Compile Data Set for Download or QSAR
Report error Found 18 Enz. Inhib. hit(s) with all data for entry = 50015555
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Human)
Australian National University

Curated by ChEMBL
LigandPNGBDBM50587468(CHEMBL2296158)
Affinity DataIC50: 90nMAssay Description:Inhibition of human (alpha4)3(beta2)2 nAChR expressed in Xenopus laevis oocytes assessed as inhibition of acetylcholine-induced current response in p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Human)
Australian National University

Curated by ChEMBL
LigandPNGBDBM50587468(CHEMBL2296158)
Affinity DataIC50: 90nMAssay Description:Inhibition of human (alpha4)3(beta2)2 nAChR expressed in Xenopus laevis oocytes assessed as inhibition of acetylcholine-induced current response in p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Human)
Australian National University

Curated by ChEMBL
LigandPNGBDBM50587468(CHEMBL2296158)
Affinity DataIC50: 140nMAssay Description:Inhibition of human (alpha4)2(beta2)3 nAChR expressed in Xenopus laevis oocytes assessed as inhibition of acetylcholine-induced current response in p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Human)
Australian National University

Curated by ChEMBL
LigandPNGBDBM50587468(CHEMBL2296158)
Affinity DataIC50: 140nMAssay Description:Inhibition of human (alpha4)2(beta2)3 nAChR expressed in Xenopus laevis oocytes assessed as inhibition of acetylcholine-induced current response in p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Human)
Australian National University

Curated by ChEMBL
LigandPNGBDBM50587471(CHEMBL5082799)
Affinity DataIC50: 3.90E+3nMAssay Description:Inhibition of human (alpha4)3(beta2)2 nAChR expressed in Xenopus laevis oocytes assessed as inhibition of acetylcholine-induced current response in p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Human)
Australian National University

Curated by ChEMBL
LigandPNGBDBM50587471(CHEMBL5082799)
Affinity DataIC50: 3.90E+3nMAssay Description:Inhibition of human (alpha4)3(beta2)2 nAChR expressed in Xenopus laevis oocytes assessed as inhibition of acetylcholine-induced current response in p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Human)
Australian National University

Curated by ChEMBL
LigandPNGBDBM50587470(CHEMBL5084512)
Affinity DataIC50: 4.10E+3nMAssay Description:Inhibition of human (alpha4)3(beta2)2 nAChR expressed in Xenopus laevis oocytes assessed as inhibition of acetylcholine-induced current response in p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Human)
Australian National University

Curated by ChEMBL
LigandPNGBDBM50587470(CHEMBL5084512)
Affinity DataIC50: 4.10E+3nMAssay Description:Inhibition of human (alpha4)3(beta2)2 nAChR expressed in Xenopus laevis oocytes assessed as inhibition of acetylcholine-induced current response in p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rat)
Australian National University

Curated by ChEMBL
LigandPNGBDBM50587472(CHEMBL5089606)
Affinity DataIC50: 4.66E+3nMAssay Description:Inhibition of rat alpha4beta2 nAChR expressed in Xenopus laevis oocytes assessed as inhibition of acetylcholine-elicited current response measured at...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Human)
Australian National University

Curated by ChEMBL
LigandPNGBDBM50587469(CHEMBL5085133)
Affinity DataIC50: 4.90E+3nMAssay Description:Inhibition of human (alpha4)3(beta2)2 nAChR expressed in Xenopus laevis oocytes assessed as inhibition of acetylcholine-induced current response in p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Human)
Australian National University

Curated by ChEMBL
LigandPNGBDBM50587469(CHEMBL5085133)
Affinity DataIC50: 4.90E+3nMAssay Description:Inhibition of human (alpha4)3(beta2)2 nAChR expressed in Xenopus laevis oocytes assessed as inhibition of acetylcholine-induced current response in p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Human)
Australian National University

Curated by ChEMBL
LigandPNGBDBM50587471(CHEMBL5082799)
Affinity DataIC50: 1.50E+4nMAssay Description:Inhibition of human (alpha4)2(beta2)3 nAChR expressed in Xenopus laevis oocytes assessed as inhibition of acetylcholine-induced current response in p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Human)
Australian National University

Curated by ChEMBL
LigandPNGBDBM50587471(CHEMBL5082799)
Affinity DataIC50: 1.50E+4nMAssay Description:Inhibition of human (alpha4)2(beta2)3 nAChR expressed in Xenopus laevis oocytes assessed as inhibition of acetylcholine-induced current response in p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Rat)
Australian National University

Curated by ChEMBL
LigandPNGBDBM50587472(CHEMBL5089606)
Affinity DataIC50: 2.07E+4nMAssay Description:Inhibition of rat alpha7 nAChR expressed in Xenopus laevis oocytes assessed as inhibition of acetylcholine-elicited current response measured at hold...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Human)
Australian National University

Curated by ChEMBL
LigandPNGBDBM50587469(CHEMBL5085133)
Affinity DataIC50: 2.73E+4nMAssay Description:Inhibition of human (alpha4)2(beta2)3 nAChR expressed in Xenopus laevis oocytes assessed as inhibition of acetylcholine-induced current response in p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Human)
Australian National University

Curated by ChEMBL
LigandPNGBDBM50587469(CHEMBL5085133)
Affinity DataIC50: 2.73E+4nMAssay Description:Inhibition of human (alpha4)2(beta2)3 nAChR expressed in Xenopus laevis oocytes assessed as inhibition of acetylcholine-induced current response in p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Human)
Australian National University

Curated by ChEMBL
LigandPNGBDBM50587470(CHEMBL5084512)
Affinity DataIC50: 2.91E+4nMAssay Description:Inhibition of human (alpha4)2(beta2)3 nAChR expressed in Xenopus laevis oocytes assessed as inhibition of acetylcholine-induced current response in p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Human)
Australian National University

Curated by ChEMBL
LigandPNGBDBM50587470(CHEMBL5084512)
Affinity DataIC50: 2.91E+4nMAssay Description:Inhibition of human (alpha4)2(beta2)3 nAChR expressed in Xenopus laevis oocytes assessed as inhibition of acetylcholine-induced current response in p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed