Compile Data Set for Download or QSAR
Report error Found 20 Enz. Inhib. hit(s) with all data for entry = 50014058
TargetProlyl endopeptidase(Pig)
University of Helsinki

Curated by ChEMBL
LigandPNGBDBM50155838((S)-1-((S)-1-(4-phenylbutanoyl)pyrrolidine-2-carbo...)
Affinity DataIC50: 0.200nMAssay Description:Inhibition of recombinant porcine PREP expressed in Escherichia coli using Suc-Gly-Pro-AMC as substrate preincubated for 30 mins followed by substrat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2022
Entry Details Article
PubMed
TargetProlyl endopeptidase(Pig)
University of Helsinki

Curated by ChEMBL
LigandPNGBDBM50037604(1-{(S)-2-[(S)-2-(1H-Imidazole-2-carbonyl)-pyrrolid...)
Affinity DataIC50: 1nMAssay Description:Inhibition of recombinant porcine PREP expressed in Escherichia coli using Suc-Gly-Pro-AMC as substrate preincubated for 30 mins followed by substrat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2022
Entry Details Article
PubMed
TargetProlyl endopeptidase(Pig)
University of Helsinki

Curated by ChEMBL
LigandPNGBDBM50572237(CHEMBL4862396)
Affinity DataIC50: 1nMAssay Description:Inhibition of recombinant porcine PREP expressed in Escherichia coli using Suc-Gly-Pro-AMC as substrate preincubated for 30 mins followed by substrat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2022
Entry Details Article
PubMed
TargetProlyl endopeptidase(Pig)
University of Helsinki

Curated by ChEMBL
LigandPNGBDBM50572235(CHEMBL4873431)
Affinity DataIC50: 1nMAssay Description:Inhibition of recombinant porcine PREP expressed in Escherichia coli using Suc-Gly-Pro-AMC as substrate preincubated for 30 mins followed by substrat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2022
Entry Details Article
PubMed
TargetProlyl endopeptidase(Pig)
University of Helsinki

Curated by ChEMBL
LigandPNGBDBM50572234(CHEMBL4861124)
Affinity DataIC50: 1nMAssay Description:Inhibition of recombinant porcine PREP expressed in Escherichia coli using Suc-Gly-Pro-AMC as substrate preincubated for 30 mins followed by substrat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2022
Entry Details Article
PubMed
TargetProlyl endopeptidase(Pig)
University of Helsinki

Curated by ChEMBL
LigandPNGBDBM50572238(CHEMBL4852321)
Affinity DataIC50: 44nMAssay Description:Inhibition of recombinant porcine PREP expressed in Escherichia coli using Suc-Gly-Pro-AMC as substrate preincubated for 30 mins followed by substrat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2022
Entry Details Article
PubMed
TargetProlyl endopeptidase(Pig)
University of Helsinki

Curated by ChEMBL
LigandPNGBDBM50572227(CHEMBL4849453)
Affinity DataIC50: 94nMAssay Description:Inhibition of recombinant porcine PREP expressed in Escherichia coli using Suc-Gly-Pro-AMC as substrate preincubated for 30 mins followed by substrat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2022
Entry Details Article
PubMed
TargetProlyl endopeptidase(Pig)
University of Helsinki

Curated by ChEMBL
LigandPNGBDBM50572225(CHEMBL4858172)
Affinity DataIC50: 770nMAssay Description:Inhibition of recombinant porcine PREP expressed in Escherichia coli using Suc-Gly-Pro-AMC as substrate preincubated for 30 mins followed by substrat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2022
Entry Details Article
PubMed
TargetProlyl endopeptidase(Pig)
University of Helsinki

Curated by ChEMBL
LigandPNGBDBM50572222(CHEMBL4859665)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of recombinant porcine PREP expressed in Escherichia coli using Suc-Gly-Pro-AMC as substrate preincubated for 30 mins followed by substrat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2022
Entry Details Article
PubMed
TargetProlyl endopeptidase(Pig)
University of Helsinki

Curated by ChEMBL
LigandPNGBDBM50572228(CHEMBL4846851)
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition of recombinant porcine PREP expressed in Escherichia coli using Suc-Gly-Pro-AMC as substrate preincubated for 30 mins followed by substrat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2022
Entry Details Article
PubMed
TargetProlyl endopeptidase(Pig)
University of Helsinki

Curated by ChEMBL
LigandPNGBDBM50572233(CHEMBL4853692)
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition of recombinant porcine PREP expressed in Escherichia coli using Suc-Gly-Pro-AMC as substrate preincubated for 30 mins followed by substrat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2022
Entry Details Article
PubMed
TargetProlyl endopeptidase(Pig)
University of Helsinki

Curated by ChEMBL
LigandPNGBDBM50572236(CHEMBL4878846)
Affinity DataIC50: 2.10E+3nMAssay Description:Inhibition of recombinant porcine PREP expressed in Escherichia coli using Suc-Gly-Pro-AMC as substrate preincubated for 30 mins followed by substrat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2022
Entry Details Article
PubMed
TargetProlyl endopeptidase(Pig)
University of Helsinki

Curated by ChEMBL
LigandPNGBDBM50572223(CHEMBL4861357)
Affinity DataIC50: 3.90E+3nMAssay Description:Inhibition of recombinant porcine PREP expressed in Escherichia coli using Suc-Gly-Pro-AMC as substrate preincubated for 30 mins followed by substrat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2022
Entry Details Article
PubMed
TargetProlyl endopeptidase(Pig)
University of Helsinki

Curated by ChEMBL
LigandPNGBDBM50572226(CHEMBL4876083)
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of recombinant porcine PREP expressed in Escherichia coli using Suc-Gly-Pro-AMC as substrate preincubated for 30 mins followed by substrat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2022
Entry Details Article
PubMed
TargetProlyl endopeptidase(Pig)
University of Helsinki

Curated by ChEMBL
LigandPNGBDBM50572230(CHEMBL4852805)
Affinity DataIC50: 1.20E+4nMAssay Description:Inhibition of recombinant porcine PREP expressed in Escherichia coli using Suc-Gly-Pro-AMC as substrate preincubated for 30 mins followed by substrat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2022
Entry Details Article
PubMed
TargetProlyl endopeptidase(Pig)
University of Helsinki

Curated by ChEMBL
LigandPNGBDBM50572231(CHEMBL4857482)
Affinity DataIC50: 2.90E+4nMAssay Description:Inhibition of recombinant porcine PREP expressed in Escherichia coli using Suc-Gly-Pro-AMC as substrate preincubated for 30 mins followed by substrat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2022
Entry Details Article
PubMed
TargetProlyl endopeptidase(Pig)
University of Helsinki

Curated by ChEMBL
LigandPNGBDBM50572232(CHEMBL4860555)
Affinity DataIC50: 5.50E+4nMAssay Description:Inhibition of recombinant porcine PREP expressed in Escherichia coli using Suc-Gly-Pro-AMC as substrate preincubated for 30 mins followed by substrat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2022
Entry Details Article
PubMed
TargetProlyl endopeptidase(Pig)
University of Helsinki

Curated by ChEMBL
LigandPNGBDBM50572224(CHEMBL4867363)
Affinity DataIC50: 6.20E+4nMAssay Description:Inhibition of recombinant porcine PREP expressed in Escherichia coli using Suc-Gly-Pro-AMC as substrate preincubated for 30 mins followed by substrat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2022
Entry Details Article
PubMed
TargetProlyl endopeptidase(Pig)
University of Helsinki

Curated by ChEMBL
LigandPNGBDBM50572239(CHEMBL4864967)
Affinity DataIC50: 7.00E+4nMAssay Description:Inhibition of recombinant porcine PREP expressed in Escherichia coli using Suc-Gly-Pro-AMC as substrate preincubated for 30 mins followed by substrat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2022
Entry Details Article
PubMed
TargetProlyl endopeptidase(Pig)
University of Helsinki

Curated by ChEMBL
LigandPNGBDBM50572229(CHEMBL4864903)
Affinity DataIC50: 5.20E+5nMAssay Description:Inhibition of recombinant porcine PREP expressed in Escherichia coli using Suc-Gly-Pro-AMC as substrate preincubated for 30 mins followed by substrat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2022
Entry Details Article
PubMed