Compile Data Set for Download or QSAR
Report error Found 45 Enz. Inhib. hit(s) with all data for entry = 50017551
TargetHistone deacetylase 4(Human)
Stony Brook University

Curated by ChEMBL
LigandPNGBDBM162865(US9056843, 156)
Affinity DataIC50: 0.0800nMAssay Description:Inhibition of recombinant human HDAC4 using fluorogenic substrate by fluorescence microplate reader assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetHistone deacetylase 9(Human)
Stony Brook University

Curated by ChEMBL
LigandPNGBDBM162865(US9056843, 156)
Affinity DataIC50: 0.900nMAssay Description:Inhibition of recombinant human HDAC9 using fluorogenic substrate by fluorescence microplate reader assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetHistone deacetylase 7(Human)
Stony Brook University

Curated by ChEMBL
LigandPNGBDBM162865(US9056843, 156)
Affinity DataIC50: 1nMAssay Description:Inhibition of recombinant human HDAC7 using fluorogenic substrate by fluorescence microplate reader assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetHistone deacetylase 5(Human)
Stony Brook University

Curated by ChEMBL
LigandPNGBDBM162865(US9056843, 156)
Affinity DataIC50: 1.20nMAssay Description:Inhibition of recombinant human HDAC5 using fluorogenic substrate by fluorescence microplate reader assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetHistone deacetylase 9(Human)
Stony Brook University

Curated by ChEMBL
LigandPNGBDBM50563276(CHEMBL4751615)
Affinity DataIC50: 2.40nMAssay Description:Inhibition of recombinant human HDAC9 using fluorogenic substrate by fluorescence microplate reader assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetHistone deacetylase 7(Human)
Stony Brook University

Curated by ChEMBL
LigandPNGBDBM50563276(CHEMBL4751615)
Affinity DataIC50: 7.70nMAssay Description:Inhibition of recombinant human HDAC7 using fluorogenic substrate by fluorescence microplate reader assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetHistone deacetylase 4(Human)
Stony Brook University

Curated by ChEMBL
LigandPNGBDBM50563276(CHEMBL4751615)
Affinity DataIC50: 128nMAssay Description:Inhibition of recombinant human HDAC4 using fluorogenic substrate by fluorescence microplate reader assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetHistone deacetylase 5(Human)
Stony Brook University

Curated by ChEMBL
LigandPNGBDBM50563276(CHEMBL4751615)
Affinity DataIC50: 148nMAssay Description:Inhibition of recombinant human HDAC5 using fluorogenic substrate by fluorescence microplate reader assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetHistone deacetylase 11(Human)
Stony Brook University

Curated by ChEMBL
LigandPNGBDBM162865(US9056843, 156)
Affinity DataIC50: 600nMAssay Description:Inhibition of recombinant human HDAC11 using fluorogenic substrate by fluorescence microplate reader assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetPolyamine deacetylase HDAC10(Human)
Stony Brook University

Curated by ChEMBL
LigandPNGBDBM162865(US9056843, 156)
Affinity DataIC50: 600nMAssay Description:Inhibition of recombinant human HDAC10 using fluorogenic substrate by fluorescence microplate reader assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetHistone deacetylase 1(Human)
Stony Brook University

Curated by ChEMBL
LigandPNGBDBM162865(US9056843, 156)
Affinity DataIC50: 600nMAssay Description:Inhibition of recombinant human HDAC1 using fluorogenic substrate by fluorescence microplate reader assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetHistone deacetylase 2(Human)
Stony Brook University

Curated by ChEMBL
LigandPNGBDBM162865(US9056843, 156)
Affinity DataIC50: 600nMAssay Description:Inhibition of recombinant human HDAC2 using fluorogenic substrate by fluorescence microplate reader assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetHistone deacetylase 3(Human)
Stony Brook University

Curated by ChEMBL
LigandPNGBDBM162865(US9056843, 156)
Affinity DataIC50: 600nMAssay Description:Inhibition of recombinant human HDAC3 using fluorogenic substrate by fluorescence microplate reader assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetHistone deacetylase 6(Human)
Stony Brook University

Curated by ChEMBL
LigandPNGBDBM162865(US9056843, 156)
Affinity DataIC50: 600nMAssay Description:Inhibition of recombinant human HDAC6 using fluorogenic substrate by fluorescence microplate reader assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetHistone deacetylase 8(Human)
Stony Brook University

Curated by ChEMBL
LigandPNGBDBM162865(US9056843, 156)
Affinity DataIC50: 600nMAssay Description:Inhibition of recombinant human HDAC8 using fluorogenic substrate by fluorescence microplate reader assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetHistone deacetylase 1/2/3/8(Human)
Stony Brook University

Curated by ChEMBL
LigandPNGBDBM19149(Zolinza | suberoylanilide hydroxamic acid | CHEMBL...)
Affinity DataIC50: 950nMAssay Description:Inhibition of HDAC class 1 in human HT-29 cells using Boc-Lys-Ac as substrate incubated for 3 hrs by microplate reader assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetHistone deacetylase 1/2/3/8(Human)
Stony Brook University

Curated by ChEMBL
LigandPNGBDBM50602709(CHEMBL5175492)
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of HDAC class 1 in human HT-29 cells using Boc-Lys-Ac as substrate incubated for 3 hrs by microplate reader assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetHistone deacetylase 1(Human)
Stony Brook University

Curated by ChEMBL
LigandPNGBDBM50563276(CHEMBL4751615)
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of recombinant human HDAC1 using fluorogenic substrate by fluorescence microplate reader assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetHistone deacetylase 1/2/3/8(Human)
Stony Brook University

Curated by ChEMBL
LigandPNGBDBM50602710(CHEMBL5207250)
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of HDAC class 1 in human HT-29 cells using Boc-Lys-Ac as substrate incubated for 3 hrs by microplate reader assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetHistone deacetylase 11(Human)
Stony Brook University

Curated by ChEMBL
LigandPNGBDBM50563276(CHEMBL4751615)
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of recombinant human HDAC11 using fluorogenic substrate by fluorescence microplate reader assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetPolyamine deacetylase HDAC10(Human)
Stony Brook University

Curated by ChEMBL
LigandPNGBDBM50563276(CHEMBL4751615)
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of recombinant human HDAC10 using fluorogenic substrate by fluorescence microplate reader assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetHistone deacetylase 2(Human)
Stony Brook University

Curated by ChEMBL
LigandPNGBDBM50563276(CHEMBL4751615)
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of recombinant human HDAC2 using fluorogenic substrate by fluorescence microplate reader assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetHistone deacetylase 3(Human)
Stony Brook University

Curated by ChEMBL
LigandPNGBDBM50563276(CHEMBL4751615)
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of recombinant human HDAC3 using fluorogenic substrate by fluorescence microplate reader assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetHistone deacetylase 6(Human)
Stony Brook University

Curated by ChEMBL
LigandPNGBDBM50563276(CHEMBL4751615)
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of recombinant human HDAC6 using fluorogenic substrate by fluorescence microplate reader assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetHistone deacetylase 8(Human)
Stony Brook University

Curated by ChEMBL
LigandPNGBDBM50563276(CHEMBL4751615)
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of recombinant human HDAC8 using fluorogenic substrate by fluorescence microplate reader assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetHistone deacetylase 1/2/3/8(Human)
Stony Brook University

Curated by ChEMBL
LigandPNGBDBM50563276(CHEMBL4751615)
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of HDAC class 1 in human PANC-1 cells using TFA-lysine as fluorogenic substrate by fluorescence microplate reader assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetHistone deacetylase 1/2/3/8(Human)
Stony Brook University

Curated by ChEMBL
LigandPNGBDBM50563276(CHEMBL4751615)
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of HDAC class 1 in human L3.6pl cells using TFA-lysine as fluorogenic substrate by fluorescence microplate reader assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetHistone deacetylase 1/2/3/8(Human)
Stony Brook University

Curated by ChEMBL
LigandPNGBDBM50563276(CHEMBL4751615)
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of HDAC class 1 in human HT-29 cells using TFA-lysine as fluorogenic substrate by fluorescence microplate reader assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetHistone deacetylase 1/2/3/8(Human)
Stony Brook University

Curated by ChEMBL
LigandPNGBDBM50563276(CHEMBL4751615)
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of HDAC class 1 in human THP-1 cells using TFA-lysine as fluorogenic substrate by fluorescence microplate reader assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetHistone deacetylase 1/2/3/8(Human)
Stony Brook University

Curated by ChEMBL
LigandPNGBDBM50602700(CHEMBL5197249)
Affinity DataIC50: 1.50E+4nMAssay Description:Inhibition of HDAC class 1 in human HT-29 cells using Boc-Lys-Ac as substrate incubated for 3 hrs by microplate reader assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetHistone deacetylase 1/2/3/8(Human)
Stony Brook University

Curated by ChEMBL
LigandPNGBDBM50602698(CHEMBL5174272)
Affinity DataIC50: 1.50E+4nMAssay Description:Inhibition of HDAC class 1 in human HT-29 cells using Boc-Lys-Ac as substrate incubated for 3 hrs by microplate reader assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetHistone deacetylase 1/2/3/8(Human)
Stony Brook University

Curated by ChEMBL
LigandPNGBDBM50602699(CHEMBL5201177)
Affinity DataIC50: 1.50E+4nMAssay Description:Inhibition of HDAC class 1 in human HT-29 cells using Boc-Lys-Ac as substrate incubated for 3 hrs by microplate reader assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetHistone deacetylase 1/2/3/8(Human)
Stony Brook University

Curated by ChEMBL
LigandPNGBDBM50602701(CHEMBL5199173)
Affinity DataIC50: 1.50E+4nMAssay Description:Inhibition of HDAC class 1 in human HT-29 cells using Boc-Lys-Ac as substrate incubated for 3 hrs by microplate reader assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetHistone deacetylase 1/2/3/8(Human)
Stony Brook University

Curated by ChEMBL
LigandPNGBDBM50602702(CHEMBL5184794)
Affinity DataIC50: 1.50E+4nMAssay Description:Inhibition of HDAC class 1 in human HT-29 cells using Boc-Lys-Ac as substrate incubated for 3 hrs by microplate reader assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetHistone deacetylase 1/2/3/8(Human)
Stony Brook University

Curated by ChEMBL
LigandPNGBDBM50602703(CHEMBL5192381)
Affinity DataIC50: 1.50E+4nMAssay Description:Inhibition of HDAC class 1 in human HT-29 cells using Boc-Lys-Ac as substrate incubated for 3 hrs by microplate reader assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetHistone deacetylase 1/2/3/8(Human)
Stony Brook University

Curated by ChEMBL
LigandPNGBDBM50602704(CHEMBL5198169)
Affinity DataIC50: 1.50E+4nMAssay Description:Inhibition of HDAC class 1 in human HT-29 cells using Boc-Lys-Ac as substrate incubated for 3 hrs by microplate reader assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetHistone deacetylase 1/2/3/8(Human)
Stony Brook University

Curated by ChEMBL
LigandPNGBDBM50602705(CHEMBL5184901)
Affinity DataIC50: 1.50E+4nMAssay Description:Inhibition of HDAC class 1 in human HT-29 cells using Boc-Lys-Ac as substrate incubated for 3 hrs by microplate reader assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetHistone deacetylase 1/2/3/8(Human)
Stony Brook University

Curated by ChEMBL
LigandPNGBDBM50602708(CHEMBL5176419)
Affinity DataIC50: 1.50E+4nMAssay Description:Inhibition of HDAC class 1 in human HT-29 cells using Boc-Lys-Ac as substrate incubated for 3 hrs by microplate reader assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetHistone deacetylase 1/2/3/8(Human)
Stony Brook University

Curated by ChEMBL
LigandPNGBDBM162865(US9056843, 156)
Affinity DataIC50: 1.50E+4nMAssay Description:Inhibition of HDAC class 1 in human HT-29 cells using Boc-Lys-Ac as substrate incubated for 3 hrs by microplate reader assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetHistone deacetylase 1/2/3/8(Human)
Stony Brook University

Curated by ChEMBL
LigandPNGBDBM50602706(CHEMBL5199111)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of HDAC class 1 in human HT-29 cells using Boc-Lys-Ac as substrate incubated for 3 hrs by microplate reader assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetHistone deacetylase 1/2/3/8(Human)
Stony Brook University

Curated by ChEMBL
LigandPNGBDBM50602697(CHEMBL5197621)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of HDAC class 1 in human HT-29 cells using Boc-Lys-Ac as substrate incubated for 3 hrs by microplate reader assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetHistone deacetylase 1/2/3/8(Human)
Stony Brook University

Curated by ChEMBL
LigandPNGBDBM50602696(CHEMBL5206794)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of HDAC class 1 in human HT-29 cells using Boc-Lys-Ac as substrate incubated for 3 hrs by microplate reader assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetHistone deacetylase 1/2/3/8(Human)
Stony Brook University

Curated by ChEMBL
LigandPNGBDBM50602695(CHEMBL5194933)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of HDAC class 1 in human HT-29 cells using Boc-Lys-Ac as substrate incubated for 3 hrs by microplate reader assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetHistone deacetylase 1/2/3/8(Human)
Stony Brook University

Curated by ChEMBL
LigandPNGBDBM50563276(CHEMBL4751615)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of HDAC class 1 in human HT-29 cells using Boc-Lys-Ac as substrate incubated for 3 hrs by microplate reader assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetHistone deacetylase 1/2/3/8(Human)
Stony Brook University

Curated by ChEMBL
LigandPNGBDBM50602707(CHEMBL5190668)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of HDAC class 1 in human HT-29 cells using Boc-Lys-Ac as substrate incubated for 3 hrs by microplate reader assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed