Compile Data Set for Download or QSAR
Report error Found 10 Enz. Inhib. hit(s) with all data for entry = 50014768
TargetCyclin-dependent kinase 8(Human)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50579915(CHEMBL4442570)
Affinity DataIC50: 4.5nMAssay Description:Inhibition of CDK8 in human HEK293 cells measured by NanoBRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/4/2023
Entry Details Article
PubMed
TargetCyclin-dependent kinase 8(Human)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50579909(CHEMBL5076378)
Affinity DataIC50: 31nMAssay Description:Inhibition of CDK8 in human HEK293 cells measured by NanoBRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/4/2023
Entry Details Article
PubMed
TargetCyclin-dependent kinase 8(Human)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM576465(US11471446, Compound DBA-6)
Affinity DataIC50: 31nMAssay Description:Inhibition of CDK8 in human HEK293 cells measured by NanoBRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/4/2023
Entry Details Article
PubMed
TargetCyclin-dependent kinase 8(Human)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50579911(CHEMBL5090279)
Affinity DataIC50: 33nMAssay Description:Inhibition of CDK8 in human HEK293 cells measured by NanoBRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/4/2023
Entry Details Article
PubMed
TargetCyclin-dependent kinase 8(Human)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50579914(CHEMBL5071605)
Affinity DataIC50: 33nMAssay Description:Inhibition of CDK8 in human HEK293 cells measured by NanoBRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/4/2023
Entry Details Article
PubMed
TargetCyclin-dependent kinase 8(Human)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50579912(CHEMBL5083027)
Affinity DataIC50: 34nMAssay Description:Inhibition of CDK8 in human HEK293 cells measured by NanoBRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/4/2023
Entry Details Article
PubMed
TargetCyclin-dependent kinase 8(Human)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50579910(CHEMBL5078832)
Affinity DataIC50: 93nMAssay Description:Inhibition of CDK8 in human HEK293 cells measured by NanoBRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/4/2023
Entry Details Article
PubMed
TargetCyclin-dependent kinase 8(Human)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50579907(CHEMBL2348334)
Affinity DataIC50: 130nMAssay Description:Inhibition of CDK8 in human HEK293 cells measured by NanoBRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/4/2023
Entry Details Article
PubMed
TargetCyclin-dependent kinase 8(Human)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50579913(CHEMBL5088336)
Affinity DataIC50: 410nMAssay Description:Inhibition of CDK8 in human HEK293 cells measured by NanoBRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/4/2023
Entry Details Article
PubMed
TargetCyclin-dependent kinase 8(Human)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50579908(CHEMBL5093576)
Affinity DataIC50: 520nMAssay Description:Inhibition of CDK8 in human HEK293 cells measured by NanoBRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/4/2023
Entry Details Article
PubMed