Compile Data Set for Download or QSAR
Report error Found 21 Enz. Inhib. hit(s) with all data for entry = 50018407
TargetHTH-type quorum-sensing regulator RhlR(Pseudomonas aeruginosa (strain ATCC 15692 / PAO1 /...)
Zhengzhou University

Curated by ChEMBL
LigandPNGBDBM50608106(CHEMBL5267863)
Affinity DataEC50:  3.82E+3nMAssay Description:Agonist activity against RhlR in Pseudomonas aeruginosa PAO-JP2 expressing prhlI-LVAgfp using CPRG as substrate by spectrophotometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetHTH-type quorum-sensing regulator RhlR(Pseudomonas aeruginosa (strain ATCC 15692 / PAO1 /...)
Zhengzhou University

Curated by ChEMBL
LigandPNGBDBM50608105(CHEMBL5291457)
Affinity DataEC50:  1.41E+3nMAssay Description:Agonist activity against RhlR in Pseudomonas aeruginosa PAO-JP2 expressing prhlI-LVAgfp using CPRG as substrate by spectrophotometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetHTH-type quorum-sensing regulator RhlR(Pseudomonas aeruginosa (strain ATCC 15692 / PAO1 /...)
Zhengzhou University

Curated by ChEMBL
LigandPNGBDBM50608104(CHEMBL5266949)
Affinity DataEC50:  1.02E+3nMAssay Description:Agonist activity against RhlR in Pseudomonas aeruginosa PAO-JP2 expressing prhlI-LVAgfp using CPRG as substrate by spectrophotometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetTranscriptional activator protein LuxR(Vibrio fischeri (strain ATCC 700601 / ES114))
Zhengzhou University

Curated by ChEMBL
LigandPNGBDBM50526999(CHEMBL458201 | CHEBI:63789)
Affinity DataEC50:  3.00E+3nMAssay Description:Agonist activity against LuxR mediated quorum sensing system in Vibrio fischeri ES114 expressing luxI assessed as increase in luminescence intensity ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetTranscriptional activator protein LuxR(Vibrio fischeri (strain ATCC 700601 / ES114))
Zhengzhou University

Curated by ChEMBL
LigandPNGBDBM50241431((S)-2-(3-nitrophenyl)-N-(2-oxo-tetrahydrofuran-3-y...)
Affinity DataEC50:  300nMAssay Description:Agonist activity against LuxR mediated quorum sensing system in Vibrio fischeri ES114 expressing luxI assessed as increase in luminescence intensity ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetTranscriptional activator protein LuxR(Vibrio fischeri (strain ATCC 700601 / ES114))
Zhengzhou University

Curated by ChEMBL
LigandPNGBDBM50266163((S)-2-(4-iodophenyl)-N-(2-oxotetrahydrofuran-3-yl)...)
Affinity DataIC50: 600nMAssay Description:Antagonist activity against LuxR mediated quorum sensing system in Vibrio fischeri ES114 expressing luxI assessed as decrease in luminescence intensi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetTranscriptional activator protein LuxR(Vibrio fischeri (strain ATCC 700601 / ES114))
Zhengzhou University

Curated by ChEMBL
LigandPNGBDBM50266165((S)-N-(2-oxotetrahydrofuran-3-yl)-2-(4-(trifluorom...)
Affinity DataIC50: 600nMAssay Description:Antagonist activity against LuxR mediated quorum sensing system in Vibrio fischeri ES114 expressing luxI assessed as decrease in luminescence intensi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetTranscriptional activator protein LuxR(Vibrio fischeri (strain ATCC 700601 / ES114))
Zhengzhou University

Curated by ChEMBL
LigandPNGBDBM50373105(CHEMBL259441)
Affinity DataIC50: 600nMAssay Description:Antagonist activity against LuxR mediated quorum sensing system in Vibrio fischeri ES114 expressing luxI assessed as decrease in luminescence intensi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetTranscriptional activator protein LuxR(Vibrio fischeri (strain ATCC 700601 / ES114))
Zhengzhou University

Curated by ChEMBL
LigandPNGBDBM50608092(CHEMBL473573)
Affinity DataIC50: 600nMAssay Description:Antagonist activity against LuxR mediated quorum sensing system in Vibrio fischeri ES114 expressing luxI assessed as decrease in luminescence intensi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetTranscriptional activator protein LuxR(Vibrio fischeri (strain ATCC 700601 / ES114))
Zhengzhou University

Curated by ChEMBL
LigandPNGBDBM50527012(CHEMBL4571277)
Affinity DataIC50: 600nMAssay Description:Antagonist activity against LuxR mediated quorum sensing system in Vibrio fischeri ES114 expressing luxI assessed as decrease in luminescence intensi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetTranscriptional activator protein LasR(Pseudomonas aeruginosa (strain ATCC 15692 / PAO1 /...)
Zhengzhou University

Curated by ChEMBL
LigandPNGBDBM50608093(CHEMBL5289392)
Affinity DataIC50: 1.74E+4nMAssay Description:Antagonist activity against LasR-mediated quorum sensing system in Pseudomonas aeruginosa PAO1 by spectrophotometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetTranscriptional activator protein LasR(Pseudomonas aeruginosa (strain ATCC 15692 / PAO1 /...)
Zhengzhou University

Curated by ChEMBL
LigandPNGBDBM50608094(CHEMBL5278841)
Affinity DataIC50: 2.65E+4nMAssay Description:Antagonist activity against LasR-mediated quorum sensing system in Pseudomonas aeruginosa PAO1 by spectrophotometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetTranscriptional activator protein LasR(Pseudomonas aeruginosa (strain ATCC 15692 / PAO1 /...)
Zhengzhou University

Curated by ChEMBL
LigandPNGBDBM50608095(CHEMBL5276204)
Affinity DataIC50: 3.76E+4nMAssay Description:Antagonist activity against LasR-mediated quorum sensing system in Pseudomonas aeruginosa PAO1 by spectrophotometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetTranscriptional activator protein LasR(Pseudomonas aeruginosa (strain ATCC 15692 / PAO1 /...)
Zhengzhou University

Curated by ChEMBL
LigandPNGBDBM50608096(CHEMBL5288036)
Affinity DataIC50: 4.68E+4nMAssay Description:Antagonist activity against LasR-mediated quorum sensing system in Pseudomonas aeruginosa PAO1 by spectrophotometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetTranscriptional activator protein LasR(Pseudomonas aeruginosa (strain ATCC 15692 / PAO1 /...)
Zhengzhou University

Curated by ChEMBL
LigandPNGBDBM50608097(CHEMBL5288514)
Affinity DataIC50: 4.68E+4nMAssay Description:Antagonist activity against LasR-mediated quorum sensing system in Pseudomonas aeruginosa PAO1 by spectrophotometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetTranscriptional activator protein LasR(Pseudomonas aeruginosa (strain ATCC 15692 / PAO1 /...)
Zhengzhou University

Curated by ChEMBL
LigandPNGBDBM50608098(CHEMBL5285099)
Affinity DataIC50: 4.68E+4nMAssay Description:Antagonist activity against LasR-mediated quorum sensing system in Pseudomonas aeruginosa PAO1 by spectrophotometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetTranscriptional activator protein LasR(Pseudomonas aeruginosa (strain ATCC 15692 / PAO1 /...)
Zhengzhou University

Curated by ChEMBL
LigandPNGBDBM50608099(CHEMBL5284855)
Affinity DataIC50: 4.68E+4nMAssay Description:Antagonist activity against LasR-mediated quorum sensing system in Pseudomonas aeruginosa PAO1 by spectrophotometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetTranscriptional activator protein LasR(Pseudomonas aeruginosa (strain ATCC 15692 / PAO1 /...)
Zhengzhou University

Curated by ChEMBL
LigandPNGBDBM50608100(CHEMBL5267270)
Affinity DataIC50: 4.68E+4nMAssay Description:Antagonist activity against LasR-mediated quorum sensing system in Pseudomonas aeruginosa PAO1 by spectrophotometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetTranscriptional activator protein LasR(Pseudomonas aeruginosa (strain ATCC 15692 / PAO1 /...)
Zhengzhou University

Curated by ChEMBL
LigandPNGBDBM50608102(CHEMBL5280601)
Affinity DataIC50: 5.65E+4nMAssay Description:Antagonist activity against LasR-mediated quorum sensing system in Pseudomonas aeruginosa PAO1 by spectrophotometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetTranscriptional activator protein LasR(Pseudomonas aeruginosa (strain ATCC 15692 / PAO1 /...)
Zhengzhou University

Curated by ChEMBL
LigandPNGBDBM50608103(CHEMBL5273161)
Affinity DataIC50: 6.25E+4nMAssay Description:Antagonist activity against LasR-mediated quorum sensing system in Pseudomonas aeruginosa PAO1 by spectrophotometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetTranscriptional activator protein LasR(Pseudomonas aeruginosa (strain ATCC 15692 / PAO1 /...)
Zhengzhou University

Curated by ChEMBL
LigandPNGBDBM50608101(CHEMBL5283130)
Affinity DataIC50: 6.78E+4nMAssay Description:Antagonist activity against LasR-mediated quorum sensing system in Pseudomonas aeruginosa PAO1 by spectrophotometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed