
Affinity DataKi:  2.50E+5nMAssay Description:Inhibition of recombinant human carbonic anhydrase 1 assessed as inhibition constant incubated for 1 hr prior to testing by phenol red based stopped-...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details
PubMedPDB3D3D Structure (crystal)