Compile Data Set for Download or QSAR
Report error Found 9 Enz. Inhib. hit(s) with all data for entry = 50017983
TargetBromodomain-containing protein 4(Human)
Universitat De Barcelona

Curated by ChEMBL
LigandPNGBDBM50606697(CHEMBL5218482)
Affinity DataIC50: 2.60E+4nMAssay Description:Inhibition of BRD4 (unknown origin) expressed in Escherichia coli BL21 (DE3) using [Lys(Ac)5/8/12/16]-histone H4 (1 to 21residues)-GGK as substrate i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2023
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
Universitat De Barcelona

Curated by ChEMBL
LigandPNGBDBM50606693(CHEMBL5219547)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of BRD4 (unknown origin) expressed in Escherichia coli BL21 (DE3) using [Lys(Ac)5/8/12/16]-histone H4 (1 to 21residues)-GGK as substrate i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2023
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetBromodomain-containing protein 4(Human)
Universitat De Barcelona

Curated by ChEMBL
LigandPNGBDBM50606690(CHEMBL197512)
Affinity DataIC50: 7.20E+4nMAssay Description:Inhibition of BRD4 (unknown origin) expressed in Escherichia coli BL21 (DE3) using [Lys(Ac)5/8/12/16]-histone H4 (1 to 21residues)-GGK as substrate i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2023
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
Universitat De Barcelona

Curated by ChEMBL
LigandPNGBDBM50606692(CHEMBL5220412)
Affinity DataIC50: 7.90E+4nMAssay Description:Inhibition of BRD4 (unknown origin) expressed in Escherichia coli BL21 (DE3) using [Lys(Ac)5/8/12/16]-histone H4 (1 to 21residues)-GGK as substrate i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2023
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
Universitat De Barcelona

Curated by ChEMBL
LigandPNGBDBM50606695(CHEMBL5220338)
Affinity DataIC50: 8.60E+4nMAssay Description:Inhibition of BRD4 (unknown origin) expressed in Escherichia coli BL21 (DE3) using [Lys(Ac)5/8/12/16]-histone H4 (1 to 21residues)-GGK as substrate i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2023
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
Universitat De Barcelona

Curated by ChEMBL
LigandPNGBDBM50440736(CHEMBL2431088)
Affinity DataIC50: 9.10E+4nMAssay Description:Inhibition of BRD4 (unknown origin) expressed in Escherichia coli BL21 (DE3) using [Lys(Ac)5/8/12/16]-histone H4 (1 to 21residues)-GGK as substrate i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2023
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
Universitat De Barcelona

Curated by ChEMBL
LigandPNGBDBM50606691(CHEMBL5220563)
Affinity DataIC50: 1.91E+5nMAssay Description:Inhibition of BRD4 (unknown origin) expressed in Escherichia coli BL21 (DE3) using [Lys(Ac)5/8/12/16]-histone H4 (1 to 21residues)-GGK as substrate i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2023
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
Universitat De Barcelona

Curated by ChEMBL
LigandPNGBDBM50606696(CHEMBL5218934)
Affinity DataIC50: 4.91E+5nMAssay Description:Inhibition of BRD4 (unknown origin) expressed in Escherichia coli BL21 (DE3) using [Lys(Ac)5/8/12/16]-histone H4 (1 to 21residues)-GGK as substrate i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2023
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
Universitat De Barcelona

Curated by ChEMBL
LigandPNGBDBM50606694(CHEMBL5219925)
Affinity DataIC50: 6.44E+5nMAssay Description:Inhibition of BRD4 (unknown origin) expressed in Escherichia coli BL21 (DE3) using [Lys(Ac)5/8/12/16]-histone H4 (1 to 21residues)-GGK as substrate i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2023
Entry Details
PubMed