Compile Data Set for Download or QSAR
Report error Found 37 Enz. Inhib. hit(s) with all data for entry = 50017110
TargetShort transient receptor potential channel 5(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50599832(CHEMBL5201831)
Affinity DataIC50: 14nMAssay Description:Inhibition of human TRPC5 channel expressed in HEK293 cells assessed as inhibition of EA-evoked channel current measured at +80 mV by whole-cell volt...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetShort transient receptor potential channel 5(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50529421(CHEMBL4530872)
Affinity DataIC50: 50nMAssay Description:Inhibition of human TRPC5 channel expressed in HEK293 cells assessed as inhibition of EA-evoked channel current measured at +80 mV by whole-cell volt...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetShort transient receptor potential channel 5(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50599832(CHEMBL5201831)
Affinity DataIC50: 60nMAssay Description:Inhibition of TRPC5 channel (unknown origin) expressed in HEK293 cells assessed as inhibition of EA-evoked Ca2+ entry by measuring reduction in intra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetShort transient receptor potential channel 4(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50599832(CHEMBL5201831)
Affinity DataIC50: 65nMAssay Description:Inhibition of TRPC4 channel (unknown origin) expressed in HEK293 cells assessed as inhibition of EA-evoked Ca2+ entry by measuring reduction in intra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetShort transient receptor potential channel 5(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50599839(CHEMBL5170160)
Affinity DataIC50: 111nMAssay Description:Inhibition of TRPC5 channel (unknown origin) expressed in HEK293 cells assessed as inhibition of EA-evoked Ca2+ entry by measuring reduction in intra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetShort transient receptor potential channel 5(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50599842(CHEMBL5187587)
Affinity DataIC50: 125nMAssay Description:Inhibition of TRPC5 channel (unknown origin) expressed in HEK293 cells assessed as inhibition of EA-evoked Ca2+ entry by measuring reduction in intra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetShort transient receptor potential channel 5(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50529421(CHEMBL4530872)
Affinity DataIC50: 211nMAssay Description:Inhibition of TRPC5 channel (unknown origin) expressed in HEK293 cells assessed as inhibition of EA-evoked Ca2+ entry by measuring reduction in intra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetShort transient receptor potential channel 5(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50599836(CHEMBL5201353)
Affinity DataIC50: 280nMAssay Description:Inhibition of TRPC5 channel (unknown origin) expressed in HEK293 cells assessed as inhibition of EA-evoked Ca2+ entry by measuring reduction in intra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetShort transient receptor potential channel 5(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50599833(CHEMBL5197504)
Affinity DataIC50: 314nMAssay Description:Inhibition of TRPC5 channel (unknown origin) expressed in HEK293 cells assessed as inhibition of EA-evoked Ca2+ entry by measuring reduction in intra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetShort transient receptor potential channel 5(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50599826(CHEMBL5203731)
Affinity DataIC50: 452nMAssay Description:Inhibition of TRPC5 channel (unknown origin) expressed in HEK293 cells assessed as inhibition of EA-evoked Ca2+ entry by measuring reduction in intra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetShort transient receptor potential channel 5(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50599837(CHEMBL5188705)
Affinity DataIC50: 629nMAssay Description:Inhibition of TRPC5 channel (unknown origin) expressed in HEK293 cells assessed as inhibition of EA-evoked Ca2+ entry by measuring reduction in intra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetShort transient receptor potential channel 5(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50599829(CHEMBL5175780)
Affinity DataIC50: 654nMAssay Description:Inhibition of TRPC5 channel (unknown origin) expressed in HEK293 cells assessed as inhibition of EA-evoked Ca2+ entry by measuring reduction in intra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetShort transient receptor potential channel 5(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50599835(CHEMBL5191955)
Affinity DataIC50: 664nMAssay Description:Inhibition of TRPC5 channel (unknown origin) expressed in HEK293 cells assessed as inhibition of EA-evoked Ca2+ entry by measuring reduction in intra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetShort transient receptor potential channel 5(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50599831(CHEMBL5177892)
Affinity DataIC50: 776nMAssay Description:Inhibition of TRPC5 channel (unknown origin) expressed in HEK293 cells assessed as inhibition of EA-evoked Ca2+ entry by measuring reduction in intra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetShort transient receptor potential channel 5(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50599843(CHEMBL5179669)
Affinity DataIC50: 798nMAssay Description:Inhibition of TRPC5 channel (unknown origin) expressed in HEK293 cells assessed as inhibition of EA-evoked Ca2+ entry by measuring reduction in intra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetShort transient receptor potential channel 5(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50599825(CHEMBL5198318)
Affinity DataIC50: 860nMAssay Description:Inhibition of TRPC5 channel (unknown origin) expressed in HEK293 cells assessed as inhibition of EA-evoked Ca2+ entry by measuring reduction in intra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetShort transient receptor potential channel 5(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50599824(CHEMBL5181130)
Affinity DataIC50: 955nMAssay Description:Inhibition of TRPC5 channel (unknown origin) expressed in HEK293 cells assessed as inhibition of EA-evoked Ca2+ entry by measuring reduction in intra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetShort transient receptor potential channel 5(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50599830(CHEMBL5188379)
Affinity DataIC50: 1.07E+3nMAssay Description:Inhibition of TRPC5 channel (unknown origin) expressed in HEK293 cells assessed as inhibition of EA-evoked Ca2+ entry by measuring reduction in intra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetShort transient receptor potential channel 5(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50599844(CHEMBL5206431)
Affinity DataIC50: 2.08E+3nMAssay Description:Inhibition of TRPC5 channel (unknown origin) expressed in HEK293 cells assessed as inhibition of EA-evoked Ca2+ entry by measuring reduction in intra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetShort transient receptor potential channel 5(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50599838(CHEMBL5172510)
Affinity DataIC50: 2.54E+3nMAssay Description:Inhibition of TRPC5 channel (unknown origin) expressed in HEK293 cells assessed as inhibition of EA-evoked Ca2+ entry by measuring reduction in intra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetShort transient receptor potential channel 5(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50599812(CHEMBL5200742)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of TRPC5 channel (unknown origin) expressed in HEK293 cells assessed as inhibition of EA-evoked Ca2+ entry by measuring reduction in intra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetShort transient receptor potential channel 5(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50599828(CHEMBL5198355)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of TRPC5 channel (unknown origin) expressed in HEK293 cells assessed as inhibition of EA-evoked Ca2+ entry by measuring reduction in intra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetShort transient receptor potential channel 5(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50599813(CHEMBL5173080)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of TRPC5 channel (unknown origin) expressed in HEK293 cells assessed as inhibition of EA-evoked Ca2+ entry by measuring reduction in intra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetShort transient receptor potential channel 5(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50599814(CHEMBL5191617)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of TRPC5 channel (unknown origin) expressed in HEK293 cells assessed as inhibition of EA-evoked Ca2+ entry by measuring reduction in intra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetShort transient receptor potential channel 5(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50599815(CHEMBL5174015)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of TRPC5 channel (unknown origin) expressed in HEK293 cells assessed as inhibition of EA-evoked Ca2+ entry by measuring reduction in intra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetShort transient receptor potential channel 5(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50599841(CHEMBL5185752)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of TRPC5 channel (unknown origin) expressed in HEK293 cells assessed as inhibition of EA-evoked Ca2+ entry by measuring reduction in intra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetShort transient receptor potential channel 5(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50599840(CHEMBL5209305)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of TRPC5 channel (unknown origin) expressed in HEK293 cells assessed as inhibition of EA-evoked Ca2+ entry by measuring reduction in intra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetShort transient receptor potential channel 5(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50599816(CHEMBL5204508)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of TRPC5 channel (unknown origin) expressed in HEK293 cells assessed as inhibition of EA-evoked Ca2+ entry by measuring reduction in intra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetShort transient receptor potential channel 5(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50599817(CHEMBL5192727)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of TRPC5 channel (unknown origin) expressed in HEK293 cells assessed as inhibition of EA-evoked Ca2+ entry by measuring reduction in intra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetShort transient receptor potential channel 5(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50599818(CHEMBL5205358)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of TRPC5 channel (unknown origin) expressed in HEK293 cells assessed as inhibition of EA-evoked Ca2+ entry by measuring reduction in intra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetShort transient receptor potential channel 5(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50599822(CHEMBL5187351)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of TRPC5 channel (unknown origin) expressed in HEK293 cells assessed as inhibition of EA-evoked Ca2+ entry by measuring reduction in intra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetShort transient receptor potential channel 5(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50599834(CHEMBL5202140)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of TRPC5 channel (unknown origin) expressed in HEK293 cells assessed as inhibition of EA-evoked Ca2+ entry by measuring reduction in intra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetShort transient receptor potential channel 5(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50599819(CHEMBL5187398)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of TRPC5 channel (unknown origin) expressed in HEK293 cells assessed as inhibition of EA-evoked Ca2+ entry by measuring reduction in intra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetShort transient receptor potential channel 5(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50599820(CHEMBL5178467)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of TRPC5 channel (unknown origin) expressed in HEK293 cells assessed as inhibition of EA-evoked Ca2+ entry by measuring reduction in intra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetShort transient receptor potential channel 5(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50599827(CHEMBL5175304)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of TRPC5 channel (unknown origin) expressed in HEK293 cells assessed as inhibition of EA-evoked Ca2+ entry by measuring reduction in intra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetShort transient receptor potential channel 5(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50599821(CHEMBL5208809)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of TRPC5 channel (unknown origin) expressed in HEK293 cells assessed as inhibition of EA-evoked Ca2+ entry by measuring reduction in intra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetShort transient receptor potential channel 5(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50599823(CHEMBL5197599)
Affinity DataIC50: 1.04E+4nMAssay Description:Inhibition of TRPC5 channel (unknown origin) expressed in HEK293 cells assessed as inhibition of EA-evoked Ca2+ entry by measuring reduction in intra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed