Compile Data Set for Download or QSAR
Report error Found 14 Enz. Inhib. hit(s) with all data for entry = 50017047
TargetStructural capsid protein(Human immunodeficiency virus type 1)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50599340(CHEMBL5191897)
Affinity DataKd:  6.42E+3nMAssay Description:Binding affinity to HIV1 capsid protein monomer assessed as dissociation constant by SPR analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetStructural capsid protein(Human immunodeficiency virus type 1)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50599341(CHEMBL5202526)
Affinity DataKd:  7.79E+3nMAssay Description:Binding affinity to HIV1 capsid protein monomer assessed as dissociation constant by SPR analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetStructural capsid protein(Human immunodeficiency virus type 1)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50511740(CHEMBL4471665)
Affinity DataKd:  1.39E+4nMAssay Description:Binding affinity to HIV1 capsid protein monomer assessed as dissociation constant by SPR analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetStructural capsid protein(Human immunodeficiency virus type 1)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50467395(CHEMBL1229713)
Affinity DataKd:  3.41E+3nMAssay Description:Binding affinity to HIV1 capsid protein monomer assessed as dissociation constant by SPR analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetStructural capsid protein(Human immunodeficiency virus type 1)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50599340(CHEMBL5191897)
Affinity DataKd:  7.20E+3nMAssay Description:Binding affinity to HIV1 capsid protein hexamer assessed as dissociation constant by SPR analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetStructural capsid protein(Human immunodeficiency virus type 1)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50599341(CHEMBL5202526)
Affinity DataKd:  9.04E+3nMAssay Description:Binding affinity to HIV1 capsid protein hexamer assessed as dissociation constant by SPR analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetStructural capsid protein(Human immunodeficiency virus type 1)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50511740(CHEMBL4471665)
Affinity DataKd:  3.98E+3nMAssay Description:Binding affinity to HIV1 capsid protein hexamer assessed as dissociation constant by SPR analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetStructural capsid protein(Human immunodeficiency virus type 1)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50467395(CHEMBL1229713)
Affinity DataKd:  160nMAssay Description:Binding affinity to HIV1 capsid protein hexamer assessed as dissociation constant by SPR analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetStructural capsid protein(Human immunodeficiency virus type 1)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50599342(CHEMBL5208013)
Affinity DataKd:  3.55E+4nMAssay Description:Binding affinity to HIV1 capsid protein hexamer assessed as dissociation constant by SPR analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetStructural capsid protein(Human immunodeficiency virus type 1)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50599343(CHEMBL5189089)
Affinity DataKd:  9.44E+4nMAssay Description:Binding affinity to HIV1 capsid protein hexamer assessed as dissociation constant by SPR analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetStructural capsid protein(Human immunodeficiency virus type 1)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50467395(CHEMBL1229713)
Affinity DataIC50: 220nMAssay Description:Displacement of CPSF6 peptide from HIV1 capsid protein by surface plasmon resonance-based competition assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetStructural capsid protein(Human immunodeficiency virus type 1)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50599341(CHEMBL5202526)
Affinity DataIC50: 3.47E+3nMAssay Description:Displacement of NUP153 peptide from HIV1 capsid protein by surface plasmon resonance-based competition assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetStructural capsid protein(Human immunodeficiency virus type 1)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50467395(CHEMBL1229713)
Affinity DataIC50: 8.93E+3nMAssay Description:Displacement of NUP153 peptide from HIV1 capsid protein by surface plasmon resonance-based competition assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetStructural capsid protein(Human immunodeficiency virus type 1)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50599341(CHEMBL5202526)
Affinity DataIC50: 2.63E+4nMAssay Description:Displacement of CPSF6 peptide from HIV1 capsid protein by surface plasmon resonance-based competition assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed