Compile Data Set for Download or QSAR
Report error Found 27 Enz. Inhib. hit(s) with all data for entry = 50014348
TargetPresenilin-1(Human)
University of Kansas

Curated by ChEMBL
LigandPNGBDBM50575197(CHEMBL4868549)
Affinity DataIC50: 0.700nMAssay Description:Inhibition of gamma secretase (unknown origin) expressed in HEK293 cells assessed as reduction of A-beta40 levels using C100-FLAG as substrate incuba...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2022
Entry Details Article
PubMed
TargetPresenilin-1(Human)
University of Kansas

Curated by ChEMBL
LigandPNGBDBM50575178(CHEMBL4853450)
Affinity DataIC50: 0.800nMAssay Description:Inhibition of gamma secretase (unknown origin) expressed in HEK293 cells assessed as reduction of A-beta40 levels using C100-FLAG as substrate incuba...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2022
Entry Details Article
PubMed
TargetPresenilin-1(Human)
University of Kansas

Curated by ChEMBL
LigandPNGBDBM50575198(CHEMBL4848394)
Affinity DataIC50: 0.870nMAssay Description:Inhibition of gamma secretase (unknown origin) expressed in HEK293 cells assessed as reduction of A-beta40 levels using C100-FLAG as substrate incuba...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2022
Entry Details Article
PubMed
TargetPresenilin-1(Human)
University of Kansas

Curated by ChEMBL
LigandPNGBDBM50575196(CHEMBL4862085)
Affinity DataIC50: 1.10nMAssay Description:Inhibition of gamma secretase (unknown origin) expressed in HEK293 cells assessed as reduction of A-beta40 levels using C100-FLAG as substrate incuba...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2022
Entry Details Article
PubMed
TargetPresenilin-1(Human)
University of Kansas

Curated by ChEMBL
LigandPNGBDBM50575195(CHEMBL4874185)
Affinity DataIC50: 1.5nMAssay Description:Inhibition of gamma secretase (unknown origin) expressed in HEK293 cells assessed as reduction of A-beta40 levels using C100-FLAG as substrate incuba...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2022
Entry Details Article
PubMed
TargetPresenilin-1(Human)
University of Kansas

Curated by ChEMBL
LigandPNGBDBM50575180(CHEMBL4874349)
Affinity DataIC50: 1.90nMAssay Description:Inhibition of gamma secretase (unknown origin) expressed in HEK293 cells assessed as reduction of A-beta40 levels using C100-FLAG as substrate incuba...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2022
Entry Details Article
PubMed
TargetPresenilin-1(Human)
University of Kansas

Curated by ChEMBL
LigandPNGBDBM50575187(CHEMBL4848116)
Affinity DataIC50: 2.10nMAssay Description:Inhibition of gamma secretase (unknown origin) expressed in HEK293 cells assessed as reduction of A-beta40 levels using C100-FLAG as substrate incuba...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2022
Entry Details Article
PubMed
TargetPresenilin-1(Human)
University of Kansas

Curated by ChEMBL
LigandPNGBDBM50575194(CHEMBL4863759)
Affinity DataIC50: 3.20nMAssay Description:Inhibition of gamma secretase (unknown origin) expressed in HEK293 cells assessed as reduction of A-beta40 levels using C100-FLAG as substrate incuba...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2022
Entry Details Article
PubMed
TargetPresenilin-1(Human)
University of Kansas

Curated by ChEMBL
LigandPNGBDBM50575179(CHEMBL4851959)
Affinity DataIC50: 4.40nMAssay Description:Inhibition of gamma secretase (unknown origin) expressed in HEK293 cells assessed as reduction of A-beta40 levels using C100-FLAG as substrate incuba...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2022
Entry Details Article
PubMed
TargetPresenilin-1(Human)
University of Kansas

Curated by ChEMBL
LigandPNGBDBM50575188(CHEMBL4866068)
Affinity DataIC50: 5.70nMAssay Description:Inhibition of gamma secretase (unknown origin) expressed in HEK293 cells assessed as reduction of A-beta40 levels using C100-FLAG as substrate incuba...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2022
Entry Details Article
PubMed
TargetPresenilin-1(Human)
University of Kansas

Curated by ChEMBL
LigandPNGBDBM50575193(CHEMBL4854028)
Affinity DataIC50: 6nMAssay Description:Inhibition of gamma secretase (unknown origin) expressed in HEK293 cells assessed as reduction of A-beta40 levels using C100-FLAG as substrate incuba...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2022
Entry Details Article
PubMed
TargetPresenilin-1(Human)
University of Kansas

Curated by ChEMBL
LigandPNGBDBM50575192(CHEMBL4870824)
Affinity DataIC50: 7.5nMAssay Description:Inhibition of gamma secretase (unknown origin) expressed in HEK293 cells assessed as reduction of A-beta40 levels using C100-FLAG as substrate incuba...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2022
Entry Details Article
PubMed
TargetPresenilin-1(Human)
University of Kansas

Curated by ChEMBL
LigandPNGBDBM50575189(CHEMBL4865718)
Affinity DataIC50: 7.70nMAssay Description:Inhibition of gamma secretase (unknown origin) expressed in HEK293 cells assessed as reduction of A-beta40 levels using C100-FLAG as substrate incuba...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2022
Entry Details Article
PubMed
TargetPresenilin-1(Human)
University of Kansas

Curated by ChEMBL
LigandPNGBDBM50575190(CHEMBL4850432)
Affinity DataIC50: 8.30nMAssay Description:Inhibition of gamma secretase (unknown origin) expressed in HEK293 cells assessed as reduction of A-beta40 levels using C100-FLAG as substrate incuba...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2022
Entry Details Article
PubMed
TargetPresenilin-1(Human)
University of Kansas

Curated by ChEMBL
LigandPNGBDBM50575191(CHEMBL4846563)
Affinity DataIC50: 35nMAssay Description:Inhibition of gamma secretase (unknown origin) expressed in HEK293 cells assessed as reduction of A-beta40 levels using C100-FLAG as substrate incuba...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2022
Entry Details Article
PubMed
LigandPNGBDBM50575176(CHEMBL4869215)
Affinity DataIC50: 41nMAssay Description:Inhibition of gamma secretase (unknown origin) expressed in HEK293 cells assessed as reduction of A-beta40 levels using C100-FLAG as substrate incuba...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2022
Entry Details Article
PubMed
TargetPresenilin-1(Human)
University of Kansas

Curated by ChEMBL
LigandPNGBDBM50575184(CHEMBL4856827)
Affinity DataIC50: 42nMAssay Description:Inhibition of gamma secretase (unknown origin) expressed in HEK293 cells assessed as reduction of A-beta40 levels using C100-FLAG as substrate incuba...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2022
Entry Details Article
PubMed
TargetPresenilin-1(Human)
University of Kansas

Curated by ChEMBL
LigandPNGBDBM50575177(CHEMBL4850178)
Affinity DataIC50: 58nMAssay Description:Inhibition of gamma secretase (unknown origin) expressed in HEK293 cells assessed as reduction of A-beta40 levels using C100-FLAG as substrate incuba...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2022
Entry Details Article
PubMed
TargetPresenilin-1(Human)
University of Kansas

Curated by ChEMBL
LigandPNGBDBM50575181(CHEMBL4871750)
Affinity DataIC50: 59nMAssay Description:Inhibition of gamma secretase (unknown origin) expressed in HEK293 cells assessed as reduction of A-beta40 levels using C100-FLAG as substrate incuba...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2022
Entry Details Article
PubMed
TargetPresenilin-1(Human)
University of Kansas

Curated by ChEMBL
LigandPNGBDBM50575185(CHEMBL4867372)
Affinity DataIC50: 81nMAssay Description:Inhibition of gamma secretase (unknown origin) expressed in HEK293 cells assessed as reduction of A-beta40 levels using C100-FLAG as substrate incuba...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2022
Entry Details Article
PubMed
TargetPresenilin-1(Human)
University of Kansas

Curated by ChEMBL
LigandPNGBDBM50575186(CHEMBL4857927)
Affinity DataIC50: 98nMAssay Description:Inhibition of gamma secretase (unknown origin) expressed in HEK293 cells assessed as reduction of A-beta40 levels using C100-FLAG as substrate incuba...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2022
Entry Details Article
PubMed
TargetPresenilin-1(Human)
University of Kansas

Curated by ChEMBL
LigandPNGBDBM50575183(CHEMBL4867660)
Affinity DataIC50: 114nMAssay Description:Inhibition of gamma secretase (unknown origin) expressed in HEK293 cells assessed as reduction of A-beta40 levels using C100-FLAG as substrate incuba...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2022
Entry Details Article
PubMed
TargetPresenilin-1(Human)
University of Kansas

Curated by ChEMBL
LigandPNGBDBM50575182(CHEMBL4858881)
Affinity DataIC50: 188nMAssay Description:Inhibition of gamma secretase (unknown origin) expressed in HEK293 cells assessed as reduction of A-beta40 levels using C100-FLAG as substrate incuba...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2022
Entry Details Article
PubMed
TargetPresenilin-1(Human)
University of Kansas

Curated by ChEMBL
LigandPNGBDBM50575178(CHEMBL4853450)
Affinity DataKi:  0.420nMAssay Description:Noncompetitive inhibition of gamma secretase (unknown origin) expressed in HEK293 cells assessed as reduction of A-beta40 levels using varying level ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2022
Entry Details Article
PubMed
TargetPresenilin-1(Human)
University of Kansas

Curated by ChEMBL
LigandPNGBDBM50575197(CHEMBL4868549)
Affinity DataKi:  0.650nMAssay Description:Noncompetitive inhibition of gamma secretase (unknown origin) expressed in HEK293 cells assessed as reduction of A-beta40 levels using varying level ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2022
Entry Details Article
PubMed
TargetPresenilin-1(Human)
University of Kansas

Curated by ChEMBL
LigandPNGBDBM50575187(CHEMBL4848116)
Affinity DataKi:  1.20nMAssay Description:Noncompetitive inhibition of gamma secretase (unknown origin) expressed in HEK293 cells assessed as reduction of A-beta40 levels using varying level ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2022
Entry Details Article
PubMed
TargetPresenilin-1(Human)
University of Kansas

Curated by ChEMBL
LigandPNGBDBM50575179(CHEMBL4851959)
Affinity DataKi:  2.60nMAssay Description:Noncompetitive inhibition of gamma secretase (unknown origin) expressed in HEK293 cells assessed as reduction of A-beta40 levels using varying level ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2022
Entry Details Article
PubMed