Compile Data Set for Download or QSAR
Report error Found 6 Enz. Inhib. hit(s) with all data for entry = 50016762
TargetSodium channel protein type 8 subunit alpha(Human)
Smith, Gambrell & Russell

Curated by ChEMBL
LigandPNGBDBM50597018(CHEMBL5182397)
Affinity DataIC50: 1.20nMAssay Description:Inhibition of human Nav1.8 channel stably expressed in HEK293 cells assessed as sodium current flow at holding potential of -90mV by whole-cell volta...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetSodium channel protein type 8 subunit alpha(Human)
Smith, Gambrell & Russell

Curated by ChEMBL
LigandPNGBDBM50597016(CHEMBL5196342)
Affinity DataIC50: 2.60nMAssay Description:Inhibition of human Nav1.8 channel stably expressed in HEK293 cells assessed as sodium current flow at holding potential of -90mV by whole-cell volta...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetSodium channel protein type 8 subunit alpha(Human)
Smith, Gambrell & Russell

Curated by ChEMBL
LigandPNGBDBM50597020(CHEMBL5193659)
Affinity DataIC50: 2.90nMAssay Description:Inhibition of human Nav1.8 channel stably expressed in HEK293 cells assessed as sodium current flow at holding potential of -90mV by whole-cell volta...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetSodium channel protein type 8 subunit alpha(Human)
Smith, Gambrell & Russell

Curated by ChEMBL
LigandPNGBDBM50597015(CHEMBL5194703)
Affinity DataIC50: 3.40nMAssay Description:Inhibition of human Nav1.8 channel stably expressed in HEK293 cells assessed as sodium current flow at holding potential of -90mV by whole-cell volta...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetSodium channel protein type 8 subunit alpha(Human)
Smith, Gambrell & Russell

Curated by ChEMBL
LigandPNGBDBM50597017(CHEMBL5183619)
Affinity DataIC50: 4.10nMAssay Description:Inhibition of human Nav1.8 channel stably expressed in HEK293 cells assessed as sodium current flow at holding potential of -90mV by whole-cell volta...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetSodium channel protein type 8 subunit alpha(Human)
Smith, Gambrell & Russell

Curated by ChEMBL
LigandPNGBDBM50597019(CHEMBL5197040)
Affinity DataIC50: 4.20nMAssay Description:Inhibition of human Nav1.8 channel stably expressed in HEK293 cells assessed as sodium current flow at holding potential of -90mV by whole-cell volta...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed