Compile Data Set for Download or QSAR
Report error Found 7 Enz. Inhib. hit(s) with all data for entry = 50015218
TargetCyclin-dependent kinase 12(Human)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50583997(CHEMBL5073005)
Affinity DataIC50: 66nMAssay Description:Inhibition of human CDK12 (696 to 1082 residues) /cyclinK (1 to 300 residues) using ac-YSPTSPpSYSPTSFpS-YSPTSPpSY-[PEG2]-RR-amid peptide as substrate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2023
Entry Details Article
PubMed
TargetCyclin-dependent kinase 12(Human)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50584001(CHEMBL5089202)
Affinity DataIC50: 119nMAssay Description:Inhibition of human CDK12 (696 to 1082 residues) /cyclinK (1 to 300 residues) using ac-YSPTSPpSYSPTSFpS-YSPTSPpSY-[PEG2]-RR-amid peptide as substrate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2023
Entry Details Article
PubMed
TargetCyclin-dependent kinase 12(Human)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50583998(CHEMBL5074219)
Affinity DataIC50: 237nMAssay Description:Inhibition of human CDK12 (696 to 1082 residues) /cyclinK (1 to 300 residues) using ac-YSPTSPpSYSPTSFpS-YSPTSPpSY-[PEG2]-RR-amid peptide as substrate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2023
Entry Details Article
PubMed
TargetCyclin-dependent kinase 12(Human)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50583999(CHEMBL5084858)
Affinity DataIC50: 411nMAssay Description:Inhibition of human CDK12 (696 to 1082 residues) /cyclinK (1 to 300 residues) using ac-YSPTSPpSYSPTSFpS-YSPTSPpSY-[PEG2]-RR-amid peptide as substrate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2023
Entry Details Article
PubMed
TargetCyclin-dependent kinase 12(Human)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50584000(CHEMBL4877117)
Affinity DataIC50: 469nMAssay Description:Inhibition of human CDK12 (696 to 1082 residues) /cyclinK (1 to 300 residues) using ac-YSPTSPpSYSPTSFpS-YSPTSPpSY-[PEG2]-RR-amid peptide as substrate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2023
Entry Details Article
PubMed
TargetCyclin-dependent kinase 12(Human)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50584002(CHEMBL5082914)
Affinity DataIC50: 645nMAssay Description:Inhibition of human CDK12 (696 to 1082 residues) /cyclinK (1 to 300 residues) using ac-YSPTSPpSYSPTSFpS-YSPTSPpSY-[PEG2]-RR-amid peptide as substrate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2023
Entry Details Article
PubMed
TargetCyclin-dependent kinase 12(Human)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50584003(CHEMBL5087182)
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of human CDK12 (696 to 1082 residues) /cyclinK (1 to 300 residues) using ac-YSPTSPpSYSPTSFpS-YSPTSPpSY-[PEG2]-RR-amid peptide as substrate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2023
Entry Details Article
PubMed