Compile Data Set for Download or QSAR
Report error Found 17 Enz. Inhib. hit(s) with all data for entry = 50035600
TargetRenin(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50024146({1-[1-[1-(2,2-Difluoro-2-{2-methyl-1-[(pyridin-2-y...)
Affinity DataIC50: 0.520nMAssay Description:Inhibition of human plasma reninMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2012
Entry Details Article
PubMed
TargetRenin(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50024149({1-[1-(1-Cyclohexylmethyl-3,3-difluoro-2-hydroxy-3...)
Affinity DataIC50: 0.570nMAssay Description:Inhibition of human plasma reninMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2012
Entry Details Article
PubMed
TargetRenin(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50024144({1-[1-(1-Benzyl-3,3-difluoro-3-{2-methyl-1-[(pyrid...)
Affinity DataIC50: 1.30nMAssay Description:Inhibition of human plasma reninMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2012
Entry Details Article
PubMed
TargetRenin(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50024145({1-[1-(1-Cyclohexylmethyl-3,3-difluoro-3-{2-methyl...)
Affinity DataIC50: 1.40nMAssay Description:Inhibition of human plasma reninMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2012
Entry Details Article
PubMed
TargetRenin(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50024147({1-[1-[1-(1-Hydroxy-2-{2-methyl-1-[(pyridin-2-ylme...)
Affinity DataIC50: 1.70nMAssay Description:Inhibition of human plasma reninMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2012
Entry Details Article
PubMed
TargetRenin(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50024143({1-[1-[1-(2,2-Difluoro-2-{2-methyl-1-[(pyridin-2-y...)
Affinity DataIC50: 2.5nMAssay Description:Inhibition of human plasma reninMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2012
Entry Details Article
PubMed
TargetPepsin A(Pig)
TBA

Curated by ChEMBL
LigandPNGBDBM912(PEPSTATIN | Pepstatine | N-[(3-Methyl-1-oxobutyl)-...)
Affinity DataIC50: 10nMAssay Description:Compound was tested for inhibition of porcine pepsinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2012
Entry Details Article
PubMed
TargetRenin(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50024141({1-[1-[1-(2,2-Difluoro-1-hydroxy-2-{2-methyl-1-[(p...)
Affinity DataIC50: 12nMAssay Description:Inhibition of human plasma reninMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2012
Entry Details Article
PubMed
TargetRenin(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50024142({1-[1-(1-Benzyl-3,3-difluoro-2-hydroxy-3-{2-methyl...)
Affinity DataIC50: 13nMAssay Description:Inhibition of human plasma reninMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2012
Entry Details Article
PubMed
TargetCathepsin D(Bovine)
TBA

Curated by ChEMBL
LigandPNGBDBM912(PEPSTATIN | Pepstatine | N-[(3-Methyl-1-oxobutyl)-...)
Affinity DataIC50: 28nMAssay Description:Compound was tested for inhibition of bovine cathepsin DMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2012
Entry Details Article
PubMed
TargetRenin(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50024148((1-{2-(2H-Imidazol-2-yl)-1-[3-methyl-1-(2-{2-methy...)
Affinity DataIC50: 34nMAssay Description:Inhibition of human plasma reninMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2012
Entry Details Article
PubMed
TargetRenin(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50024150({1-[1-[1-(2,2-Difluoro-1-hydroxy-2-{2-methyl-1-[(p...)
Affinity DataIC50: 730nMAssay Description:Inhibition of human plasma reninMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2012
Entry Details Article
PubMed
TargetCathepsin D(Bovine)
TBA

Curated by ChEMBL
LigandPNGBDBM50024145({1-[1-(1-Cyclohexylmethyl-3,3-difluoro-3-{2-methyl...)
Affinity DataIC50: 1.70E+3nMAssay Description:Compound was tested for inhibition of bovine cathepsin DMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2012
Entry Details Article
PubMed
TargetRenin(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM912(PEPSTATIN | Pepstatine | N-[(3-Methyl-1-oxobutyl)-...)
Affinity DataIC50: 6.00E+3nMAssay Description:Inhibition of human plasma reninMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2012
Entry Details Article
PubMed
TargetRenin(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50022851(Pro-His-Pro-Phe-His-Phe-Phe-Val-Tyr-Lys | CHEMBL41...)
Affinity DataIC50: 9.40E+3nMAssay Description:Compound was tested for inhibition of human plasma renin.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2012
Entry Details Article
PubMed
TargetAngiotensin-converting enzyme(Rabbit)
TBA

Curated by ChEMBL
LigandPNGBDBM50022851(Pro-His-Pro-Phe-His-Phe-Phe-Val-Tyr-Lys | CHEMBL41...)
Affinity DataIC50: 1.20E+4nMAssay Description:Compound was tested for inhibition of Angiotensin I converting enzyme from rabbit lung.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2012
Entry Details Article
PubMed
TargetPepsin A(Pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50024145({1-[1-(1-Cyclohexylmethyl-3,3-difluoro-3-{2-methyl...)
Affinity DataIC50: 4.20E+4nMAssay Description:Compound was tested for inhibition of porcine pepsinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2012
Entry Details Article
PubMed