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Report error Found 20 Enz. Inhib. hit(s) with all data for entry = 50017615
TargetSerine/threonine-protein kinase Nek1(Human)
Technische Universit£T Darmstadt

Curated by ChEMBL
LigandPNGBDBM50603394(CHEMBL5201686)
Affinity DataIC50: 330nMAssay Description:Inhibition of human recombinant NEK1 (1 to 505 residues) using ULight-p70 S6K peptide as substrate incubated for 30 mins by LANCE Ultra TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetSerine/threonine-protein kinase Nek1(Human)
Technische Universit£T Darmstadt

Curated by ChEMBL
LigandPNGBDBM50603394(CHEMBL5201686)
Affinity DataIC50: 330nMAssay Description:Inhibition of human recombinant NEK1 (1 to 505 residues) using RLGRDKYKTLRQIRQ as substrate incubated for 40 mins in presence of [gamma-33P]-ATP by r...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetSerine/threonine-protein kinase Nek1(Human)
Technische Universit£T Darmstadt

Curated by ChEMBL
LigandPNGBDBM50603408(CHEMBL5206874)
Affinity DataIC50: 990nMAssay Description:Inhibition of human recombinant NEK1 (1 to 505 residues) using ULight-p70 S6K peptide as substrate incubated for 30 mins by LANCE Ultra TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetSerine/threonine-protein kinase Nek1(Human)
Technische Universit£T Darmstadt

Curated by ChEMBL
LigandPNGBDBM50603405(CHEMBL5189609)
Affinity DataIC50: 1.30E+3nMAssay Description:Inhibition of human recombinant NEK1 (1 to 505 residues) using ULight-p70 S6K peptide as substrate incubated for 30 mins by LANCE Ultra TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetSerine/threonine-protein kinase Nek1(Human)
Technische Universit£T Darmstadt

Curated by ChEMBL
LigandPNGBDBM50603407(CHEMBL5200819)
Affinity DataIC50: 1.60E+3nMAssay Description:Inhibition of human recombinant NEK1 (1 to 505 residues) using ULight-p70 S6K peptide as substrate incubated for 30 mins by LANCE Ultra TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetSerine/threonine-protein kinase Nek1(Human)
Technische Universit£T Darmstadt

Curated by ChEMBL
LigandPNGBDBM50603404(CHEMBL5174141)
Affinity DataIC50: 1.90E+3nMAssay Description:Inhibition of human recombinant NEK1 (1 to 505 residues) using ULight-p70 S6K peptide as substrate incubated for 30 mins by LANCE Ultra TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetSerine/threonine-protein kinase Nek1(Human)
Technische Universit£T Darmstadt

Curated by ChEMBL
LigandPNGBDBM50603393(CHEMBL5197597)
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of human recombinant NEK1 (1 to 505 residues) using RLGRDKYKTLRQIRQ as substrate incubated for 40 mins in presence of [gamma-33P]-ATP by r...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetSerine/threonine-protein kinase Nek1(Human)
Technische Universit£T Darmstadt

Curated by ChEMBL
LigandPNGBDBM50603406(CHEMBL5182208)
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of human recombinant NEK1 (1 to 505 residues) using ULight-p70 S6K peptide as substrate incubated for 30 mins by LANCE Ultra TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetSerine/threonine-protein kinase Nek1(Human)
Technische Universit£T Darmstadt

Curated by ChEMBL
LigandPNGBDBM50603400(CHEMBL5182549)
Affinity DataIC50: 2.70E+3nMAssay Description:Inhibition of human recombinant NEK1 (1 to 505 residues) using ULight-p70 S6K peptide as substrate incubated for 30 mins by LANCE Ultra TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetSerine/threonine-protein kinase Nek1(Human)
Technische Universit£T Darmstadt

Curated by ChEMBL
LigandPNGBDBM50603393(CHEMBL5197597)
Affinity DataIC50: 3.20E+3nMAssay Description:Inhibition of human recombinant NEK1 (1 to 505 residues) using ULight-p70 S6K peptide as substrate incubated for 30 mins by LANCE Ultra TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetSerine/threonine-protein kinase Nek1(Human)
Technische Universit£T Darmstadt

Curated by ChEMBL
LigandPNGBDBM50413876(CHEMBL520954)
Affinity DataIC50: 4.30E+3nMAssay Description:Inhibition of human recombinant NEK1 (1 to 505 residues) using RLGRDKYKTLRQIRQ as substrate incubated for 40 mins in presence of [gamma-33P]-ATP by r...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetSerine/threonine-protein kinase Nek1(Human)
Technische Universit£T Darmstadt

Curated by ChEMBL
LigandPNGBDBM50603402(CHEMBL5203616)
Affinity DataIC50: 5.80E+3nMAssay Description:Inhibition of human recombinant NEK1 (1 to 505 residues) using ULight-p70 S6K peptide as substrate incubated for 30 mins by LANCE Ultra TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetSerine/threonine-protein kinase Nek1(Human)
Technische Universit£T Darmstadt

Curated by ChEMBL
LigandPNGBDBM50603396(CHEMBL5208840)
Affinity DataIC50: 6.60E+3nMAssay Description:Inhibition of human recombinant NEK1 (1 to 505 residues) using ULight-p70 S6K peptide as substrate incubated for 30 mins by LANCE Ultra TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetSerine/threonine-protein kinase Nek1(Human)
Technische Universit£T Darmstadt

Curated by ChEMBL
LigandPNGBDBM50413876(CHEMBL520954)
Affinity DataIC50: 7.10E+3nMAssay Description:Inhibition of human recombinant NEK1 (1 to 505 residues) using ULight-p70 S6K peptide as substrate incubated for 30 mins by LANCE Ultra TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetSerine/threonine-protein kinase Nek1(Human)
Technische Universit£T Darmstadt

Curated by ChEMBL
LigandPNGBDBM50603401(CHEMBL5197360)
Affinity DataIC50: 8.80E+3nMAssay Description:Inhibition of human recombinant NEK1 (1 to 505 residues) using ULight-p70 S6K peptide as substrate incubated for 30 mins by LANCE Ultra TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetSerine/threonine-protein kinase Nek1(Human)
Technische Universit£T Darmstadt

Curated by ChEMBL
LigandPNGBDBM50603395(CHEMBL5181887)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human recombinant NEK1 (1 to 505 residues) using ULight-p70 S6K peptide as substrate incubated for 30 mins by LANCE Ultra TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetSerine/threonine-protein kinase Nek1(Human)
Technische Universit£T Darmstadt

Curated by ChEMBL
LigandPNGBDBM50603398(CHEMBL5172286)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human recombinant NEK1 (1 to 505 residues) using ULight-p70 S6K peptide as substrate incubated for 30 mins by LANCE Ultra TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetSerine/threonine-protein kinase Nek1(Human)
Technische Universit£T Darmstadt

Curated by ChEMBL
LigandPNGBDBM50603397(CHEMBL5197075)
Affinity DataIC50: 2.70E+4nMAssay Description:Inhibition of human recombinant NEK1 (1 to 505 residues) using ULight-p70 S6K peptide as substrate incubated for 30 mins by LANCE Ultra TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetSerine/threonine-protein kinase Nek1(Human)
Technische Universit£T Darmstadt

Curated by ChEMBL
LigandPNGBDBM50603403(CHEMBL5180286)
Affinity DataIC50: 2.90E+4nMAssay Description:Inhibition of human recombinant NEK1 (1 to 505 residues) using ULight-p70 S6K peptide as substrate incubated for 30 mins by LANCE Ultra TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetSerine/threonine-protein kinase Nek1(Human)
Technische Universit£T Darmstadt

Curated by ChEMBL
LigandPNGBDBM50603399(CHEMBL5180705)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of human recombinant NEK1 (1 to 505 residues) using ULight-p70 S6K peptide as substrate incubated for 30 mins by LANCE Ultra TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed