Compile Data Set for Download or QSAR
Report error Found 29 Enz. Inhib. hit(s) with all data for entry = 50017137
Target5'-nucleotidase(Human)
The Second Military Medical University

Curated by ChEMBL
LigandPNGBDBM50599943(CHEMBL5177276)
Affinity DataIC50: 1.39E+3nMAssay Description:Inhibition of human CD73 assessed as reduction in inorganic phosphate release upon substrate hydrolysis using AMP/ATP as substrate incubated for 1 hr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
Target5'-nucleotidase(Human)
The Second Military Medical University

Curated by ChEMBL
LigandPNGBDBM18136(alpha, beta-methyleneadenosine 5 -diphosphate | ci...)
Affinity DataIC50: 3.97E+3nMAssay Description:Inhibition of human CD73 assessed as reduction in inorganic phosphate release upon substrate hydrolysis using AMP/ATP as substrate incubated for 1 hr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
Target5'-nucleotidase(Mouse)
The Second Military Medical University

Curated by ChEMBL
LigandPNGBDBM18136(alpha, beta-methyleneadenosine 5 -diphosphate | ci...)
Affinity DataIC50: 4.63E+3nMAssay Description:Inhibition of mouse CD73 assessed as reduction in inorganic phosphate release upon substrate hydrolysis using AMP/ATP as substrate incubated for 1 hr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
Target5'-nucleotidase(Human)
The Second Military Medical University

Curated by ChEMBL
LigandPNGBDBM50599941(CHEMBL5190085)
Affinity DataIC50: 5.69E+3nMAssay Description:Inhibition of human CD73 assessed as reduction in inorganic phosphate release upon substrate hydrolysis using AMP/ATP as substrate incubated for 1 hr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
Target5'-nucleotidase(Human)
The Second Military Medical University

Curated by ChEMBL
LigandPNGBDBM23208(cid_64971 | CHEMBL269277 | (1R,2R,5S,8R,9R,10R,13R...)
Affinity DataIC50: 7.28E+3nMAssay Description:Inhibition of human CD73 assessed as reduction in inorganic phosphate release upon substrate hydrolysis using AMP/ATP as substrate incubated for 1 hr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
Target5'-nucleotidase(Mouse)
The Second Military Medical University

Curated by ChEMBL
LigandPNGBDBM50599943(CHEMBL5177276)
Affinity DataIC50: 1.47E+4nMAssay Description:Inhibition of mouse CD73 assessed as reduction in inorganic phosphate release upon substrate hydrolysis using AMP/ATP as substrate incubated for 1 hr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
Target5'-nucleotidase(Human)
The Second Military Medical University

Curated by ChEMBL
LigandPNGBDBM50599939(CHEMBL5185215)
Affinity DataIC50: 1.68E+4nMAssay Description:Inhibition of human CD73 assessed as reduction in inorganic phosphate release upon substrate hydrolysis using AMP/ATP as substrate incubated for 1 hr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
Target5'-nucleotidase(Human)
The Second Military Medical University

Curated by ChEMBL
LigandPNGBDBM23207((1R,2R,5S,8R,9R,10R,13R,14R,17S,19R)-5-(hydroxymet...)
Affinity DataIC50: 2.27E+4nMAssay Description:Inhibition of human CD73 assessed as reduction in inorganic phosphate release upon substrate hydrolysis using AMP/ATP as substrate incubated for 1 hr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
Target5'-nucleotidase(Mouse)
The Second Military Medical University

Curated by ChEMBL
LigandPNGBDBM50599939(CHEMBL5185215)
Affinity DataIC50: 3.36E+4nMAssay Description:Inhibition of mouse CD73 assessed as reduction in inorganic phosphate release upon substrate hydrolysis using AMP/ATP as substrate incubated for 1 hr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
Target5'-nucleotidase(Human)
The Second Military Medical University

Curated by ChEMBL
LigandPNGBDBM50599942(CHEMBL5207600)
Affinity DataIC50: 3.72E+4nMAssay Description:Inhibition of human CD73 assessed as reduction in inorganic phosphate release upon substrate hydrolysis using AMP/ATP as substrate incubated for 1 hr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
Target5'-nucleotidase(Human)
The Second Military Medical University

Curated by ChEMBL
LigandPNGBDBM50240499((1R,3aS,5aR,5bR,11aR)-1-Isopropenyl-5a,5b,8,8,11a-...)
Affinity DataIC50: 4.33E+4nMAssay Description:Inhibition of human CD73 assessed as reduction in inorganic phosphate release upon substrate hydrolysis using AMP/ATP as substrate incubated for 1 hr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
Target5'-nucleotidase(Mouse)
The Second Military Medical University

Curated by ChEMBL
LigandPNGBDBM50599941(CHEMBL5190085)
Affinity DataIC50: 5.90E+4nMAssay Description:Inhibition of mouse CD73 assessed as reduction in inorganic phosphate release upon substrate hydrolysis using AMP/ATP as substrate incubated for 1 hr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
Target5'-nucleotidase(Mouse)
The Second Military Medical University

Curated by ChEMBL
LigandPNGBDBM23208(cid_64971 | CHEMBL269277 | (1R,2R,5S,8R,9R,10R,13R...)
Affinity DataIC50: 6.88E+4nMAssay Description:Inhibition of mouse CD73 assessed as reduction in inorganic phosphate release upon substrate hydrolysis using AMP/ATP as substrate incubated for 1 hr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
Target5'-nucleotidase(Human)
The Second Military Medical University

Curated by ChEMBL
LigandPNGBDBM50599940(CHEMBL5207447)
Affinity DataIC50: 8.14E+4nMAssay Description:Inhibition of human CD73 assessed as reduction in inorganic phosphate release upon substrate hydrolysis using AMP/ATP as substrate incubated for 1 hr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
Target5'-nucleotidase(Human)
The Second Military Medical University

Curated by ChEMBL
LigandPNGBDBM50599944(CHEMBL5187845)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human CD73 assessed as reduction in inorganic phosphate release upon substrate hydrolysis using AMP/ATP as substrate incubated for 1 hr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
Target5'-nucleotidase(Mouse)
The Second Military Medical University

Curated by ChEMBL
LigandPNGBDBM50599940(CHEMBL5207447)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of mouse CD73 assessed as reduction in inorganic phosphate release upon substrate hydrolysis using AMP/ATP as substrate incubated for 1 hr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
Target5'-nucleotidase(Mouse)
The Second Military Medical University

Curated by ChEMBL
LigandPNGBDBM50599942(CHEMBL5207600)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of mouse CD73 assessed as reduction in inorganic phosphate release upon substrate hydrolysis using AMP/ATP as substrate incubated for 1 hr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
Target5'-nucleotidase(Mouse)
The Second Military Medical University

Curated by ChEMBL
LigandPNGBDBM50599944(CHEMBL5187845)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of mouse CD73 assessed as reduction in inorganic phosphate release upon substrate hydrolysis using AMP/ATP as substrate incubated for 1 hr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
Target5'-nucleotidase(Mouse)
The Second Military Medical University

Curated by ChEMBL
LigandPNGBDBM50599945(CHEMBL5170520)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of mouse CD73 assessed as reduction in inorganic phosphate release upon substrate hydrolysis using AMP/ATP as substrate incubated for 1 hr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
Target5'-nucleotidase(Mouse)
The Second Military Medical University

Curated by ChEMBL
LigandPNGBDBM50599938(CHEMBL5170776)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of mouse CD73 assessed as reduction in inorganic phosphate release upon substrate hydrolysis using AMP/ATP as substrate incubated for 1 hr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
Target5'-nucleotidase(Mouse)
The Second Military Medical University

Curated by ChEMBL
LigandPNGBDBM50599937(CHEMBL5177221)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of mouse CD73 assessed as reduction in inorganic phosphate release upon substrate hydrolysis using AMP/ATP as substrate incubated for 1 hr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
Target5'-nucleotidase(Mouse)
The Second Military Medical University

Curated by ChEMBL
LigandPNGBDBM50599936(CHEMBL5191234)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of mouse CD73 assessed as reduction in inorganic phosphate release upon substrate hydrolysis using AMP/ATP as substrate incubated for 1 hr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
Target5'-nucleotidase(Human)
The Second Military Medical University

Curated by ChEMBL
LigandPNGBDBM50599945(CHEMBL5170520)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human CD73 assessed as reduction in inorganic phosphate release upon substrate hydrolysis using AMP/ATP as substrate incubated for 1 hr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
Target5'-nucleotidase(Human)
The Second Military Medical University

Curated by ChEMBL
LigandPNGBDBM50599938(CHEMBL5170776)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human CD73 assessed as reduction in inorganic phosphate release upon substrate hydrolysis using AMP/ATP as substrate incubated for 1 hr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
Target5'-nucleotidase(Human)
The Second Military Medical University

Curated by ChEMBL
LigandPNGBDBM50599937(CHEMBL5177221)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human CD73 assessed as reduction in inorganic phosphate release upon substrate hydrolysis using AMP/ATP as substrate incubated for 1 hr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
Target5'-nucleotidase(Human)
The Second Military Medical University

Curated by ChEMBL
LigandPNGBDBM50599936(CHEMBL5191234)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human CD73 assessed as reduction in inorganic phosphate release upon substrate hydrolysis using AMP/ATP as substrate incubated for 1 hr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
Target5'-nucleotidase(Human)
The Second Military Medical University

Curated by ChEMBL
LigandPNGBDBM23209((1R,2R,5S,8R,9R,10R,13R,14R,17S,18R,19R)-17-hydrox...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human CD73 assessed as reduction in inorganic phosphate release upon substrate hydrolysis using AMP/ATP as substrate incubated for 1 hr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
Target5'-nucleotidase(Human)
The Second Military Medical University

Curated by ChEMBL
LigandPNGBDBM50599935(Betulin Aldehyde | Betulinaldehyde | BETULINALDEHY...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human CD73 assessed as reduction in inorganic phosphate release upon substrate hydrolysis using AMP/ATP as substrate incubated for 1 hr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
Target5'-nucleotidase(Human)
The Second Military Medical University

Curated by ChEMBL
LigandPNGBDBM18136(alpha, beta-methyleneadenosine 5 -diphosphate | ci...)
Affinity DataKi:  88nMAssay Description:Inhibition of CD73 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed