Compile Data Set for Download or QSAR
Report error Found 28 Enz. Inhib. hit(s) with all data for entry = 50017895
TargetSerine/threonine-protein kinase RIO2(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM31095(5-[(Z)-(5-fluoranyl-2-oxidanylidene-1H-indol-3-yli...)
Affinity DataKd: <200nMAssay Description:Binding affinity to RIOK2 (unknown origin) assessed as dissociation constantMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetSerine/threonine-protein kinase RIO2(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM50605926(CHEMBL5170056)
Affinity DataKd: >1.00E+3nMAssay Description:Binding affinity to wild-type human partial length RIOK2 (M1 to D313 residues) expressed in mammalian expression system assessed as dissociation cons...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetSerine/threonine-protein kinase RIO2(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM50605925(CHEMBL5202446)
Affinity DataKd: >1.00E+3nMAssay Description:Binding affinity to wild-type human partial length RIOK2 (M1 to D313 residues) expressed in mammalian expression system assessed as dissociation cons...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetSerine/threonine-protein kinase RIO2(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM50605924(CHEMBL5182037)
Affinity DataKd: >1.00E+3nMAssay Description:Binding affinity to wild-type human partial length RIOK2 (M1 to D313 residues) expressed in mammalian expression system assessed as dissociation cons...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetSerine/threonine-protein kinase RIO2(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM50605923(CHEMBL5205484)
Affinity DataKd: >1.00E+3nMAssay Description:Binding affinity to wild-type human partial length RIOK2 (M1 to D313 residues) expressed in mammalian expression system assessed as dissociation cons...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetSerine/threonine-protein kinase RIO2(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM50605922(CHEMBL5179811)
Affinity DataKd: >1.00E+3nMAssay Description:Binding affinity to wild-type human partial length RIOK2 (M1 to D313 residues) expressed in mammalian expression system assessed as dissociation cons...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetSerine/threonine-protein kinase RIO2(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM50605921(CHEMBL5188981)
Affinity DataKd:  840nMAssay Description:Binding affinity to wild-type human partial length RIOK2 (M1 to D313 residues) expressed in mammalian expression system assessed as dissociation cons...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetSerine/threonine-protein kinase RIO2(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM50605920(CHEMBL5205288)
Affinity DataKd:  810nMAssay Description:Binding affinity to wild-type human partial length RIOK2 (M1 to D313 residues) expressed in mammalian expression system assessed as dissociation cons...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetSerine/threonine-protein kinase RIO2(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM50605919(CHEMBL5177849)
Affinity DataKd:  575nMAssay Description:Binding affinity to wild-type human partial length RIOK2 (M1 to D313 residues) expressed in mammalian expression system assessed as dissociation cons...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetSerine/threonine-protein kinase RIO2(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM50605918(CHEMBL5189953)
Affinity DataKd:  455nMAssay Description:Binding affinity to wild-type human partial length RIOK2 (M1 to D313 residues) expressed in mammalian expression system assessed as dissociation cons...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetSerine/threonine-protein kinase RIO2(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM50605917(CHEMBL5184335)
Affinity DataKd:  385nMAssay Description:Binding affinity to wild-type human partial length RIOK2 (M1 to D313 residues) expressed in mammalian expression system assessed as dissociation cons...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetSerine/threonine-protein kinase RIO2(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM50605916(CHEMBL5187692)
Affinity DataKd:  235nMAssay Description:Binding affinity to wild-type human partial length RIOK2 (M1 to D313 residues) expressed in mammalian expression system assessed as dissociation cons...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetSerine/threonine-protein kinase RIO2(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM50605915(CHEMBL5174394)
Affinity DataKd:  200nMAssay Description:Binding affinity to wild-type human partial length RIOK2 (M1 to D313 residues) expressed in mammalian expression system assessed as dissociation cons...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetSerine/threonine-protein kinase RIO2(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM50550127(CHEMBL4781866)
Affinity DataKd:  150nMAssay Description:Binding affinity to wild-type human partial length RIOK2 (M1 to D313 residues) expressed in mammalian expression system assessed as dissociation cons...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetSerine/threonine-protein kinase RIO2(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM50605914(CHEMBL5190993)
Affinity DataKd:  120nMAssay Description:Binding affinity to wild-type human partial length RIOK2 (M1 to D313 residues) expressed in mammalian expression system assessed as dissociation cons...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetSerine/threonine-protein kinase RIO2(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM50605913(CHEMBL5194039)
Affinity DataKd:  63nMAssay Description:Binding affinity to wild-type human partial length RIOK2 (M1 to D313 residues) expressed in mammalian expression system assessed as dissociation cons...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetSerine/threonine-protein kinase RIO2(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM50605912(CHEMBL5190197)
Affinity DataKd:  63nMAssay Description:Binding affinity to wild-type human partial length RIOK2 (M1 to D313 residues) expressed in mammalian expression system assessed as dissociation cons...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetSerine/threonine-protein kinase RIO2(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM50605911(CHEMBL5192566)
Affinity DataKd:  49nMAssay Description:Binding affinity to wild-type human partial length RIOK2 (M1 to D313 residues) expressed in mammalian expression system assessed as dissociation cons...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetSerine/threonine-protein kinase RIO2(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM50605910(CHEMBL5184015)
Affinity DataKd:  48nMAssay Description:Binding affinity to wild-type human partial length RIOK2 (M1 to D313 residues) expressed in mammalian expression system assessed as dissociation cons...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetSerine/threonine-protein kinase RIO2(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM50605909(CHEMBL5190698)
Affinity DataKd:  18nMAssay Description:Binding affinity to wild-type human partial length RIOK2 (M1 to D313 residues) expressed in mammalian expression system assessed as dissociation cons...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetSerine/threonine-protein kinase RIO2(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM50605908(CHEMBL5199096)
Affinity DataKd:  8.40nMAssay Description:Binding affinity to wild-type human partial length RIOK2 (M1 to D313 residues) expressed in mammalian expression system assessed as dissociation cons...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetSerine/threonine-protein kinase RIO2(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM50605907(CHEMBL5174723)
Affinity DataKd:  7.30nMAssay Description:Binding affinity to wild-type human partial length RIOK2 (M1 to D313 residues) expressed in mammalian expression system assessed as dissociation cons...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetSerine/threonine-protein kinase RIO2(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM50605906(CHEMBL5172767)
Affinity DataKd:  6.10nMAssay Description:Binding affinity to wild-type human partial length RIOK2 (M1 to D313 residues) expressed in mammalian expression system assessed as dissociation cons...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetSerine/threonine-protein kinase RIO2(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM4814(SUNITINIB MALATE | CHEMBL535 | N-[2-(diethylamino)...)
Affinity DataKd: <200nMAssay Description:Binding affinity to RIOK2 (unknown origin) assessed as dissociation constantMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetSerine/threonine-protein kinase RIO2(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM50605905(CHEMBL5184068)
Affinity DataKd: <200nMAssay Description:Binding affinity to RIOK2 (unknown origin) assessed as dissociation constantMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetSerine/threonine-protein kinase RIO2(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM50605906(CHEMBL5172767)
Affinity DataIC50: 139nMAssay Description:Inhibition of N-terminal hexahistidine-SUMO-tagged human full length RIOK2 (residues 1 to 321) expressed in Escherichia coli BL21 (DE3) incubated for...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetSerine/threonine-protein kinase RIO2(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM50550133(CHEMBL4754518)
Affinity DataIC50: 6.60E+3nMAssay Description:Displacement of fluorescent tracer K5 from N-terminal full-length NanoLuc-fused RIOK2 (unknown origin) expressed in HEK293 cells using NanoGlo substr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetSerine/threonine-protein kinase RIO2(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM50550127(CHEMBL4781866)
Affinity DataIC50: 1.46E+4nMAssay Description:Displacement of fluorescent tracer K5 from N-terminal full-length NanoLuc-fused RIOK2 (unknown origin) expressed in HEK293 cells using NanoGlo substr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed