Compile Data Set for Download or QSAR
Report error Found 33 Enz. Inhib. hit(s) with all data for entry = 50016272
TargetReceptor tyrosine-protein kinase erbB-2(Human)
China Medical University

Curated by ChEMBL
LigandPNGBDBM50593742(CHEMBL5189852)
Affinity DataIC50: 30nMAssay Description:Inhibition of human HER2 incubated for 25 mins by ADP-Glo reagent based microplate reader analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details
PubMed
TargetReceptor tyrosine-protein kinase erbB-2(Human)
China Medical University

Curated by ChEMBL
LigandPNGBDBM50593741(CHEMBL5171922)
Affinity DataIC50: 230nMAssay Description:Inhibition of human HER2 incubated for 25 mins by ADP-Glo reagent based microplate reader analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details
PubMed
TargetReceptor tyrosine-protein kinase erbB-2(Human)
China Medical University

Curated by ChEMBL
LigandPNGBDBM50593757(CHEMBL5196657)
Affinity DataIC50: 250nMAssay Description:Inhibition of human HER2 incubated for 25 mins by ADP-Glo reagent based microplate reader analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details
PubMed
TargetReceptor tyrosine-protein kinase erbB-2(Human)
China Medical University

Curated by ChEMBL
LigandPNGBDBM50593765(Mubritinib | TAK-165 | MUBRITINIB)
Affinity DataIC50: 350nMAssay Description:Inhibition of human HER2 incubated for 25 mins by ADP-Glo reagent based microplate reader analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details
PubMed
TargetReceptor tyrosine-protein kinase erbB-2(Human)
China Medical University

Curated by ChEMBL
LigandPNGBDBM50593743(CHEMBL5207091)
Affinity DataIC50: 440nMAssay Description:Inhibition of human HER2 incubated for 25 mins by ADP-Glo reagent based microplate reader analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details
PubMed
TargetReceptor tyrosine-protein kinase erbB-2(Human)
China Medical University

Curated by ChEMBL
LigandPNGBDBM50593760(CHEMBL5201807)
Affinity DataIC50: 820nMAssay Description:Inhibition of human HER2 incubated for 25 mins by ADP-Glo reagent based microplate reader analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details
PubMed
TargetReceptor tyrosine-protein kinase erbB-2(Human)
China Medical University

Curated by ChEMBL
LigandPNGBDBM50593744(CHEMBL5189871)
Affinity DataIC50: 860nMAssay Description:Inhibition of human HER2 incubated for 25 mins by ADP-Glo reagent based microplate reader analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details
PubMed
TargetReceptor tyrosine-protein kinase erbB-2(Human)
China Medical University

Curated by ChEMBL
LigandPNGBDBM50593740(CHEMBL5187503)
Affinity DataIC50: 1.07E+3nMAssay Description:Inhibition of human HER2 incubated for 25 mins by ADP-Glo reagent based microplate reader analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details
PubMed
TargetReceptor tyrosine-protein kinase erbB-2(Human)
China Medical University

Curated by ChEMBL
LigandPNGBDBM50593764(CHEMBL5174917)
Affinity DataIC50: 1.11E+3nMAssay Description:Inhibition of human HER2 incubated for 25 mins by ADP-Glo reagent based microplate reader analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details
PubMed
TargetReceptor tyrosine-protein kinase erbB-2(Human)
China Medical University

Curated by ChEMBL
LigandPNGBDBM50593739(CHEMBL5186640)
Affinity DataIC50: 1.29E+3nMAssay Description:Inhibition of human HER2 incubated for 25 mins by ADP-Glo reagent based microplate reader analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details
PubMed
TargetReceptor tyrosine-protein kinase erbB-2(Human)
China Medical University

Curated by ChEMBL
LigandPNGBDBM50593745(CHEMBL5190408)
Affinity DataIC50: 1.83E+3nMAssay Description:Inhibition of human HER2 incubated for 25 mins by ADP-Glo reagent based microplate reader analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details
PubMed
TargetReceptor tyrosine-protein kinase erbB-2(Human)
China Medical University

Curated by ChEMBL
LigandPNGBDBM50593748(CHEMBL5204707)
Affinity DataIC50: 1.84E+3nMAssay Description:Inhibition of human HER2 incubated for 25 mins by ADP-Glo reagent based microplate reader analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details
PubMed
TargetReceptor tyrosine-protein kinase erbB-2(Human)
China Medical University

Curated by ChEMBL
LigandPNGBDBM50593751(CHEMBL5179098)
Affinity DataIC50: 1.94E+3nMAssay Description:Inhibition of human HER2 incubated for 25 mins by ADP-Glo reagent based microplate reader analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details
PubMed
TargetReceptor tyrosine-protein kinase erbB-2(Human)
China Medical University

Curated by ChEMBL
LigandPNGBDBM50593738(CHEMBL5183608)
Affinity DataIC50: 2.01E+3nMAssay Description:Inhibition of human HER2 incubated for 25 mins by ADP-Glo reagent based microplate reader analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details
PubMed
TargetReceptor tyrosine-protein kinase erbB-2(Human)
China Medical University

Curated by ChEMBL
LigandPNGBDBM50593736(CHEMBL5193804)
Affinity DataIC50: 2.17E+3nMAssay Description:Inhibition of human HER2 incubated for 25 mins by ADP-Glo reagent based microplate reader analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details
PubMed
TargetReceptor tyrosine-protein kinase erbB-2(Human)
China Medical University

Curated by ChEMBL
LigandPNGBDBM50593762(CHEMBL5171924)
Affinity DataIC50: 2.21E+3nMAssay Description:Inhibition of human HER2 incubated for 25 mins by ADP-Glo reagent based microplate reader analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details
PubMed
TargetReceptor tyrosine-protein kinase erbB-2(Human)
China Medical University

Curated by ChEMBL
LigandPNGBDBM50593754(CHEMBL5181577)
Affinity DataIC50: 2.25E+3nMAssay Description:Inhibition of human HER2 incubated for 25 mins by ADP-Glo reagent based microplate reader analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details
PubMed
TargetReceptor tyrosine-protein kinase erbB-2(Human)
China Medical University

Curated by ChEMBL
LigandPNGBDBM50593737(CHEMBL5186298)
Affinity DataIC50: 2.79E+3nMAssay Description:Inhibition of human HER2 incubated for 25 mins by ADP-Glo reagent based microplate reader analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details
PubMed
TargetReceptor tyrosine-protein kinase erbB-2(Human)
China Medical University

Curated by ChEMBL
LigandPNGBDBM50593746(CHEMBL5174515)
Affinity DataIC50: 3.07E+3nMAssay Description:Inhibition of human HER2 incubated for 25 mins by ADP-Glo reagent based microplate reader analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details
PubMed
TargetReceptor tyrosine-protein kinase erbB-2(Human)
China Medical University

Curated by ChEMBL
LigandPNGBDBM50593763(CHEMBL5193926)
Affinity DataIC50: 3.25E+3nMAssay Description:Inhibition of human HER2 incubated for 25 mins by ADP-Glo reagent based microplate reader analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details
PubMed
TargetReceptor tyrosine-protein kinase erbB-2(Human)
China Medical University

Curated by ChEMBL
LigandPNGBDBM50593755(CHEMBL5180538)
Affinity DataIC50: 3.58E+3nMAssay Description:Inhibition of human HER2 incubated for 25 mins by ADP-Glo reagent based microplate reader analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details
PubMed
TargetReceptor tyrosine-protein kinase erbB-2(Human)
China Medical University

Curated by ChEMBL
LigandPNGBDBM50593758(CHEMBL5174439)
Affinity DataIC50: 4.86E+3nMAssay Description:Inhibition of human HER2 incubated for 25 mins by ADP-Glo reagent based microplate reader analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details
PubMed
TargetReceptor tyrosine-protein kinase erbB-2(Human)
China Medical University

Curated by ChEMBL
LigandPNGBDBM50593752(CHEMBL5183407)
Affinity DataIC50: 5.26E+3nMAssay Description:Inhibition of human HER2 incubated for 25 mins by ADP-Glo reagent based microplate reader analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details
PubMed
TargetReceptor tyrosine-protein kinase erbB-2(Human)
China Medical University

Curated by ChEMBL
LigandPNGBDBM50593733(CHEMBL5206700)
Affinity DataIC50: 5.30E+3nMAssay Description:Inhibition of human HER2 incubated for 25 mins by ADP-Glo reagent based microplate reader analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details
PubMed
TargetReceptor tyrosine-protein kinase erbB-2(Human)
China Medical University

Curated by ChEMBL
LigandPNGBDBM50593734(CHEMBL5202630)
Affinity DataIC50: 5.79E+3nMAssay Description:Inhibition of human HER2 incubated for 25 mins by ADP-Glo reagent based microplate reader analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details
PubMed
TargetReceptor tyrosine-protein kinase erbB-2(Human)
China Medical University

Curated by ChEMBL
LigandPNGBDBM50593749(CHEMBL5180660)
Affinity DataIC50: 7.59E+3nMAssay Description:Inhibition of human HER2 incubated for 25 mins by ADP-Glo reagent based microplate reader analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details
PubMed
TargetReceptor tyrosine-protein kinase erbB-2(Human)
China Medical University

Curated by ChEMBL
LigandPNGBDBM50593735(CHEMBL5182590)
Affinity DataIC50: 8.63E+3nMAssay Description:Inhibition of human HER2 incubated for 25 mins by ADP-Glo reagent based microplate reader analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details
PubMed
TargetReceptor tyrosine-protein kinase erbB-2(Human)
China Medical University

Curated by ChEMBL
LigandPNGBDBM50593756(CHEMBL5193640)
Affinity DataIC50: 9.28E+3nMAssay Description:Inhibition of human HER2 incubated for 25 mins by ADP-Glo reagent based microplate reader analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details
PubMed
TargetReceptor tyrosine-protein kinase erbB-2(Human)
China Medical University

Curated by ChEMBL
LigandPNGBDBM50593753(CHEMBL5169997)
Affinity DataIC50: 1.02E+4nMAssay Description:Inhibition of human HER2 incubated for 25 mins by ADP-Glo reagent based microplate reader analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details
PubMed
TargetReceptor tyrosine-protein kinase erbB-2(Human)
China Medical University

Curated by ChEMBL
LigandPNGBDBM50593750(CHEMBL5192580)
Affinity DataIC50: 1.21E+4nMAssay Description:Inhibition of human HER2 incubated for 25 mins by ADP-Glo reagent based microplate reader analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details
PubMed
TargetReceptor tyrosine-protein kinase erbB-2(Human)
China Medical University

Curated by ChEMBL
LigandPNGBDBM50593759(CHEMBL5183228)
Affinity DataIC50: 1.33E+4nMAssay Description:Inhibition of human HER2 incubated for 25 mins by ADP-Glo reagent based microplate reader analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details
PubMed
TargetReceptor tyrosine-protein kinase erbB-2(Human)
China Medical University

Curated by ChEMBL
LigandPNGBDBM50593761(CHEMBL5172914)
Affinity DataIC50: 3.47E+4nMAssay Description:Inhibition of human HER2 incubated for 25 mins by ADP-Glo reagent based microplate reader analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details
PubMed
TargetReceptor tyrosine-protein kinase erbB-2(Human)
China Medical University

Curated by ChEMBL
LigandPNGBDBM50593747(CHEMBL5192229)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human HER2 incubated for 25 mins by ADP-Glo reagent based microplate reader analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details
PubMed