Compile Data Set for Download or QSAR
Report error Found 7 Enz. Inhib. hit(s) with all data for entry = 50015727
TargetTyrosine-protein kinase receptor UFO(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50589184(CHEMBL5177673)
Affinity DataIC50: 12nMAssay Description:Inhibition of AXL (unknown origin) using peptide substrate in presence of ATP by radiometric HotSpot assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/18/2023
Entry Details
PubMed
TargetTyrosine-protein kinase ABL1(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM332700(US10196378, Compound C03)
Affinity DataIC50: 16nMAssay Description:Inhibition of NanoLuc-tagged ABL1 wild type (unknown origin) expressed in HEK293 cells by NanoBRET TE assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/18/2023
Entry Details
PubMed
TargetTyrosine-protein kinase ABL1(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM332702(US10196378, Compound C05)
Affinity DataIC50: 38nMAssay Description:Inhibition of NanoLuc-tagged ABL1 wild type (unknown origin) expressed in HEK293 cells by NanoBRET TE assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/18/2023
Entry Details
PubMed
TargetTyrosine-protein kinase ABL1(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM332705(US10196378, Compound C08)
Affinity DataIC50: 65nMAssay Description:Inhibition of NanoLuc-tagged ABL1 wild type (unknown origin) expressed in HEK293 cells by NanoBRET TE assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/18/2023
Entry Details
PubMed
TargetTyrosine-protein kinase ABL1(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50589184(CHEMBL5177673)
Affinity DataIC50: 345nMAssay Description:Inhibition of NanoLuc-tagged ABL1 wild type (unknown origin) expressed in HEK293 cells by NanoBRET TE assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/18/2023
Entry Details
PubMed
TargetTyrosine-protein kinase ABL1(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM332703(US10196378, Compound C06)
Affinity DataIC50: 637nMAssay Description:Inhibition of NanoLuc-tagged ABL1 wild type (unknown origin) expressed in HEK293 cells by NanoBRET TE assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/18/2023
Entry Details
PubMed
TargetTyrosine-protein kinase ABL1(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM332706(US10196378, Compound C10 | US10196378, Compound C0...)
Affinity DataIC50: 719nMAssay Description:Inhibition of NanoLuc-tagged ABL1 wild type (unknown origin) expressed in HEK293 cells by NanoBRET TE assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/18/2023
Entry Details
PubMed