Compile Data Set for Download or QSAR
Report error Found 18 Enz. Inhib. hit(s) with all data for entry = 50015518
TargetTyrosine-protein kinase BTK(Human)
Fudan University

Curated by ChEMBL
LigandPNGBDBM499812((2-chloro-4-phenoxyphenyl)(4- (((3S,6R)-6-(hydroxy...)
Affinity DataIC50: 0.390nMAssay Description:Inhibition of BTK C481S mutant (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetTyrosine-protein kinase BTK(Human)
Fudan University

Curated by ChEMBL
LigandPNGBDBM499812((2-chloro-4-phenoxyphenyl)(4- (((3S,6R)-6-(hydroxy...)
Affinity DataIC50: 0.850nMAssay Description:Inhibition of wild type BTK (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetTyrosine-protein kinase BTK(Human)
Fudan University

Curated by ChEMBL
LigandPNGBDBM499829((4-((cis-4-aminocyclohexyl)amino)-7H- pyrrolo[2,3-...)
Affinity DataIC50: 4.30nMAssay Description:Inhibition of full length N-terminal GST fusion tagged human BTK expressed in baculovirus expression system using FAM-P2 peptide solution as substrat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetTyrosine-protein kinase BTK(Human)
Fudan University

Curated by ChEMBL
LigandPNGBDBM499812((2-chloro-4-phenoxyphenyl)(4- (((3S,6R)-6-(hydroxy...)
Affinity DataIC50: 8.20nMAssay Description:Inhibition of full length N-terminal GST fusion tagged human BTK expressed in baculovirus expression system using FAM-P2 peptide solution as substrat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetTyrosine-protein kinase BTK(Human)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50587217(CHEMBL5075076)
Affinity DataIC50: 16nMAssay Description:Inhibition of full length N-terminal GST fusion tagged human BTK expressed in baculovirus expression system using FAM-P2 peptide solution as substrat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetTyrosine-protein kinase BTK(Human)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50587218(CHEMBL5089407)
Affinity DataIC50: 22nMAssay Description:Inhibition of full length N-terminal GST fusion tagged human BTK expressed in baculovirus expression system using FAM-P2 peptide solution as substrat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetTyrosine-protein kinase BTK(Human)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50587216(CHEMBL5094253)
Affinity DataIC50: 23nMAssay Description:Inhibition of full length N-terminal GST fusion tagged human BTK expressed in baculovirus expression system using FAM-P2 peptide solution as substrat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetTyrosine-protein kinase BTK(Human)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50587210(CHEMBL5077877)
Affinity DataIC50: 25nMAssay Description:Inhibition of full length N-terminal GST fusion tagged human BTK expressed in baculovirus expression system using FAM-P2 peptide solution as substrat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetTyrosine-protein kinase BTK(Human)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50587219(CHEMBL5087717)
Affinity DataIC50: 47nMAssay Description:Inhibition of full length N-terminal GST fusion tagged human BTK expressed in baculovirus expression system using FAM-P2 peptide solution as substrat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetTyrosine-protein kinase BTK(Human)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50587220(CHEMBL5071105)
Affinity DataIC50: 56nMAssay Description:Inhibition of full length N-terminal GST fusion tagged human BTK expressed in baculovirus expression system using FAM-P2 peptide solution as substrat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetTyrosine-protein kinase BTK(Human)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50587208(CHEMBL5076659)
Affinity DataIC50: 81nMAssay Description:Inhibition of full length N-terminal GST fusion tagged human BTK expressed in baculovirus expression system using FAM-P2 peptide solution as substrat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetTyrosine-protein kinase BTK(Human)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50587209(CHEMBL5085223)
Affinity DataIC50: 407nMAssay Description:Inhibition of full length N-terminal GST fusion tagged human BTK expressed in baculovirus expression system using FAM-P2 peptide solution as substrat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetTyrosine-protein kinase BTK(Human)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50587214(CHEMBL5085368)
Affinity DataIC50: 1.21E+3nMAssay Description:Inhibition of full length N-terminal GST fusion tagged human BTK expressed in baculovirus expression system using FAM-P2 peptide solution as substrat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetTyrosine-protein kinase BTK(Human)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50587215(CHEMBL5094571)
Affinity DataIC50: 1.39E+3nMAssay Description:Inhibition of full length N-terminal GST fusion tagged human BTK expressed in baculovirus expression system using FAM-P2 peptide solution as substrat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetTyrosine-protein kinase BTK(Human)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50587212(CHEMBL5082685)
Affinity DataIC50: 1.93E+3nMAssay Description:Inhibition of full length N-terminal GST fusion tagged human BTK expressed in baculovirus expression system using FAM-P2 peptide solution as substrat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetTyrosine-protein kinase BTK(Human)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50587213(CHEMBL5076235)
Affinity DataIC50: 2.20E+3nMAssay Description:Inhibition of full length N-terminal GST fusion tagged human BTK expressed in baculovirus expression system using FAM-P2 peptide solution as substrat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetTyrosine-protein kinase BTK(Human)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50587211(CHEMBL5089998)
Affinity DataIC50: 3.78E+3nMAssay Description:Inhibition of full length N-terminal GST fusion tagged human BTK expressed in baculovirus expression system using FAM-P2 peptide solution as substrat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetTyrosine-protein kinase BTK(Human)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50587207(CHEMBL5089431)
Affinity DataIC50: 5.97E+3nMAssay Description:Inhibition of full length N-terminal GST fusion tagged human BTK expressed in baculovirus expression system using FAM-P2 peptide solution as substrat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed