Compile Data Set for Download or QSAR
Report error Found 34 Enz. Inhib. hit(s) with all data for entry = 50017071
TargetSodium/glucose cotransporter 2(Human)
Gc Pharma

Curated by ChEMBL
LigandPNGBDBM159528(US9034921, E171 | US9340521, E028)
Affinity DataIC50: 0.370nMAssay Description:Inhibition of human SGLT2 expressed in CHO cells by methyl-alpha-D-glucopyranoside assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetSodium/glucose cotransporter 2(Human)
Gc Pharma

Curated by ChEMBL
LigandPNGBDBM159387(US9034921, E001 | US9340521, E001)
Affinity DataIC50: 0.440nMAssay Description:Inhibition of human SGLT2 expressed in CHO cells by methyl-alpha-D-glucopyranoside assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetSodium/glucose cotransporter 2(Human)
Gc Pharma

Curated by ChEMBL
LigandPNGBDBM159529(US9034921, E172)
Affinity DataIC50: 0.460nMAssay Description:Inhibition of human SGLT2 expressed in CHO cells by methyl-alpha-D-glucopyranoside assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetSodium/glucose cotransporter 2(Human)
Gc Pharma

Curated by ChEMBL
LigandPNGBDBM20880(CHEMBL429910 | C-aryl glucoside, 6 | BMS-512148 | ...)
Affinity DataIC50: 0.490nMAssay Description:Inhibition of human SGLT2 expressed in CHO cells by methyl-alpha-D-glucopyranoside assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetSodium/glucose cotransporter 2(Human)
Gc Pharma

Curated by ChEMBL
LigandPNGBDBM159391(US9034921, E005 | US9340521, E004)
Affinity DataIC50: 0.680nMAssay Description:Inhibition of human SGLT2 expressed in CHO cells by methyl-alpha-D-glucopyranoside assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetSodium/glucose cotransporter 2(Human)
Gc Pharma

Curated by ChEMBL
LigandPNGBDBM159403(US9034921, E020)
Affinity DataIC50: 0.720nMAssay Description:Inhibition of human SGLT2 expressed in CHO cells by methyl-alpha-D-glucopyranoside assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetSodium/glucose cotransporter 2(Human)
Gc Pharma

Curated by ChEMBL
LigandPNGBDBM159538(US9034921, E181)
Affinity DataIC50: 0.790nMAssay Description:Inhibition of human SGLT2 expressed in CHO cells by methyl-alpha-D-glucopyranoside assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetSodium/glucose cotransporter 2(Human)
Gc Pharma

Curated by ChEMBL
LigandPNGBDBM159393(US9034921, E009 | US9034921, E007 | US9340521, E00...)
Affinity DataIC50: 0.790nMAssay Description:Inhibition of human SGLT2 expressed in CHO cells by methyl-alpha-D-glucopyranoside assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetSodium/glucose cotransporter 2(Human)
Gc Pharma

Curated by ChEMBL
LigandPNGBDBM159400(US9034921, E016 | US9340521, E010)
Affinity DataIC50: 0.980nMAssay Description:Inhibition of human SGLT2 expressed in CHO cells by methyl-alpha-D-glucopyranoside assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetSodium/glucose cotransporter 2(Human)
Gc Pharma

Curated by ChEMBL
LigandPNGBDBM159544(US9034921, E187)
Affinity DataIC50: 1.20nMAssay Description:Inhibition of human SGLT2 expressed in CHO cells by methyl-alpha-D-glucopyranoside assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetSodium/glucose cotransporter 2(Human)
Gc Pharma

Curated by ChEMBL
LigandPNGBDBM159590(US9034921, E233)
Affinity DataIC50: 1.20nMAssay Description:Inhibition of human SGLT2 expressed in CHO cells by methyl-alpha-D-glucopyranoside assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetSodium/glucose cotransporter 2(Human)
Gc Pharma

Curated by ChEMBL
LigandPNGBDBM159551(US9034921, E194)
Affinity DataIC50: 1.20nMAssay Description:Inhibition of human SGLT2 expressed in CHO cells by methyl-alpha-D-glucopyranoside assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetSodium/glucose cotransporter 2(Human)
Gc Pharma

Curated by ChEMBL
LigandPNGBDBM50599550(CHEMBL5208827)
Affinity DataIC50: 1.40nMAssay Description:Inhibition of human SGLT2 expressed in CHO cells by methyl-alpha-D-glucopyranoside assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetSodium/glucose cotransporter 2(Human)
Gc Pharma

Curated by ChEMBL
LigandPNGBDBM159402(US9034921, E019)
Affinity DataIC50: 1.5nMAssay Description:Inhibition of human SGLT2 expressed in CHO cells by methyl-alpha-D-glucopyranoside assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetSodium/glucose cotransporter 2(Human)
Gc Pharma

Curated by ChEMBL
LigandPNGBDBM159407(US9034921, E024)
Affinity DataIC50: 1.5nMAssay Description:Inhibition of human SGLT2 expressed in CHO cells by methyl-alpha-D-glucopyranoside assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetSodium/glucose cotransporter 2(Human)
Gc Pharma

Curated by ChEMBL
LigandPNGBDBM159404(US9034921, E021 | US9340521, E012)
Affinity DataIC50: 1.70nMAssay Description:Inhibition of human SGLT2 expressed in CHO cells by methyl-alpha-D-glucopyranoside assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetSodium/glucose cotransporter 2(Human)
Gc Pharma

Curated by ChEMBL
LigandPNGBDBM159392(US9034921, E006)
Affinity DataIC50: 2nMAssay Description:Inhibition of human SGLT2 expressed in CHO cells by methyl-alpha-D-glucopyranoside assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetSodium/glucose cotransporter 2(Human)
Gc Pharma

Curated by ChEMBL
LigandPNGBDBM159514(US9034921, E156 | US9340521, E023)
Affinity DataIC50: 2.10nMAssay Description:Inhibition of human SGLT2 expressed in CHO cells by methyl-alpha-D-glucopyranoside assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetSodium/glucose cotransporter 2(Human)
Gc Pharma

Curated by ChEMBL
LigandPNGBDBM159524(US9034921, E166)
Affinity DataIC50: 4.20nMAssay Description:Inhibition of human SGLT2 expressed in CHO cells by methyl-alpha-D-glucopyranoside assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetSodium/glucose cotransporter 2(Human)
Gc Pharma

Curated by ChEMBL
LigandPNGBDBM50599549(CHEMBL5205876)
Affinity DataIC50: 7.40nMAssay Description:Inhibition of human SGLT2 expressed in CHO cells by methyl-alpha-D-glucopyranoside assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetSodium/glucose cotransporter 1(Human)
Gc Pharma

Curated by ChEMBL
LigandPNGBDBM159387(US9034921, E001 | US9340521, E001)
Affinity DataIC50: 15nMAssay Description:Inhibition of human SGLT1 expressed in CHO cells by methyl-alpha-D-glucopyranoside assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetSodium/glucose cotransporter 1(Human)
Gc Pharma

Curated by ChEMBL
LigandPNGBDBM159400(US9034921, E016 | US9340521, E010)
Affinity DataIC50: 17nMAssay Description:Inhibition of human SGLT1 expressed in CHO cells by methyl-alpha-D-glucopyranoside assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetSodium/glucose cotransporter 1(Human)
Gc Pharma

Curated by ChEMBL
LigandPNGBDBM159404(US9034921, E021 | US9340521, E012)
Affinity DataIC50: 34nMAssay Description:Inhibition of human SGLT1 expressed in CHO cells by methyl-alpha-D-glucopyranoside assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetSodium/glucose cotransporter 1(Human)
Gc Pharma

Curated by ChEMBL
LigandPNGBDBM159391(US9034921, E005 | US9340521, E004)
Affinity DataIC50: 37nMAssay Description:Inhibition of human SGLT1 expressed in CHO cells by methyl-alpha-D-glucopyranoside assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetSodium/glucose cotransporter 1(Human)
Gc Pharma

Curated by ChEMBL
LigandPNGBDBM159514(US9034921, E156 | US9340521, E023)
Affinity DataIC50: 78nMAssay Description:Inhibition of human SGLT1 expressed in CHO cells by methyl-alpha-D-glucopyranoside assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetSodium/glucose cotransporter 1(Human)
Gc Pharma

Curated by ChEMBL
LigandPNGBDBM159528(US9034921, E171 | US9340521, E028)
Affinity DataIC50: 163nMAssay Description:Inhibition of human SGLT1 expressed in CHO cells by methyl-alpha-D-glucopyranoside assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetSodium/glucose cotransporter 1(Human)
Gc Pharma

Curated by ChEMBL
LigandPNGBDBM159529(US9034921, E172)
Affinity DataIC50: 359nMAssay Description:Inhibition of human SGLT1 expressed in CHO cells by methyl-alpha-D-glucopyranoside assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetSodium/glucose cotransporter 1(Human)
Gc Pharma

Curated by ChEMBL
LigandPNGBDBM159402(US9034921, E019)
Affinity DataIC50: 400nMAssay Description:Inhibition of human SGLT1 expressed in CHO cells by methyl-alpha-D-glucopyranoside assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetSodium/glucose cotransporter 1(Human)
Gc Pharma

Curated by ChEMBL
LigandPNGBDBM159403(US9034921, E020)
Affinity DataIC50: 556nMAssay Description:Inhibition of human SGLT1 expressed in CHO cells by methyl-alpha-D-glucopyranoside assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetSodium/glucose cotransporter 1(Human)
Gc Pharma

Curated by ChEMBL
LigandPNGBDBM159544(US9034921, E187)
Affinity DataIC50: 1.37E+3nMAssay Description:Inhibition of human SGLT1 expressed in CHO cells by methyl-alpha-D-glucopyranoside assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetSodium/glucose cotransporter 1(Human)
Gc Pharma

Curated by ChEMBL
LigandPNGBDBM159407(US9034921, E024)
Affinity DataIC50: 2.14E+3nMAssay Description:Inhibition of human SGLT1 expressed in CHO cells by methyl-alpha-D-glucopyranoside assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetSodium/glucose cotransporter 1(Human)
Gc Pharma

Curated by ChEMBL
LigandPNGBDBM159538(US9034921, E181)
Affinity DataIC50: 4.94E+3nMAssay Description:Inhibition of human SGLT1 expressed in CHO cells by methyl-alpha-D-glucopyranoside assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetSodium/glucose cotransporter 1(Human)
Gc Pharma

Curated by ChEMBL
LigandPNGBDBM159551(US9034921, E194)
Affinity DataIC50: 6.28E+3nMAssay Description:Inhibition of human SGLT1 expressed in CHO cells by methyl-alpha-D-glucopyranoside assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetSodium/glucose cotransporter 1(Human)
Gc Pharma

Curated by ChEMBL
LigandPNGBDBM159590(US9034921, E233)
Affinity DataIC50: 9.93E+3nMAssay Description:Inhibition of human SGLT1 expressed in CHO cells by methyl-alpha-D-glucopyranoside assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed