Report error Found 112 Enz. Inhib. hit(s) with all data for entry = 50015340
TargetCannabinoid receptor 1(Human)
National Institute On Alcohol Abuse and Alcoholism
Curated by ChEMBL
National Institute On Alcohol Abuse and Alcoholism
Curated by ChEMBL
Affinity DataIC50: 0.800nMAssay Description:Inverse agonist activity at human CB1R expressed in CHO-K1 cell membrane assessed as increase in [35S]GTPgammaS bindingMore data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Human)
National Institute On Alcohol Abuse and Alcoholism
Curated by ChEMBL
National Institute On Alcohol Abuse and Alcoholism
Curated by ChEMBL
Affinity DataIC50: 1.20nMAssay Description:Antagonist activity at human CB1R expressed in CHO-K1 cell membranes assessed as stimulation of [35S]-GTPgammaS binding by liquid scintillation count...More data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Human)
National Institute On Alcohol Abuse and Alcoholism
Curated by ChEMBL
National Institute On Alcohol Abuse and Alcoholism
Curated by ChEMBL
Affinity DataIC50: 1.60nMAssay Description:Inverse agonist activity at human CB1R expressed in CHO-K1 cell membrane assessed as increase in [35S]GTPgammaS bindingMore data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Human)
National Institute On Alcohol Abuse and Alcoholism
Curated by ChEMBL
National Institute On Alcohol Abuse and Alcoholism
Curated by ChEMBL
Affinity DataIC50: 1.80nMAssay Description:Inverse agonist activity at human CB1R expressed in CHO-K1 cell membrane assessed as increase in [35S]GTPgammaS bindingMore data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Human)
National Institute On Alcohol Abuse and Alcoholism
Curated by ChEMBL
National Institute On Alcohol Abuse and Alcoholism
Curated by ChEMBL
Affinity DataIC50: 1.90nMAssay Description:Antagonist activity at human CB1R expressed in CHO-K1 cell membranes assessed as stimulation of [35S]-GTPgammaS binding by liquid scintillation count...More data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Human)
National Institute On Alcohol Abuse and Alcoholism
Curated by ChEMBL
National Institute On Alcohol Abuse and Alcoholism
Curated by ChEMBL
Affinity DataIC50: 2nMAssay Description:Antagonist activity at human CB1R expressed in CHO-K1 cell membranes assessed as stimulation of [35S]-GTPgammaS binding by liquid scintillation count...More data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Human)
National Institute On Alcohol Abuse and Alcoholism
Curated by ChEMBL
National Institute On Alcohol Abuse and Alcoholism
Curated by ChEMBL
Affinity DataIC50: 2nMAssay Description:Antagonist activity at human CB1R expressed in CHO-K1 cell membranes assessed as stimulation of [35S]-GTPgammaS binding by liquid scintillation count...More data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Human)
National Institute On Alcohol Abuse and Alcoholism
Curated by ChEMBL
National Institute On Alcohol Abuse and Alcoholism
Curated by ChEMBL
Affinity DataIC50: 2nMAssay Description:Inverse agonist activity at human CB1R expressed in CHO-K1 cell membrane assessed as increase in [35S]GTPgammaS bindingMore data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Human)
National Institute On Alcohol Abuse and Alcoholism
Curated by ChEMBL
National Institute On Alcohol Abuse and Alcoholism
Curated by ChEMBL
Affinity DataIC50: 2.5nMAssay Description:Inverse agonist activity at human CB1R expressed in CHO-K1 cell membrane assessed as increase in [35S]GTPgammaS bindingMore data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Human)
National Institute On Alcohol Abuse and Alcoholism
Curated by ChEMBL
National Institute On Alcohol Abuse and Alcoholism
Curated by ChEMBL
Affinity DataIC50: 2.80nMAssay Description:Antagonist activity at human CB1R expressed in CHO-K1 cell membranes assessed as stimulation of [35S]-GTPgammaS binding by liquid scintillation count...More data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Human)
National Institute On Alcohol Abuse and Alcoholism
Curated by ChEMBL
National Institute On Alcohol Abuse and Alcoholism
Curated by ChEMBL
Affinity DataIC50: 3.20nMAssay Description:Inverse agonist activity at human CB1R expressed in CHO-K1 cell membrane assessed as increase in [35S]GTPgammaS bindingMore data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Human)
National Institute On Alcohol Abuse and Alcoholism
Curated by ChEMBL
National Institute On Alcohol Abuse and Alcoholism
Curated by ChEMBL
Affinity DataIC50: 3.60nMAssay Description:Antagonist activity at human CB1R expressed in CHO-K1 cell membranes assessed as stimulation of [35S]-GTPgammaS binding by liquid scintillation count...More data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Human)
National Institute On Alcohol Abuse and Alcoholism
Curated by ChEMBL
National Institute On Alcohol Abuse and Alcoholism
Curated by ChEMBL
Affinity DataIC50: 4nMAssay Description:Antagonist activity at human CB1R expressed in CHO-K1 cell membranes assessed as stimulation of [35S]-GTPgammaS binding by liquid scintillation count...More data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Human)
National Institute On Alcohol Abuse and Alcoholism
Curated by ChEMBL
National Institute On Alcohol Abuse and Alcoholism
Curated by ChEMBL
Affinity DataIC50: 4nMAssay Description:Antagonist activity at human CB1R expressed in CHO-K1 cell membranes assessed as stimulation of [35S]-GTPgammaS binding by liquid scintillation count...More data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Human)
National Institute On Alcohol Abuse and Alcoholism
Curated by ChEMBL
National Institute On Alcohol Abuse and Alcoholism
Curated by ChEMBL
Affinity DataIC50: 4.20nMAssay Description:Antagonist activity at human CB1R expressed in CHO-K1 cell membranes assessed as stimulation of [35S]-GTPgammaS binding by liquid scintillation count...More data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Human)
National Institute On Alcohol Abuse and Alcoholism
Curated by ChEMBL
National Institute On Alcohol Abuse and Alcoholism
Curated by ChEMBL
Affinity DataIC50: 4.40nMAssay Description:Antagonist activity at human CB1R expressed in CHO-K1 cell membranes assessed as stimulation of [35S]-GTPgammaS binding by liquid scintillation count...More data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Human)
National Institute On Alcohol Abuse and Alcoholism
Curated by ChEMBL
National Institute On Alcohol Abuse and Alcoholism
Curated by ChEMBL
Affinity DataIC50: 5.40nMAssay Description:Antagonist activity at human CB1R expressed in CHO-K1 cell membranes assessed as stimulation of [35S]-GTPgammaS binding by liquid scintillation count...More data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Human)
National Institute On Alcohol Abuse and Alcoholism
Curated by ChEMBL
National Institute On Alcohol Abuse and Alcoholism
Curated by ChEMBL
Affinity DataIC50: 6nMAssay Description:Antagonist activity at human CB1R expressed in CHO-K1 cell membranes assessed as stimulation of [35S]-GTPgammaS binding by liquid scintillation count...More data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Human)
National Institute On Alcohol Abuse and Alcoholism
Curated by ChEMBL
National Institute On Alcohol Abuse and Alcoholism
Curated by ChEMBL
Affinity DataIC50: 10nMAssay Description:Antagonist activity at human CB1R expressed in CHO-K1 cell membranes assessed as stimulation of [35S]-GTPgammaS binding by liquid scintillation count...More data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Human)
National Institute On Alcohol Abuse and Alcoholism
Curated by ChEMBL
National Institute On Alcohol Abuse and Alcoholism
Curated by ChEMBL
Affinity DataIC50: 15nMAssay Description:Antagonist activity at human CB1R expressed in CHO-K1 cell membranes assessed as stimulation of [35S]-GTPgammaS binding by liquid scintillation count...More data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Human)
National Institute On Alcohol Abuse and Alcoholism
Curated by ChEMBL
National Institute On Alcohol Abuse and Alcoholism
Curated by ChEMBL
Affinity DataIC50: 19nMAssay Description:Antagonist activity at human CB1R expressed in CHO-K1 cell membranes assessed as stimulation of [35S]-GTPgammaS binding by liquid scintillation count...More data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Human)
National Institute On Alcohol Abuse and Alcoholism
Curated by ChEMBL
National Institute On Alcohol Abuse and Alcoholism
Curated by ChEMBL
Affinity DataIC50: 25nMAssay Description:Antagonist activity at human CB1R expressed in CHO-K1 cell membranes assessed as stimulation of [35S]-GTPgammaS binding by liquid scintillation count...More data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Human)
National Institute On Alcohol Abuse and Alcoholism
Curated by ChEMBL
National Institute On Alcohol Abuse and Alcoholism
Curated by ChEMBL
Affinity DataIC50: 34nMAssay Description:Antagonist activity at human CB1R expressed in CHO-K1 cell membranes assessed as stimulation of [35S]-GTPgammaS binding by liquid scintillation count...More data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Human)
National Institute On Alcohol Abuse and Alcoholism
Curated by ChEMBL
National Institute On Alcohol Abuse and Alcoholism
Curated by ChEMBL
Affinity DataIC50: 57nMAssay Description:Antagonist activity at human CB1R expressed in CHO-K1 cell membranes assessed as stimulation of [35S]-GTPgammaS binding by liquid scintillation count...More data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Human)
National Institute On Alcohol Abuse and Alcoholism
Curated by ChEMBL
National Institute On Alcohol Abuse and Alcoholism
Curated by ChEMBL
Affinity DataIC50: 61nMAssay Description:Antagonist activity at human CB1R expressed in CHO-K1 cell membranes assessed as stimulation of [35S]-GTPgammaS binding by liquid scintillation count...More data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Human)
National Institute On Alcohol Abuse and Alcoholism
Curated by ChEMBL
National Institute On Alcohol Abuse and Alcoholism
Curated by ChEMBL
Affinity DataIC50: 63nMAssay Description:Antagonist activity at human CB1R expressed in CHO-K1 cell membranes assessed as stimulation of [35S]-GTPgammaS binding by liquid scintillation count...More data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Human)
National Institute On Alcohol Abuse and Alcoholism
Curated by ChEMBL
National Institute On Alcohol Abuse and Alcoholism
Curated by ChEMBL
Affinity DataIC50: 86nMAssay Description:Antagonist activity at human CB1R expressed in CHO-K1 cell membranes assessed as stimulation of [35S]-GTPgammaS binding by liquid scintillation count...More data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Human)
National Institute On Alcohol Abuse and Alcoholism
Curated by ChEMBL
National Institute On Alcohol Abuse and Alcoholism
Curated by ChEMBL
Affinity DataIC50: 91nMAssay Description:Antagonist activity at human CB1R expressed in CHO-K1 cell membranes assessed as stimulation of [35S]-GTPgammaS binding by liquid scintillation count...More data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Human)
National Institute On Alcohol Abuse and Alcoholism
Curated by ChEMBL
National Institute On Alcohol Abuse and Alcoholism
Curated by ChEMBL
Affinity DataIC50: 108nMAssay Description:Antagonist activity at human CB1R expressed in CHO-K1 cell membranes assessed as stimulation of [35S]-GTPgammaS binding by liquid scintillation count...More data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Human)
National Institute On Alcohol Abuse and Alcoholism
Curated by ChEMBL
National Institute On Alcohol Abuse and Alcoholism
Curated by ChEMBL
Affinity DataIC50: 115nMAssay Description:Antagonist activity at human CB1R expressed in CHO-K1 cell membranes assessed as stimulation of [35S]-GTPgammaS binding by liquid scintillation count...More data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Human)
National Institute On Alcohol Abuse and Alcoholism
Curated by ChEMBL
National Institute On Alcohol Abuse and Alcoholism
Curated by ChEMBL
Affinity DataIC50: 127nMAssay Description:Antagonist activity at human CB1R expressed in CHO-K1 cell membranes assessed as stimulation of [35S]-GTPgammaS binding by liquid scintillation count...More data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Human)
National Institute On Alcohol Abuse and Alcoholism
Curated by ChEMBL
National Institute On Alcohol Abuse and Alcoholism
Curated by ChEMBL
Affinity DataIC50: 129nMAssay Description:Antagonist activity at human CB1R expressed in CHO-K1 cell membranes assessed as stimulation of [35S]-GTPgammaS binding by liquid scintillation count...More data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Human)
National Institute On Alcohol Abuse and Alcoholism
Curated by ChEMBL
National Institute On Alcohol Abuse and Alcoholism
Curated by ChEMBL
Affinity DataIC50: 137nMAssay Description:Antagonist activity at human CB1R expressed in CHO-K1 cell membranes assessed as stimulation of [35S]-GTPgammaS binding by liquid scintillation count...More data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Human)
National Institute On Alcohol Abuse and Alcoholism
Curated by ChEMBL
National Institute On Alcohol Abuse and Alcoholism
Curated by ChEMBL
Affinity DataIC50: 166nMAssay Description:Antagonist activity at human CB1R expressed in CHO-K1 cell membranes assessed as stimulation of [35S]-GTPgammaS binding by liquid scintillation count...More data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Human)
National Institute On Alcohol Abuse and Alcoholism
Curated by ChEMBL
National Institute On Alcohol Abuse and Alcoholism
Curated by ChEMBL
Affinity DataIC50: 273nMAssay Description:Antagonist activity at human CB1R expressed in CHO-K1 cell membranes assessed as stimulation of [35S]-GTPgammaS binding by liquid scintillation count...More data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Human)
National Institute On Alcohol Abuse and Alcoholism
Curated by ChEMBL
National Institute On Alcohol Abuse and Alcoholism
Curated by ChEMBL
Affinity DataIC50: 375nMAssay Description:Antagonist activity at human CB1R expressed in CHO-K1 cell membranes assessed as stimulation of [35S]-GTPgammaS binding by liquid scintillation count...More data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Human)
National Institute On Alcohol Abuse and Alcoholism
Curated by ChEMBL
National Institute On Alcohol Abuse and Alcoholism
Curated by ChEMBL
Affinity DataIC50: 388nMAssay Description:Antagonist activity at human CB1R expressed in CHO-K1 cell membranes assessed as stimulation of [35S]-GTPgammaS binding by liquid scintillation count...More data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Human)
National Institute On Alcohol Abuse and Alcoholism
Curated by ChEMBL
National Institute On Alcohol Abuse and Alcoholism
Curated by ChEMBL
Affinity DataIC50: 427nMAssay Description:Antagonist activity at human CB1R expressed in CHO-K1 cell membranes assessed as stimulation of [35S]-GTPgammaS binding by liquid scintillation count...More data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Human)
National Institute On Alcohol Abuse and Alcoholism
Curated by ChEMBL
National Institute On Alcohol Abuse and Alcoholism
Curated by ChEMBL
Affinity DataIC50: 462nMAssay Description:Antagonist activity at human CB1R expressed in CHO-K1 cell membranes assessed as stimulation of [35S]-GTPgammaS binding by liquid scintillation count...More data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Human)
National Institute On Alcohol Abuse and Alcoholism
Curated by ChEMBL
National Institute On Alcohol Abuse and Alcoholism
Curated by ChEMBL
Affinity DataKi: 0.700nMAssay Description:Displacement of [3H]- CP55940 from human CB1R expressed in CHO-K1 cells membrane by Cheng-Prusoff equation analysisMore data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Human)
National Institute On Alcohol Abuse and Alcoholism
Curated by ChEMBL
National Institute On Alcohol Abuse and Alcoholism
Curated by ChEMBL
Affinity DataKi: 1.10nMAssay Description:Displacement of [3H]- CP55940 from human CB1R expressed in CHO-K1 cells membrane by Cheng-Prusoff equation analysisMore data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Human)
National Institute On Alcohol Abuse and Alcoholism
Curated by ChEMBL
National Institute On Alcohol Abuse and Alcoholism
Curated by ChEMBL
Affinity DataKi: 1.20nMAssay Description:Displacement of [3H]- CP55940 from human CB1R expressed in CHO-K1 cells membrane by Cheng-Prusoff equation analysisMore data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Human)
National Institute On Alcohol Abuse and Alcoholism
Curated by ChEMBL
National Institute On Alcohol Abuse and Alcoholism
Curated by ChEMBL
Affinity DataKi: 1.60nMAssay Description:Displacement of [3H]- CP55940 from human CB1R expressed in CHO-K1 cells membrane by Cheng-Prusoff equation analysisMore data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Human)
National Institute On Alcohol Abuse and Alcoholism
Curated by ChEMBL
National Institute On Alcohol Abuse and Alcoholism
Curated by ChEMBL
Affinity DataKi: 2.40nMAssay Description:Displacement of [3H]- CP55940 from human CB1R expressed in CHO-K1 cells membrane by Cheng-Prusoff equation analysisMore data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Human)
National Institute On Alcohol Abuse and Alcoholism
Curated by ChEMBL
National Institute On Alcohol Abuse and Alcoholism
Curated by ChEMBL
Affinity DataKi: 3nMAssay Description:Displacement of [3H]- CP55940 from human CB1R expressed in CHO-K1 cells membrane by Cheng-Prusoff equation analysisMore data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Human)
National Institute On Alcohol Abuse and Alcoholism
Curated by ChEMBL
National Institute On Alcohol Abuse and Alcoholism
Curated by ChEMBL
Affinity DataKi: 3.30nMAssay Description:Displacement of [3H]- CP55940 from human CB1R expressed in CHO-K1 cells membrane by Cheng-Prusoff equation analysisMore data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Human)
National Institute On Alcohol Abuse and Alcoholism
Curated by ChEMBL
National Institute On Alcohol Abuse and Alcoholism
Curated by ChEMBL
Affinity DataKi: 3.40nMAssay Description:Displacement of [3H]- CP55940 from human CB1R expressed in CHO-K1 cells membrane by Cheng-Prusoff equation analysisMore data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Human)
National Institute On Alcohol Abuse and Alcoholism
Curated by ChEMBL
National Institute On Alcohol Abuse and Alcoholism
Curated by ChEMBL
Affinity DataKi: 3.90nMAssay Description:Displacement of [3H]- CP55940 from human CB1R expressed in CHO-K1 cells membrane by Cheng-Prusoff equation analysisMore data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Human)
National Institute On Alcohol Abuse and Alcoholism
Curated by ChEMBL
National Institute On Alcohol Abuse and Alcoholism
Curated by ChEMBL
Affinity DataKi: 5.5nMAssay Description:Displacement of [3H]- CP55940 from human CB1R expressed in CHO-K1 cells membrane by Cheng-Prusoff equation analysisMore data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Human)
National Institute On Alcohol Abuse and Alcoholism
Curated by ChEMBL
National Institute On Alcohol Abuse and Alcoholism
Curated by ChEMBL
Affinity DataKi: 5.5nMAssay Description:Displacement of [3H]- CP55940 from human CB1R expressed in CHO-K1 cells membrane by Cheng-Prusoff equation analysisMore data for this Ligand-Target Pair
