Compile Data Set for Download or QSAR
Report error Found 26 Enz. Inhib. hit(s) with all data for entry = 50017149
TargetCholecystokinin receptor type A(Human)
Jiangsu Normal University

Curated by ChEMBL
LigandPNGBDBM50600024(CHEMBL5182331)
Affinity DataEC50:  0.830nMAssay Description:Agonist activity at human CCK1R expressed in HEK293 cells assessed as ERK1/2 phosphorylation incubated for 5 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetGlucagon-like peptide 1 receptor(Human)
Jiangsu Normal University

Curated by ChEMBL
LigandPNGBDBM50600024(CHEMBL5182331)
Affinity DataEC50:  0.0570nMAssay Description:Agonist activity at human GLP-1R expressed in CHO cells assessed as cAMP release incubated for 20 min by HTRF analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetGlucagon-like peptide 1 receptor(Human)
Jiangsu Normal University

Curated by ChEMBL
LigandPNGBDBM50600022(CHEMBL5181266)
Affinity DataEC50:  0.110nMAssay Description:Agonist activity at human GLP-1R expressed in CHO cells assessed as cAMP release incubated for 20 min by HTRF analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetGastrin/cholecystokinin type B receptor(Human)
Jiangsu Normal University

Curated by ChEMBL
LigandPNGBDBM50600026(CHEMBL5177923)
Affinity DataEC50:  2.40nMAssay Description:Agonist activity at human CCK2R expressed in HEK293 cells assessed as ERK1/2 phosphorylation incubated for 5 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetGastrin/cholecystokinin type B receptor(Human)
Jiangsu Normal University

Curated by ChEMBL
LigandPNGBDBM50600025(CHEMBL5182775)
Affinity DataEC50: >100nMAssay Description:Agonist activity at human CCK2R expressed in HEK293 cells assessed as ERK1/2 phosphorylation incubated for 5 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetGastrin/cholecystokinin type B receptor(Human)
Jiangsu Normal University

Curated by ChEMBL
LigandPNGBDBM50600024(CHEMBL5182331)
Affinity DataEC50: >100nMAssay Description:Agonist activity at human CCK2R expressed in HEK293 cells assessed as ERK1/2 phosphorylation incubated for 5 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetGastrin/cholecystokinin type B receptor(Human)
Jiangsu Normal University

Curated by ChEMBL
LigandPNGBDBM50600023(CHEMBL5182323)
Affinity DataEC50: >100nMAssay Description:Agonist activity at human CCK2R expressed in HEK293 cells assessed as ERK1/2 phosphorylation incubated for 5 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetGastrin/cholecystokinin type B receptor(Human)
Jiangsu Normal University

Curated by ChEMBL
LigandPNGBDBM50600022(CHEMBL5181266)
Affinity DataEC50: >100nMAssay Description:Agonist activity at human CCK2R expressed in HEK293 cells assessed as ERK1/2 phosphorylation incubated for 5 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetGastrin/cholecystokinin type B receptor(Human)
Jiangsu Normal University

Curated by ChEMBL
LigandPNGBDBM50600021(CHEMBL5185239)
Affinity DataEC50: >100nMAssay Description:Agonist activity at human CCK2R expressed in HEK293 cells assessed as ERK1/2 phosphorylation incubated for 5 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetGastrin/cholecystokinin type B receptor(Human)
Jiangsu Normal University

Curated by ChEMBL
LigandPNGBDBM50600020(CHEMBL5182173)
Affinity DataEC50: >100nMAssay Description:Agonist activity at human CCK2R expressed in HEK293 cells assessed as ERK1/2 phosphorylation incubated for 5 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetGastrin/cholecystokinin type B receptor(Human)
Jiangsu Normal University

Curated by ChEMBL
LigandPNGBDBM50517333(CHEMBL4440419)
Affinity DataEC50: >100nMAssay Description:Agonist activity at human CCK2R expressed in HEK293 cells assessed as ERK1/2 phosphorylation incubated for 5 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetCholecystokinin receptor type A(Human)
Jiangsu Normal University

Curated by ChEMBL
LigandPNGBDBM50600026(CHEMBL5177923)
Affinity DataEC50: >100nMAssay Description:Agonist activity at human CCK1R expressed in HEK293 cells assessed as ERK1/2 phosphorylation incubated for 5 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetCholecystokinin receptor type A(Human)
Jiangsu Normal University

Curated by ChEMBL
LigandPNGBDBM50600025(CHEMBL5182775)
Affinity DataEC50:  1nMAssay Description:Agonist activity at human CCK1R expressed in HEK293 cells assessed as ERK1/2 phosphorylation incubated for 5 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetGlucagon-like peptide 1 receptor(Human)
Jiangsu Normal University

Curated by ChEMBL
LigandPNGBDBM50152769(GLP-1(7-36)-NH2 | NH2-HAEGTFTSDVSSYLEGQAAKEFIAWLVK...)
Affinity DataEC50:  0.0840nMAssay Description:Agonist activity at human GLP-1R expressed in HEK293 cells assessed as cAMP release incubated for 20 min by HTRF analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetCholecystokinin receptor type A(Human)
Jiangsu Normal University

Curated by ChEMBL
LigandPNGBDBM50600023(CHEMBL5182323)
Affinity DataEC50:  1.20nMAssay Description:Agonist activity at human CCK1R expressed in HEK293 cells assessed as ERK1/2 phosphorylation incubated for 5 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetCholecystokinin receptor type A(Human)
Jiangsu Normal University

Curated by ChEMBL
LigandPNGBDBM50600022(CHEMBL5181266)
Affinity DataEC50:  1.30nMAssay Description:Agonist activity at human CCK1R expressed in HEK293 cells assessed as ERK1/2 phosphorylation incubated for 5 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetCholecystokinin receptor type A(Human)
Jiangsu Normal University

Curated by ChEMBL
LigandPNGBDBM50600021(CHEMBL5185239)
Affinity DataEC50:  0.950nMAssay Description:Agonist activity at human CCK1R expressed in HEK293 cells assessed as ERK1/2 phosphorylation incubated for 5 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetCholecystokinin receptor type A(Human)
Jiangsu Normal University

Curated by ChEMBL
LigandPNGBDBM50600020(CHEMBL5182173)
Affinity DataEC50:  1.10nMAssay Description:Agonist activity at human CCK1R expressed in HEK293 cells assessed as ERK1/2 phosphorylation incubated for 5 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetCholecystokinin receptor type A(Human)
Jiangsu Normal University

Curated by ChEMBL
LigandPNGBDBM50517333(CHEMBL4440419)
Affinity DataEC50:  0.210nMAssay Description:Agonist activity at human CCK1R expressed in HEK293 cells assessed as ERK1/2 phosphorylation incubated for 5 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetGlucagon-like peptide 1 receptor(Human)
Jiangsu Normal University

Curated by ChEMBL
LigandPNGBDBM50600025(CHEMBL5182775)
Affinity DataEC50:  0.310nMAssay Description:Agonist activity at human GLP-1R expressed in HEK293 cells assessed as cAMP release incubated for 20 min by HTRF analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetGlucagon-like peptide 1 receptor(Human)
Jiangsu Normal University

Curated by ChEMBL
LigandPNGBDBM50600024(CHEMBL5182331)
Affinity DataEC50:  0.0740nMAssay Description:Agonist activity at human GLP-1R expressed in HEK293 cells assessed as cAMP release incubated for 20 min by HTRF analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetGlucagon-like peptide 1 receptor(Human)
Jiangsu Normal University

Curated by ChEMBL
LigandPNGBDBM50600023(CHEMBL5182323)
Affinity DataEC50:  0.520nMAssay Description:Agonist activity at human GLP-1R expressed in HEK293 cells assessed as cAMP release incubated for 20 min by HTRF analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetGlucagon-like peptide 1 receptor(Human)
Jiangsu Normal University

Curated by ChEMBL
LigandPNGBDBM50600022(CHEMBL5181266)
Affinity DataEC50:  0.150nMAssay Description:Agonist activity at human GLP-1R expressed in HEK293 cells assessed as cAMP release incubated for 20 min by HTRF analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetGlucagon-like peptide 1 receptor(Human)
Jiangsu Normal University

Curated by ChEMBL
LigandPNGBDBM50600021(CHEMBL5185239)
Affinity DataEC50:  0.0920nMAssay Description:Agonist activity at human GLP-1R expressed in HEK293 cells assessed as cAMP release incubated for 20 min by HTRF analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetGlucagon-like peptide 1 receptor(Human)
Jiangsu Normal University

Curated by ChEMBL
LigandPNGBDBM50600020(CHEMBL5182173)
Affinity DataEC50:  0.160nMAssay Description:Agonist activity at human GLP-1R expressed in HEK293 cells assessed as cAMP release incubated for 20 min by HTRF analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetGlucagon-like peptide 1 receptor(Human)
Jiangsu Normal University

Curated by ChEMBL
LigandPNGBDBM50600019(CHEMBL5205878)
Affinity DataEC50:  0.0560nMAssay Description:Agonist activity at human GLP-1R expressed in HEK293 cells assessed as cAMP release incubated for 20 min by HTRF analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed