Compile Data Set for Download or QSAR
Report error Found 6 Enz. Inhib. hit(s) with all data for entry = 50017595
TargetGTPase KRas(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM50514402(CHEMBL4535757 | US11345701, Compound Amg-510)
Affinity DataIC50: 9.70nMAssay Description:Inhibition of KRAS G12C mutant (unknown origin) assessed as inhibition of SOS1-catalyzed nucleotide exchange measured by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetGTPase KRas(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM50603203(CHEMBL5171974)
Affinity DataIC50: 25nMAssay Description:Inhibition of KRAS G12C mutant (unknown origin) assessed as inhibition of SOS1-catalyzed nucleotide exchange measured by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetGTPase KRas(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM50603200(CHEMBL5206068)
Affinity DataIC50: 96nMAssay Description:Inhibition of KRAS G12C mutant (unknown origin) assessed as inhibition of SOS1-catalyzed nucleotide exchange measured by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetGTPase KRas(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM50603201(CHEMBL5205064)
Affinity DataIC50: 271nMAssay Description:Inhibition of KRAS G12C mutant (unknown origin) assessed as inhibition of SOS1-catalyzed nucleotide exchange measured by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetGTPase KRas(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM50603202(CHEMBL5194712)
Affinity DataIC50: 284nMAssay Description:Inhibition of KRAS G12C mutant (unknown origin) assessed as inhibition of SOS1-catalyzed nucleotide exchange measured by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetGTPase KRas(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM50603204(CHEMBL5185805)
Affinity DataIC50: 640nMAssay Description:Inhibition of KRAS G12C mutant (unknown origin) assessed as inhibition of SOS1-catalyzed nucleotide exchange measured by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed