Compile Data Set for Download or QSAR
Report error Found 10 Enz. Inhib. hit(s) with all data for entry = 50017218
TargetLegumain(Human)
University of Florence

Curated by ChEMBL
LigandPNGBDBM50600333(CHEMBL5183094)
Affinity DataIC50: 89nMAssay Description:Inhibition of recombinant human Asparagine endopeptidase preincubated for 5 mins followed by Z-Ala-Ala-Asn-AMC substrate addition measured after 2 hr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetLegumain(Human)
University of Florence

Curated by ChEMBL
LigandPNGBDBM50600329(CHEMBL5197937)
Affinity DataIC50: 498nMAssay Description:Inhibition of recombinant human Asparagine endopeptidase preincubated for 5 mins followed by Z-Ala-Ala-Asn-AMC substrate addition measured after 2 hr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetLegumain(Human)
University of Florence

Curated by ChEMBL
LigandPNGBDBM50600332(CHEMBL5194542)
Affinity DataIC50: 547nMAssay Description:Inhibition of recombinant human Asparagine endopeptidase preincubated for 5 mins followed by Z-Ala-Ala-Asn-AMC substrate addition measured after 2 hr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetLegumain(Human)
University of Florence

Curated by ChEMBL
LigandPNGBDBM50600334(CHEMBL5175987)
Affinity DataIC50: 757nMAssay Description:Inhibition of recombinant human Asparagine endopeptidase preincubated for 5 mins followed by Z-Ala-Ala-Asn-AMC substrate addition measured after 2 hr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetLegumain(Human)
University of Florence

Curated by ChEMBL
LigandPNGBDBM50600328(CHEMBL5185780)
Affinity DataIC50: 844nMAssay Description:Inhibition of recombinant human Asparagine endopeptidase preincubated for 5 mins followed by Z-Ala-Ala-Asn-AMC substrate addition measured after 2 hr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetLegumain(Human)
University of Florence

Curated by ChEMBL
LigandPNGBDBM50600335(CHEMBL5208689)
Affinity DataIC50: 4.83E+3nMAssay Description:Inhibition of recombinant human Asparagine endopeptidase preincubated for 5 mins followed by Z-Ala-Ala-Asn-AMC substrate addition measured after 2 hr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetLegumain(Human)
University of Florence

Curated by ChEMBL
LigandPNGBDBM50600330(CHEMBL5186940)
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of recombinant human Asparagine endopeptidase preincubated for 5 mins followed by Z-Ala-Ala-Asn-AMC substrate addition measured after 2 hr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetLegumain(Human)
University of Florence

Curated by ChEMBL
LigandPNGBDBM50600331(CHEMBL5175999)
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of recombinant human Asparagine endopeptidase preincubated for 5 mins followed by Z-Ala-Ala-Asn-AMC substrate addition measured after 2 hr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetLegumain(Human)
University of Florence

Curated by ChEMBL
LigandPNGBDBM50600336(CHEMBL5194228)
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of recombinant human Asparagine endopeptidase preincubated for 5 mins followed by Z-Ala-Ala-Asn-AMC substrate addition measured after 2 hr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetLegumain(Human)
University of Florence

Curated by ChEMBL
LigandPNGBDBM50600337(CHEMBL5185358)
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of recombinant human Asparagine endopeptidase preincubated for 5 mins followed by Z-Ala-Ala-Asn-AMC substrate addition measured after 2 hr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed