Compile Data Set for Download or QSAR
Report error Found 5 Enz. Inhib. hit(s) with all data for entry = 50015327
TargetCarboxy-terminal domain RNA polymerase II polypeptide A small phosphatase 1(Human)
University of California San Diego

Curated by ChEMBL
LigandPNGBDBM50585529(CHEMBL5077686)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of wild type human SCP1 using pNPP as substrate incubated for 0.5 to 18 hrs followed by substrate addition by absorbance based analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetCarboxy-terminal domain RNA polymerase II polypeptide A small phosphatase 1(Human)
University of California San Diego

Curated by ChEMBL
LigandPNGBDBM50585531(CHEMBL5079017)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of wild type human SCP1 using pNPP as substrate incubated for 0.5 to 18 hrs followed by substrate addition by absorbance based analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetCarboxy-terminal domain RNA polymerase II polypeptide A small phosphatase 1(Human)
University of California San Diego

Curated by ChEMBL
LigandPNGBDBM50585530(CHEMBL5093163)
Affinity DataIC50: 2.20E+5nMAssay Description:Inhibition of wild type human SCP1 using pNPP as substrate incubated for 0.5 to 18 hrs followed by substrate addition by absorbance based analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetCarboxy-terminal domain RNA polymerase II polypeptide A small phosphatase 1(Human)
University of California San Diego

Curated by ChEMBL
LigandPNGBDBM50585532(CHEMBL5092456)
Affinity DataIC50: 7.97E+5nMAssay Description:Inhibition of wild type human SCP1 using pNPP as substrate incubated for 0.5 to 18 hrs followed by substrate addition by absorbance based analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetCarboxy-terminal domain RNA polymerase II polypeptide A small phosphatase 1(Human)
University of California San Diego

Curated by ChEMBL
LigandPNGBDBM50585529(CHEMBL5077686)
Affinity DataKi:  4.80E+3nMAssay Description:Covalent inhibition of wild type human SCP1 assessed as inhibition constant using Ac-EDLphosphoSPPSPPLPK-NH2 peptide as substrate preincubated for 0....More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed