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Report error Found 72 Enz. Inhib. hit(s) with all data for entry = 50017653
TargetCarbonic anhydrase 12(Human)
Tanta University

Curated by ChEMBL
LigandPNGBDBM10880(Acetazolamide, AAZ | AZA2 | CHEMBL20 | Acetazolami...)
Affinity DataKi:  5.70nMAssay Description:Inhibition of recombinant human CA 12 preincubated for 15 mins by phenol red dye based stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetCarbonic anhydrase 12(Human)
Tanta University

Curated by ChEMBL
LigandPNGBDBM50603710(CHEMBL5174617)
Affinity DataKi:  8.20nMAssay Description:Inhibition of recombinant human CA 12 preincubated for 15 mins by phenol red dye based stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetCarbonic anhydrase 12(Human)
Tanta University

Curated by ChEMBL
LigandPNGBDBM50603707(CHEMBL5186966)
Affinity DataKi:  8.5nMAssay Description:Inhibition of recombinant human CA 12 preincubated for 15 mins by phenol red dye based stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetCarbonic anhydrase 12(Human)
Tanta University

Curated by ChEMBL
LigandPNGBDBM50603713(CHEMBL5186050)
Affinity DataKi:  8.5nMAssay Description:Inhibition of recombinant human CA 12 preincubated for 15 mins by phenol red dye based stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetCarbonic anhydrase 12(Human)
Tanta University

Curated by ChEMBL
LigandPNGBDBM50603720(CHEMBL5182616)
Affinity DataKi:  8.70nMAssay Description:Inhibition of recombinant human CA 12 preincubated for 15 mins by phenol red dye based stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetCarbonic anhydrase 12(Human)
Tanta University

Curated by ChEMBL
LigandPNGBDBM50603714(CHEMBL5182270)
Affinity DataKi:  8.80nMAssay Description:Inhibition of recombinant human CA 12 preincubated for 15 mins by phenol red dye based stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetCarbonic anhydrase 12(Human)
Tanta University

Curated by ChEMBL
LigandPNGBDBM50603708(CHEMBL5194622)
Affinity DataKi:  8.90nMAssay Description:Inhibition of recombinant human CA 12 preincubated for 15 mins by phenol red dye based stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetCarbonic anhydrase 12(Human)
Tanta University

Curated by ChEMBL
LigandPNGBDBM50603711(CHEMBL5184758)
Affinity DataKi:  9.20nMAssay Description:Inhibition of recombinant human CA 12 preincubated for 15 mins by phenol red dye based stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetCarbonic anhydrase 12(Human)
Tanta University

Curated by ChEMBL
LigandPNGBDBM50603709(CHEMBL5181787)
Affinity DataKi:  9.40nMAssay Description:Inhibition of recombinant human CA 12 preincubated for 15 mins by phenol red dye based stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetCarbonic anhydrase 12(Human)
Tanta University

Curated by ChEMBL
LigandPNGBDBM50603712(CHEMBL5181015)
Affinity DataKi:  9.80nMAssay Description:Inhibition of recombinant human CA 12 preincubated for 15 mins by phenol red dye based stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetCarbonic anhydrase 2(Human)
Tanta University

Curated by ChEMBL
LigandPNGBDBM10880(Acetazolamide, AAZ | AZA2 | CHEMBL20 | Acetazolami...)
Affinity DataKi:  12nMAssay Description:Inhibition of recombinant human CA 2 preincubated for 15 mins by phenol red dye based stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetCarbonic anhydrase 9(Human)
Tanta University

Curated by ChEMBL
LigandPNGBDBM50603713(CHEMBL5186050)
Affinity DataKi:  13nMAssay Description:Inhibition of recombinant human CA 9 preincubated for 15 mins by phenol red dye based stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetCarbonic anhydrase 12(Human)
Tanta University

Curated by ChEMBL
LigandPNGBDBM50603722(CHEMBL5189506)
Affinity DataKi:  18nMAssay Description:Inhibition of recombinant human CA 12 preincubated for 15 mins by phenol red dye based stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetCarbonic anhydrase 9(Human)
Tanta University

Curated by ChEMBL
LigandPNGBDBM50603706(CHEMBL5190747)
Affinity DataKi:  23nMAssay Description:Inhibition of recombinant human CA 9 preincubated for 15 mins by phenol red dye based stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetCarbonic anhydrase 12(Human)
Tanta University

Curated by ChEMBL
LigandPNGBDBM50603718(CHEMBL5206040)
Affinity DataKi:  23nMAssay Description:Inhibition of recombinant human CA 12 preincubated for 15 mins by phenol red dye based stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetCarbonic anhydrase 12(Human)
Tanta University

Curated by ChEMBL
LigandPNGBDBM50603706(CHEMBL5190747)
Affinity DataKi:  24nMAssay Description:Inhibition of recombinant human CA 12 preincubated for 15 mins by phenol red dye based stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetCarbonic anhydrase 9(Human)
Tanta University

Curated by ChEMBL
LigandPNGBDBM10880(Acetazolamide, AAZ | AZA2 | CHEMBL20 | Acetazolami...)
Affinity DataKi:  25nMAssay Description:Inhibition of recombinant human CA 9 preincubated for 15 mins by phenol red dye based stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetCarbonic anhydrase 9(Human)
Tanta University

Curated by ChEMBL
LigandPNGBDBM50603718(CHEMBL5206040)
Affinity DataKi:  26nMAssay Description:Inhibition of recombinant human CA 9 preincubated for 15 mins by phenol red dye based stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetCarbonic anhydrase 9(Human)
Tanta University

Curated by ChEMBL
LigandPNGBDBM50603716(CHEMBL5203064)
Affinity DataKi:  27nMAssay Description:Inhibition of recombinant human CA 9 preincubated for 15 mins by phenol red dye based stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetCarbonic anhydrase 9(Human)
Tanta University

Curated by ChEMBL
LigandPNGBDBM50603710(CHEMBL5174617)
Affinity DataKi:  27nMAssay Description:Inhibition of recombinant human CA 9 preincubated for 15 mins by phenol red dye based stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetCarbonic anhydrase 9(Human)
Tanta University

Curated by ChEMBL
LigandPNGBDBM50603715(CHEMBL5173544)
Affinity DataKi:  28nMAssay Description:Inhibition of recombinant human CA 9 preincubated for 15 mins by phenol red dye based stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetCarbonic anhydrase 9(Human)
Tanta University

Curated by ChEMBL
LigandPNGBDBM50603721(CHEMBL5194072)
Affinity DataKi:  29nMAssay Description:Inhibition of recombinant human CA 9 preincubated for 15 mins by phenol red dye based stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetCarbonic anhydrase 9(Human)
Tanta University

Curated by ChEMBL
LigandPNGBDBM50603714(CHEMBL5182270)
Affinity DataKi:  29nMAssay Description:Inhibition of recombinant human CA 9 preincubated for 15 mins by phenol red dye based stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetCarbonic anhydrase 9(Human)
Tanta University

Curated by ChEMBL
LigandPNGBDBM50603708(CHEMBL5194622)
Affinity DataKi:  30nMAssay Description:Inhibition of recombinant human CA 9 preincubated for 15 mins by phenol red dye based stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetCarbonic anhydrase 9(Human)
Tanta University

Curated by ChEMBL
LigandPNGBDBM50603709(CHEMBL5181787)
Affinity DataKi:  30nMAssay Description:Inhibition of recombinant human CA 9 preincubated for 15 mins by phenol red dye based stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetCarbonic anhydrase 9(Human)
Tanta University

Curated by ChEMBL
LigandPNGBDBM50603712(CHEMBL5181015)
Affinity DataKi:  32nMAssay Description:Inhibition of recombinant human CA 9 preincubated for 15 mins by phenol red dye based stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetCarbonic anhydrase 12(Human)
Tanta University

Curated by ChEMBL
LigandPNGBDBM50603715(CHEMBL5173544)
Affinity DataKi:  32nMAssay Description:Inhibition of recombinant human CA 12 preincubated for 15 mins by phenol red dye based stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetCarbonic anhydrase 9(Human)
Tanta University

Curated by ChEMBL
LigandPNGBDBM50603707(CHEMBL5186966)
Affinity DataKi:  61nMAssay Description:Inhibition of recombinant human CA 9 preincubated for 15 mins by phenol red dye based stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetCarbonic anhydrase 12(Human)
Tanta University

Curated by ChEMBL
LigandPNGBDBM50603717(CHEMBL5182583)
Affinity DataKi:  70nMAssay Description:Inhibition of recombinant human CA 12 preincubated for 15 mins by phenol red dye based stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetCarbonic anhydrase 12(Human)
Tanta University

Curated by ChEMBL
LigandPNGBDBM50603716(CHEMBL5203064)
Affinity DataKi:  71nMAssay Description:Inhibition of recombinant human CA 12 preincubated for 15 mins by phenol red dye based stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetCarbonic anhydrase 12(Human)
Tanta University

Curated by ChEMBL
LigandPNGBDBM50603719(CHEMBL5176338)
Affinity DataKi:  77nMAssay Description:Inhibition of recombinant human CA 12 preincubated for 15 mins by phenol red dye based stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetCarbonic anhydrase 12(Human)
Tanta University

Curated by ChEMBL
LigandPNGBDBM50603721(CHEMBL5194072)
Affinity DataKi:  82nMAssay Description:Inhibition of recombinant human CA 12 preincubated for 15 mins by phenol red dye based stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetCarbonic anhydrase 2(Human)
Tanta University

Curated by ChEMBL
LigandPNGBDBM50603713(CHEMBL5186050)
Affinity DataKi:  84nMAssay Description:Inhibition of recombinant human CA 2 preincubated for 15 mins by phenol red dye based stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetCarbonic anhydrase 2(Human)
Tanta University

Curated by ChEMBL
LigandPNGBDBM50603716(CHEMBL5203064)
Affinity DataKi:  89nMAssay Description:Inhibition of recombinant human CA 2 preincubated for 15 mins by phenol red dye based stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetCarbonic anhydrase 9(Human)
Tanta University

Curated by ChEMBL
LigandPNGBDBM50603711(CHEMBL5184758)
Affinity DataKi:  99nMAssay Description:Inhibition of recombinant human CA 9 preincubated for 15 mins by phenol red dye based stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetCarbonic anhydrase 2(Human)
Tanta University

Curated by ChEMBL
LigandPNGBDBM50603718(CHEMBL5206040)
Affinity DataKi:  131nMAssay Description:Inhibition of recombinant human CA 2 preincubated for 15 mins by phenol red dye based stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetCarbonic anhydrase 9(Human)
Tanta University

Curated by ChEMBL
LigandPNGBDBM50603720(CHEMBL5182616)
Affinity DataKi:  207nMAssay Description:Inhibition of recombinant human CA 9 preincubated for 15 mins by phenol red dye based stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetCarbonic anhydrase 2(Human)
Tanta University

Curated by ChEMBL
LigandPNGBDBM50603707(CHEMBL5186966)
Affinity DataKi:  210nMAssay Description:Inhibition of recombinant human CA 2 preincubated for 15 mins by phenol red dye based stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetCarbonic anhydrase 9(Human)
Tanta University

Curated by ChEMBL
LigandPNGBDBM50603722(CHEMBL5189506)
Affinity DataKi:  233nMAssay Description:Inhibition of recombinant human CA 9 preincubated for 15 mins by phenol red dye based stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetCarbonic anhydrase 1(Human)
Tanta University

Curated by ChEMBL
LigandPNGBDBM10880(Acetazolamide, AAZ | AZA2 | CHEMBL20 | Acetazolami...)
Affinity DataKi:  250nMAssay Description:Inhibition of recombinant human CA 1 preincubated for 15 mins by phenol red dye based stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetCarbonic anhydrase 9(Human)
Tanta University

Curated by ChEMBL
LigandPNGBDBM50603717(CHEMBL5182583)
Affinity DataKi:  255nMAssay Description:Inhibition of recombinant human CA 9 preincubated for 15 mins by phenol red dye based stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetCarbonic anhydrase 9(Human)
Tanta University

Curated by ChEMBL
LigandPNGBDBM50603719(CHEMBL5176338)
Affinity DataKi:  259nMAssay Description:Inhibition of recombinant human CA 9 preincubated for 15 mins by phenol red dye based stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetCarbonic anhydrase 2(Human)
Tanta University

Curated by ChEMBL
LigandPNGBDBM50603717(CHEMBL5182583)
Affinity DataKi:  289nMAssay Description:Inhibition of recombinant human CA 2 preincubated for 15 mins by phenol red dye based stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetCarbonic anhydrase 2(Human)
Tanta University

Curated by ChEMBL
LigandPNGBDBM50603719(CHEMBL5176338)
Affinity DataKi:  367nMAssay Description:Inhibition of recombinant human CA 2 preincubated for 15 mins by phenol red dye based stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetCarbonic anhydrase 2(Human)
Tanta University

Curated by ChEMBL
LigandPNGBDBM50603706(CHEMBL5190747)
Affinity DataKi:  480nMAssay Description:Inhibition of recombinant human CA 2 preincubated for 15 mins by phenol red dye based stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetCarbonic anhydrase 2(Human)
Tanta University

Curated by ChEMBL
LigandPNGBDBM50603711(CHEMBL5184758)
Affinity DataKi:  543nMAssay Description:Inhibition of recombinant human CA 2 preincubated for 15 mins by phenol red dye based stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetCarbonic anhydrase 2(Human)
Tanta University

Curated by ChEMBL
LigandPNGBDBM50603721(CHEMBL5194072)
Affinity DataKi:  598nMAssay Description:Inhibition of recombinant human CA 2 preincubated for 15 mins by phenol red dye based stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetCarbonic anhydrase 1(Human)
Tanta University

Curated by ChEMBL
LigandPNGBDBM50603711(CHEMBL5184758)
Affinity DataKi:  602nMAssay Description:Inhibition of recombinant human CA 1 preincubated for 15 mins by phenol red dye based stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetCarbonic anhydrase 2(Human)
Tanta University

Curated by ChEMBL
LigandPNGBDBM50603714(CHEMBL5182270)
Affinity DataKi:  621nMAssay Description:Inhibition of recombinant human CA 2 preincubated for 15 mins by phenol red dye based stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetCarbonic anhydrase 1(Human)
Tanta University

Curated by ChEMBL
LigandPNGBDBM50603716(CHEMBL5203064)
Affinity DataKi:  622nMAssay Description:Inhibition of recombinant human CA 1 preincubated for 15 mins by phenol red dye based stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
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