Compile Data Set for Download or QSAR
Report error Found 102 Enz. Inhib. hit(s) with all data for entry = 50015271
TargetNuclear factor erythroid 2-related factor 2(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50556867(CHEMBL4757224)
Affinity DataKd:  3.70E+3nMAssay Description:Inhibition of Keap1-Nrf2 (unknown origin) interaction assessed as dissociation constant by isothermal titration calorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2023
Entry Details Article
PubMed
TargetNuclear factor erythroid 2-related factor 2(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50584786(CHEMBL5089493)
Affinity DataKd:  1.00E+3nMAssay Description:Inhibition of Keap1-Nrf2 (unknown origin) interaction assessed as dissociation constant by isothermal titration calorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2023
Entry Details Article
PubMed
TargetNuclear factor erythroid 2-related factor 2(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50584787(CHEMBL5087800)
Affinity DataKd:  4.10E+3nMAssay Description:Inhibition of Keap1-Nrf2 (unknown origin) interaction assessed as dissociation constant by isothermal titration calorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2023
Entry Details Article
PubMed
TargetNuclear factor erythroid 2-related factor 2(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50584788(CHEMBL5094633)
Affinity DataKd:  1.60E+3nMAssay Description:Inhibition of Keap1-Nrf2 (unknown origin) interaction assessed as dissociation constant by isothermal titration calorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2023
Entry Details Article
PubMed
TargetNuclear factor erythroid 2-related factor 2(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50556867(CHEMBL4757224)
Affinity DataKd:  4.10E+3nMAssay Description:Inhibition of Keap1-Nrf2 (unknown origin) interaction assessed as dissociation constant by surface plasmon resonance based inhibition-in-solution ass...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2023
Entry Details Article
PubMed
TargetNuclear factor erythroid 2-related factor 2(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50584786(CHEMBL5089493)
Affinity DataKd:  3.00E+3nMAssay Description:Inhibition of Keap1-Nrf2 (unknown origin) interaction assessed as dissociation constant by surface plasmon resonance based inhibition-in-solution ass...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2023
Entry Details Article
PubMed
TargetNuclear factor erythroid 2-related factor 2(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50584789(CHEMBL5080393)
Affinity DataKd:  8.60E+4nMAssay Description:Inhibition of Keap1-Nrf2 (unknown origin) interaction assessed as dissociation constant by surface plasmon resonance based inhibition-in-solution ass...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2023
Entry Details Article
PubMed
TargetNuclear factor erythroid 2-related factor 2(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50584790(CHEMBL5088719)
Affinity DataKd:  4.19E+5nMAssay Description:Inhibition of Keap1-Nrf2 (unknown origin) interaction assessed as dissociation constant by surface plasmon resonance based inhibition-in-solution ass...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2023
Entry Details Article
PubMed
TargetNuclear factor erythroid 2-related factor 2(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50584791(CHEMBL5092406)
Affinity DataKd: >5.00E+5nMAssay Description:Inhibition of Keap1-Nrf2 (unknown origin) interaction assessed as dissociation constant by surface plasmon resonance based inhibition-in-solution ass...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2023
Entry Details Article
PubMed
TargetNuclear factor erythroid 2-related factor 2(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50584792(CHEMBL5078590)
Affinity DataKd: >5.00E+5nMAssay Description:Inhibition of Keap1-Nrf2 (unknown origin) interaction assessed as dissociation constant by surface plasmon resonance based inhibition-in-solution ass...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2023
Entry Details Article
PubMed
TargetNuclear factor erythroid 2-related factor 2(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50584787(CHEMBL5087800)
Affinity DataKd:  9.30E+3nMAssay Description:Inhibition of Keap1-Nrf2 (unknown origin) interaction assessed as dissociation constant by surface plasmon resonance based inhibition-in-solution ass...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2023
Entry Details Article
PubMed
TargetNuclear factor erythroid 2-related factor 2(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50584793(CHEMBL5091283)
Affinity DataKd: >5.00E+5nMAssay Description:Inhibition of Keap1-Nrf2 (unknown origin) interaction assessed as dissociation constant by surface plasmon resonance based inhibition-in-solution ass...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2023
Entry Details Article
PubMed
TargetNuclear factor erythroid 2-related factor 2(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50584794(CHEMBL5082179)
Affinity DataKd: >5.00E+5nMAssay Description:Inhibition of Keap1-Nrf2 (unknown origin) interaction assessed as dissociation constant by surface plasmon resonance based inhibition-in-solution ass...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2023
Entry Details Article
PubMed
TargetNuclear factor erythroid 2-related factor 2(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50584795(CHEMBL5077207)
Affinity DataKd:  2.80E+4nMAssay Description:Inhibition of Keap1-Nrf2 (unknown origin) interaction assessed as dissociation constant by surface plasmon resonance based inhibition-in-solution ass...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2023
Entry Details Article
PubMed
TargetNuclear factor erythroid 2-related factor 2(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50584796(CHEMBL5094789)
Affinity DataKd:  4.81E+5nMAssay Description:Inhibition of Keap1-Nrf2 (unknown origin) interaction assessed as dissociation constant by surface plasmon resonance based inhibition-in-solution ass...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2023
Entry Details Article
PubMed
TargetNuclear factor erythroid 2-related factor 2(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50584788(CHEMBL5094633)
Affinity DataKd:  4.10E+3nMAssay Description:Inhibition of Keap1-Nrf2 (unknown origin) interaction assessed as dissociation constant by surface plasmon resonance based inhibition-in-solution ass...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2023
Entry Details Article
PubMed
TargetNuclear factor erythroid 2-related factor 2(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50584797(CHEMBL5090693)
Affinity DataKd:  3.40E+4nMAssay Description:Inhibition of Keap1-Nrf2 (unknown origin) interaction assessed as dissociation constant by surface plasmon resonance based inhibition-in-solution ass...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2023
Entry Details Article
PubMed
TargetNuclear factor erythroid 2-related factor 2(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50584798(CHEMBL5075731)
Affinity DataKd:  1.70E+4nMAssay Description:Inhibition of Keap1-Nrf2 (unknown origin) interaction assessed as dissociation constant by surface plasmon resonance based inhibition-in-solution ass...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2023
Entry Details Article
PubMed
TargetNuclear factor erythroid 2-related factor 2(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50584799(CHEMBL5087113)
Affinity DataKd:  2.04E+5nMAssay Description:Inhibition of Keap1-Nrf2 (unknown origin) interaction assessed as dissociation constant by surface plasmon resonance based inhibition-in-solution ass...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2023
Entry Details Article
PubMed
TargetNuclear factor erythroid 2-related factor 2(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50584800(CHEMBL5078177)
Affinity DataKd: >5.00E+5nMAssay Description:Inhibition of Keap1-Nrf2 (unknown origin) interaction assessed as dissociation constant by surface plasmon resonance based inhibition-in-solution ass...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2023
Entry Details Article
PubMed
TargetNuclear factor erythroid 2-related factor 2(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50584801(CHEMBL5091973)
Affinity DataKd:  2.90E+4nMAssay Description:Inhibition of Keap1-Nrf2 (unknown origin) interaction assessed as dissociation constant by surface plasmon resonance based inhibition-in-solution ass...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2023
Entry Details Article
PubMed
TargetNuclear factor erythroid 2-related factor 2(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50584802(CHEMBL5090725)
Affinity DataKd:  1.00E+4nMAssay Description:Inhibition of Keap1-Nrf2 (unknown origin) interaction assessed as dissociation constant by surface plasmon resonance based inhibition-in-solution ass...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2023
Entry Details Article
PubMed
TargetNuclear factor erythroid 2-related factor 2(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50584803(CHEMBL5080701)
Affinity DataKd:  1.60E+4nMAssay Description:Inhibition of Keap1-Nrf2 (unknown origin) interaction assessed as dissociation constant by surface plasmon resonance based inhibition-in-solution ass...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2023
Entry Details Article
PubMed
TargetNuclear factor erythroid 2-related factor 2(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50584804(CHEMBL5077431)
Affinity DataKd:  2.60E+4nMAssay Description:Inhibition of Keap1-Nrf2 (unknown origin) interaction assessed as dissociation constant by surface plasmon resonance based inhibition-in-solution ass...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2023
Entry Details Article
PubMed
TargetNuclear factor erythroid 2-related factor 2(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50584805(CHEMBL5079115)
Affinity DataKd: >5.00E+5nMAssay Description:Inhibition of Keap1-Nrf2 (unknown origin) interaction assessed as dissociation constant by surface plasmon resonance based inhibition-in-solution ass...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2023
Entry Details Article
PubMed
TargetNuclear factor erythroid 2-related factor 2(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50584806(CHEMBL5072745)
Affinity DataKd:  1.71E+5nMAssay Description:Inhibition of Keap1-Nrf2 (unknown origin) interaction assessed as dissociation constant by surface plasmon resonance based inhibition-in-solution ass...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2023
Entry Details Article
PubMed
TargetNuclear factor erythroid 2-related factor 2(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50584807(CHEMBL5076911)
Affinity DataKd:  3.16E+5nMAssay Description:Inhibition of Keap1-Nrf2 (unknown origin) interaction assessed as dissociation constant by surface plasmon resonance based inhibition-in-solution ass...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2023
Entry Details Article
PubMed
TargetNuclear factor erythroid 2-related factor 2(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50584808(CHEMBL5076160)
Affinity DataKd:  2.46E+5nMAssay Description:Inhibition of Keap1-Nrf2 (unknown origin) interaction assessed as dissociation constant by surface plasmon resonance based inhibition-in-solution ass...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2023
Entry Details Article
PubMed
TargetNuclear factor erythroid 2-related factor 2(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50584809(CHEMBL5085131)
Affinity DataKd:  2.60E+4nMAssay Description:Inhibition of Keap1-Nrf2 (unknown origin) interaction assessed as dissociation constant by surface plasmon resonance based inhibition-in-solution ass...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2023
Entry Details Article
PubMed
TargetNuclear factor erythroid 2-related factor 2(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50584810(CHEMBL5090715)
Affinity DataKd:  2.30E+4nMAssay Description:Inhibition of Keap1-Nrf2 (unknown origin) interaction assessed as dissociation constant by surface plasmon resonance based inhibition-in-solution ass...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2023
Entry Details Article
PubMed
TargetNuclear factor erythroid 2-related factor 2(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50584811(CHEMBL5093665)
Affinity DataKd:  1.30E+4nMAssay Description:Inhibition of Keap1-Nrf2 (unknown origin) interaction assessed as dissociation constant by surface plasmon resonance based inhibition-in-solution ass...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2023
Entry Details Article
PubMed
TargetNuclear factor erythroid 2-related factor 2(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50584812(CHEMBL5072541)
Affinity DataKd:  3.10E+4nMAssay Description:Inhibition of Keap1-Nrf2 (unknown origin) interaction assessed as dissociation constant by surface plasmon resonance based inhibition-in-solution ass...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2023
Entry Details Article
PubMed
TargetNuclear factor erythroid 2-related factor 2(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50584813(CHEMBL5089255)
Affinity DataKd:  1.00E+4nMAssay Description:Inhibition of Keap1-Nrf2 (unknown origin) interaction assessed as dissociation constant by surface plasmon resonance based inhibition-in-solution ass...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2023
Entry Details Article
PubMed
TargetNuclear factor erythroid 2-related factor 2(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50584814(CHEMBL5081080)
Affinity DataKd:  9.00E+3nMAssay Description:Inhibition of Keap1-Nrf2 (unknown origin) interaction assessed as dissociation constant by surface plasmon resonance based inhibition-in-solution ass...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2023
Entry Details Article
PubMed
TargetNuclear factor erythroid 2-related factor 2(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50584815(CHEMBL5086590)
Affinity DataKd:  2.00E+4nMAssay Description:Inhibition of Keap1-Nrf2 (unknown origin) interaction assessed as dissociation constant by surface plasmon resonance based inhibition-in-solution ass...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2023
Entry Details Article
PubMed
TargetNuclear factor erythroid 2-related factor 2(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50584816(CHEMBL5087038)
Affinity DataKd:  1.70E+4nMAssay Description:Inhibition of Keap1-Nrf2 (unknown origin) interaction assessed as dissociation constant by surface plasmon resonance based inhibition-in-solution ass...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2023
Entry Details Article
PubMed
TargetNuclear factor erythroid 2-related factor 2(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50584817(CHEMBL5085870)
Affinity DataKd:  1.30E+4nMAssay Description:Inhibition of Keap1-Nrf2 (unknown origin) interaction assessed as dissociation constant by surface plasmon resonance based inhibition-in-solution ass...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2023
Entry Details Article
PubMed
TargetNuclear factor erythroid 2-related factor 2(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50584818(CHEMBL5082507)
Affinity DataKd:  3.30E+4nMAssay Description:Inhibition of Keap1-Nrf2 (unknown origin) interaction assessed as dissociation constant by surface plasmon resonance based inhibition-in-solution ass...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2023
Entry Details Article
PubMed
TargetNuclear factor erythroid 2-related factor 2(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50584819(CHEMBL5085792)
Affinity DataKd:  1.10E+4nMAssay Description:Inhibition of Keap1-Nrf2 (unknown origin) interaction assessed as dissociation constant by surface plasmon resonance based inhibition-in-solution ass...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2023
Entry Details Article
PubMed
TargetNuclear factor erythroid 2-related factor 2(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50584820(CHEMBL5080311)
Affinity DataKd:  2.10E+4nMAssay Description:Inhibition of Keap1-Nrf2 (unknown origin) interaction assessed as dissociation constant by surface plasmon resonance based inhibition-in-solution ass...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2023
Entry Details Article
PubMed
TargetNuclear factor erythroid 2-related factor 2(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50584821(CHEMBL5076435)
Affinity DataKd:  3.60E+4nMAssay Description:Inhibition of Keap1-Nrf2 (unknown origin) interaction assessed as dissociation constant by surface plasmon resonance based inhibition-in-solution ass...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2023
Entry Details Article
PubMed
TargetKelch-like ECH-associated protein 1(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50584822(CHEMBL5092602)
Affinity DataKd:  41nMAssay Description:Binding affinity to Keap1 (unknown origin) at R415 assessed as dissociation constant by surface plasmon resonance based inhibition-in-solution assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2023
Entry Details Article
PubMed
TargetKelch-like ECH-associated protein 1(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50584823(CHEMBL5075717)
Affinity DataKd:  2.40E+3nMAssay Description:Binding affinity to Keap1 (unknown origin) at R415 assessed as dissociation constant by surface plasmon resonance based inhibition-in-solution assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2023
Entry Details Article
PubMed
TargetKelch-like ECH-associated protein 1(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50584824(CHEMBL5080665)
Affinity DataKd:  4.70E+3nMAssay Description:Binding affinity to Keap1 (unknown origin) at R415 assessed as dissociation constant by surface plasmon resonance based inhibition-in-solution assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2023
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetKelch-like ECH-associated protein 1(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50584825(CHEMBL5084413)
Affinity DataKd:  7.80E+3nMAssay Description:Binding affinity to Keap1 (unknown origin) at R415 assessed as dissociation constant by surface plasmon resonance based inhibition-in-solution assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2023
Entry Details Article
PubMed
TargetKelch-like ECH-associated protein 1(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50584826(CHEMBL5090939)
Affinity DataKd:  1.70E+3nMAssay Description:Binding affinity to Keap1 (unknown origin) at R415 assessed as dissociation constant by surface plasmon resonance based inhibition-in-solution assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2023
Entry Details Article
PubMed
TargetKelch-like ECH-associated protein 1(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50584827(CHEMBL5082071)
Affinity DataKd:  7.30E+3nMAssay Description:Binding affinity to Keap1 (unknown origin) at R415 assessed as dissociation constant by surface plasmon resonance based inhibition-in-solution assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2023
Entry Details Article
PubMed
TargetKelch-like ECH-associated protein 1(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50584828(CHEMBL5093123)
Affinity DataKd:  8.30E+3nMAssay Description:Binding affinity to Keap1 (unknown origin) at R415 assessed as dissociation constant by surface plasmon resonance based inhibition-in-solution assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2023
Entry Details Article
PubMed
TargetKelch-like ECH-associated protein 1(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50584829(CHEMBL5086087)
Affinity DataKd:  9.60E+3nMAssay Description:Binding affinity to Keap1 (unknown origin) at R415 assessed as dissociation constant by surface plasmon resonance based inhibition-in-solution assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2023
Entry Details Article
PubMed
TargetKelch-like ECH-associated protein 1(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50584830(CHEMBL5085704)
Affinity DataKd:  7.70E+3nMAssay Description:Binding affinity to Keap1 (unknown origin) at R415 assessed as dissociation constant by surface plasmon resonance based inhibition-in-solution assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2023
Entry Details Article
PubMed
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