Compile Data Set for Download or QSAR
Report error Found 38 Enz. Inhib. hit(s) with all data for entry = 50017272
TargetOxysterols receptor LXR-beta(Human)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50600562(CHEMBL5184224)
Affinity DataEC50:  740nMAssay Description:Agonist activity against human LXRbeta expressed in human HEK293T cells co-expressing CMX-GAL4N-hLXRbeta incubated for 24 hrs by reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetOxysterols receptor LXR-beta(Human)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50179869(N-methyl-N-[4-(2,2,2-trifluoro-1-hydroxy-1-trifluo...)
Affinity DataEC50:  2.93E+3nMAssay Description:Agonist activity against human LXRbeta expressed in human HEK293T cells co-expressing CMX-GAL4N-hLXRbeta incubated for 24 hrs by reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetOxysterols receptor LXR-beta(Human)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50600554(CHEMBL5173460)
Affinity DataEC50:  1.41E+3nMAssay Description:Agonist activity against human LXRbeta expressed in human HEK293T cells co-expressing CMX-GAL4N-hLXRbeta incubated for 24 hrs by reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetOxysterols receptor LXR-beta(Human)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50600555(CHEMBL5173224)
Affinity DataEC50:  530nMAssay Description:Agonist activity against human LXRbeta expressed in human HEK293T cells co-expressing CMX-GAL4N-hLXRbeta incubated for 24 hrs by reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetOxysterols receptor LXR-beta(Human)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50600556(CHEMBL5203561)
Affinity DataEC50:  590nMAssay Description:Agonist activity against human LXRbeta expressed in human HEK293T cells co-expressing CMX-GAL4N-hLXRbeta incubated for 24 hrs by reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetOxysterols receptor LXR-beta(Human)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50600557(CHEMBL5200504)
Affinity DataEC50:  1.98E+3nMAssay Description:Agonist activity against human LXRbeta expressed in human HEK293T cells co-expressing CMX-GAL4N-hLXRbeta incubated for 24 hrs by reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetOxysterols receptor LXR-beta(Human)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50600558(CHEMBL5182815)
Affinity DataEC50:  1.80E+3nMAssay Description:Agonist activity against human LXRbeta expressed in human HEK293T cells co-expressing CMX-GAL4N-hLXRbeta incubated for 24 hrs by reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetOxysterols receptor LXR-beta(Human)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50600559(CHEMBL5183659)
Affinity DataEC50:  450nMAssay Description:Agonist activity against human LXRbeta expressed in human HEK293T cells co-expressing CMX-GAL4N-hLXRbeta incubated for 24 hrs by reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetOxysterols receptor LXR-beta(Human)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50600560(CHEMBL5169521)
Affinity DataEC50:  1.70E+3nMAssay Description:Agonist activity against human LXRbeta expressed in human HEK293T cells co-expressing CMX-GAL4N-hLXRbeta incubated for 24 hrs by reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetOxysterols receptor LXR-beta(Human)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50600561(CHEMBL5184494)
Affinity DataEC50:  650nMAssay Description:Agonist activity against human LXRbeta expressed in human HEK293T cells co-expressing CMX-GAL4N-hLXRbeta incubated for 24 hrs by reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetOxysterols receptor LXR-beta(Human)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM19993(CHEMBL62136 | [3H]T0901317 | T 0901317 | N-[4-(1,1...)
Affinity DataEC50:  260nMAssay Description:Agonist activity against human LXRbeta expressed in human HEK293T cells co-expressing CMX-GAL4N-hLXRbeta incubated for 24 hrs by reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetOxysterols receptor LXR-beta(Human)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50600563(CHEMBL5195024)
Affinity DataEC50:  740nMAssay Description:Agonist activity against human LXRbeta expressed in human HEK293T cells co-expressing CMX-GAL4N-hLXRbeta incubated for 24 hrs by reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetOxysterols receptor LXR-beta(Human)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50600564(CHEMBL5187585)
Affinity DataEC50:  720nMAssay Description:Agonist activity against human LXRbeta expressed in human HEK293T cells co-expressing CMX-GAL4N-hLXRbeta incubated for 24 hrs by reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetOxysterols receptor LXR-beta(Human)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50600565(CHEMBL5188694)
Affinity DataEC50:  510nMAssay Description:Agonist activity against human LXRbeta expressed in human HEK293T cells co-expressing CMX-GAL4N-hLXRbeta incubated for 24 hrs by reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetOxysterols receptor LXR-beta(Human)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50600566(CHEMBL5179248)
Affinity DataEC50:  690nMAssay Description:Agonist activity against human LXRbeta expressed in human HEK293T cells co-expressing CMX-GAL4N-hLXRbeta incubated for 24 hrs by reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetOxysterols receptor LXR-beta(Human)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50600567(CHEMBL5196110)
Affinity DataEC50:  1.73E+3nMAssay Description:Agonist activity against human LXRbeta expressed in human HEK293T cells co-expressing CMX-GAL4N-hLXRbeta incubated for 24 hrs by reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetOxysterols receptor LXR-beta(Human)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50600568(CHEMBL5192368)
Affinity DataEC50:  3.34E+3nMAssay Description:Agonist activity against human LXRbeta expressed in human HEK293T cells co-expressing CMX-GAL4N-hLXRbeta incubated for 24 hrs by reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetOxysterols receptor LXR-beta(Human)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50600569(CHEMBL5198099)
Affinity DataEC50:  4.03E+3nMAssay Description:Agonist activity against human LXRbeta expressed in human HEK293T cells co-expressing CMX-GAL4N-hLXRbeta incubated for 24 hrs by reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetOxysterols receptor LXR-beta(Human)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50600570(CHEMBL5195914)
Affinity DataEC50:  5.03E+3nMAssay Description:Agonist activity against human LXRbeta expressed in human HEK293T cells co-expressing CMX-GAL4N-hLXRbeta incubated for 24 hrs by reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetOxysterols receptor LXR-alpha(Human)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50600562(CHEMBL5184224)
Affinity DataEC50:  1.43E+3nMAssay Description:Agonist activity against human LXRalpha expressed in human HEK293T cells co-expressing CMX-GAL4N-hLXRalpha incubated for 24 hrs by reporter gene assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetOxysterols receptor LXR-alpha(Human)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50179869(N-methyl-N-[4-(2,2,2-trifluoro-1-hydroxy-1-trifluo...)
Affinity DataEC50:  3.76E+3nMAssay Description:Agonist activity against human LXRalpha expressed in human HEK293T cells co-expressing CMX-GAL4N-hLXRalpha incubated for 24 hrs by reporter gene assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetOxysterols receptor LXR-alpha(Human)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50600554(CHEMBL5173460)
Affinity DataEC50:  3.12E+3nMAssay Description:Agonist activity against human LXRalpha expressed in human HEK293T cells co-expressing CMX-GAL4N-hLXRalpha incubated for 24 hrs by reporter gene assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetOxysterols receptor LXR-alpha(Human)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50600555(CHEMBL5173224)
Affinity DataEC50:  620nMAssay Description:Agonist activity against human LXRalpha expressed in human HEK293T cells co-expressing CMX-GAL4N-hLXRalpha incubated for 24 hrs by reporter gene assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetOxysterols receptor LXR-alpha(Human)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50600556(CHEMBL5203561)
Affinity DataEC50:  430nMAssay Description:Agonist activity against human LXRalpha expressed in human HEK293T cells co-expressing CMX-GAL4N-hLXRalpha incubated for 24 hrs by reporter gene assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetOxysterols receptor LXR-alpha(Human)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50600557(CHEMBL5200504)
Affinity DataEC50:  4.98E+3nMAssay Description:Agonist activity against human LXRalpha expressed in human HEK293T cells co-expressing CMX-GAL4N-hLXRalpha incubated for 24 hrs by reporter gene assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetOxysterols receptor LXR-alpha(Human)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50600558(CHEMBL5182815)
Affinity DataEC50:  2.06E+3nMAssay Description:Agonist activity against human LXRalpha expressed in human HEK293T cells co-expressing CMX-GAL4N-hLXRalpha incubated for 24 hrs by reporter gene assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetOxysterols receptor LXR-alpha(Human)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50600559(CHEMBL5183659)
Affinity DataEC50:  500nMAssay Description:Agonist activity against human LXRalpha expressed in human HEK293T cells co-expressing CMX-GAL4N-hLXRalpha incubated for 24 hrs by reporter gene assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetOxysterols receptor LXR-alpha(Human)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50600560(CHEMBL5169521)
Affinity DataEC50:  2.35E+3nMAssay Description:Agonist activity against human LXRalpha expressed in human HEK293T cells co-expressing CMX-GAL4N-hLXRalpha incubated for 24 hrs by reporter gene assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetOxysterols receptor LXR-alpha(Human)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50600561(CHEMBL5184494)
Affinity DataEC50:  1.13E+3nMAssay Description:Agonist activity against human LXRalpha expressed in human HEK293T cells co-expressing CMX-GAL4N-hLXRalpha incubated for 24 hrs by reporter gene assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetOxysterols receptor LXR-alpha(Human)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM19993(CHEMBL62136 | [3H]T0901317 | T 0901317 | N-[4-(1,1...)
Affinity DataEC50:  260nMAssay Description:Agonist activity against human LXRalpha expressed in human HEK293T cells co-expressing CMX-GAL4N-hLXRalpha incubated for 24 hrs by reporter gene assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetOxysterols receptor LXR-alpha(Human)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50600563(CHEMBL5195024)
Affinity DataEC50:  2.15E+3nMAssay Description:Agonist activity against human LXRalpha expressed in human HEK293T cells co-expressing CMX-GAL4N-hLXRalpha incubated for 24 hrs by reporter gene assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetOxysterols receptor LXR-alpha(Human)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50600564(CHEMBL5187585)
Affinity DataEC50:  940nMAssay Description:Agonist activity against human LXRalpha expressed in human HEK293T cells co-expressing CMX-GAL4N-hLXRalpha incubated for 24 hrs by reporter gene assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetOxysterols receptor LXR-alpha(Human)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50600565(CHEMBL5188694)
Affinity DataEC50:  580nMAssay Description:Agonist activity against human LXRalpha expressed in human HEK293T cells co-expressing CMX-GAL4N-hLXRalpha incubated for 24 hrs by reporter gene assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetOxysterols receptor LXR-alpha(Human)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50600566(CHEMBL5179248)
Affinity DataEC50:  590nMAssay Description:Agonist activity against human LXRalpha expressed in human HEK293T cells co-expressing CMX-GAL4N-hLXRalpha incubated for 24 hrs by reporter gene assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetOxysterols receptor LXR-alpha(Human)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50600567(CHEMBL5196110)
Affinity DataEC50:  1.46E+3nMAssay Description:Agonist activity against human LXRalpha expressed in human HEK293T cells co-expressing CMX-GAL4N-hLXRalpha incubated for 24 hrs by reporter gene assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetOxysterols receptor LXR-alpha(Human)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50600568(CHEMBL5192368)
Affinity DataEC50:  4.45E+3nMAssay Description:Agonist activity against human LXRalpha expressed in human HEK293T cells co-expressing CMX-GAL4N-hLXRalpha incubated for 24 hrs by reporter gene assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetOxysterols receptor LXR-alpha(Human)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50600569(CHEMBL5198099)
Affinity DataEC50:  4.45E+3nMAssay Description:Agonist activity against human LXRalpha expressed in human HEK293T cells co-expressing CMX-GAL4N-hLXRalpha incubated for 24 hrs by reporter gene assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetOxysterols receptor LXR-alpha(Human)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50600570(CHEMBL5195914)
Affinity DataEC50:  8.50E+3nMAssay Description:Agonist activity against human LXRalpha expressed in human HEK293T cells co-expressing CMX-GAL4N-hLXRalpha incubated for 24 hrs by reporter gene assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed