Report error Found 55 Enz. Inhib. hit(s) with all data for entry = 50014825
TargetMu-type opioid receptor(Human)
University of Health Sciences & Pharmacy At St. Louis
Curated by ChEMBL
University of Health Sciences & Pharmacy At St. Louis
Curated by ChEMBL
Affinity DataEC50: 5.93nMAssay Description:Agonist activity at human MOR expressed in HEK293T cells assessed as inhibition of forskolin-stimulated cAMP accumulation incubated for 30 mins by Gl...More data for this Ligand-Target Pair
TargetMu-type opioid receptor(Human)
University of Health Sciences & Pharmacy At St. Louis
Curated by ChEMBL
University of Health Sciences & Pharmacy At St. Louis
Curated by ChEMBL
Affinity DataEC50: 85nMAssay Description:Agonist activity at human MOR expressed in HEK293T cells assessed as inhibition of forskolin-stimulated cAMP accumulation incubated for 30 mins by Gl...More data for this Ligand-Target Pair
TargetMu-type opioid receptor(Human)
University of Health Sciences & Pharmacy At St. Louis
Curated by ChEMBL
University of Health Sciences & Pharmacy At St. Louis
Curated by ChEMBL
Affinity DataEC50: 372nMAssay Description:Agonist activity at human MOR expressed in HEK293T cells assessed as inhibition of forskolin-stimulated cAMP accumulation incubated for 30 mins by Gl...More data for this Ligand-Target Pair
TargetMu-type opioid receptor(Human)
University of Health Sciences & Pharmacy At St. Louis
Curated by ChEMBL
University of Health Sciences & Pharmacy At St. Louis
Curated by ChEMBL
Affinity DataEC50: 105nMAssay Description:Agonist activity at human MOR expressed in HEK293T cells assessed as inhibition of forskolin-stimulated cAMP accumulation incubated for 30 mins by Gl...More data for this Ligand-Target Pair
TargetMu-type opioid receptor(Human)
University of Health Sciences & Pharmacy At St. Louis
Curated by ChEMBL
University of Health Sciences & Pharmacy At St. Louis
Curated by ChEMBL
Affinity DataEC50: 537nMAssay Description:Agonist activity at human MOR expressed in HEK293T cells assessed as inhibition of forskolin-stimulated cAMP accumulation incubated for 30 mins by Gl...More data for this Ligand-Target Pair
TargetMu-type opioid receptor(Human)
University of Health Sciences & Pharmacy At St. Louis
Curated by ChEMBL
University of Health Sciences & Pharmacy At St. Louis
Curated by ChEMBL
Affinity DataEC50: 30nMAssay Description:Agonist activity at human MOR expressed in HEK293T cells assessed as inhibition of forskolin-stimulated cAMP accumulation incubated for 30 mins by Gl...More data for this Ligand-Target Pair
TargetMu-type opioid receptor(Human)
University of Health Sciences & Pharmacy At St. Louis
Curated by ChEMBL
University of Health Sciences & Pharmacy At St. Louis
Curated by ChEMBL
Affinity DataEC50: 1.12E+3nMAssay Description:Agonist activity at human MOR expressed in HEK293T cells assessed as inhibition of forskolin-stimulated cAMP accumulation incubated for 30 mins by Gl...More data for this Ligand-Target Pair
TargetMu-type opioid receptor(Human)
University of Health Sciences & Pharmacy At St. Louis
Curated by ChEMBL
University of Health Sciences & Pharmacy At St. Louis
Curated by ChEMBL
Affinity DataEC50: 186nMAssay Description:Agonist activity at human MOR expressed in HEK293T cells assessed as inhibition of forskolin-stimulated cAMP accumulation incubated for 30 mins by Gl...More data for this Ligand-Target Pair
TargetMu-type opioid receptor(Human)
University of Health Sciences & Pharmacy At St. Louis
Curated by ChEMBL
University of Health Sciences & Pharmacy At St. Louis
Curated by ChEMBL
Affinity DataEC50: 71nMAssay Description:Agonist activity at human MOR expressed in HEK293T cells assessed as inhibition of forskolin-stimulated cAMP accumulation incubated for 30 mins by Gl...More data for this Ligand-Target Pair
TargetMu-type opioid receptor(Human)
University of Health Sciences & Pharmacy At St. Louis
Curated by ChEMBL
University of Health Sciences & Pharmacy At St. Louis
Curated by ChEMBL
Affinity DataEC50: 1.74E+4nMAssay Description:Agonist activity at human MOR expressed in HEK293T cells assessed as inhibition of forskolin-stimulated cAMP accumulation incubated for 30 mins by Gl...More data for this Ligand-Target Pair
TargetMu-type opioid receptor(Human)
University of Health Sciences & Pharmacy At St. Louis
Curated by ChEMBL
University of Health Sciences & Pharmacy At St. Louis
Curated by ChEMBL
Affinity DataEC50: 1.55E+3nMAssay Description:Agonist activity at human MOR expressed in HEK293T cells assessed as inhibition of forskolin-stimulated cAMP accumulation incubated for 30 mins by Gl...More data for this Ligand-Target Pair
TargetMu-type opioid receptor(Human)
University of Health Sciences & Pharmacy At St. Louis
Curated by ChEMBL
University of Health Sciences & Pharmacy At St. Louis
Curated by ChEMBL
Affinity DataEC50: 11nMAssay Description:Agonist activity at human MOR expressed in HEK293T cells assessed as inhibition of forskolin-stimulated cAMP accumulation incubated for 30 mins by Gl...More data for this Ligand-Target Pair
TargetMu-type opioid receptor(Human)
University of Health Sciences & Pharmacy At St. Louis
Curated by ChEMBL
University of Health Sciences & Pharmacy At St. Louis
Curated by ChEMBL
Affinity DataEC50: 7.20nMAssay Description:Agonist activity at human MOR expressed in HEK293T cells assessed as inhibition of forskolin-stimulated cAMP accumulation incubated for 30 mins by Gl...More data for this Ligand-Target Pair
TargetMu-type opioid receptor(Human)
University of Health Sciences & Pharmacy At St. Louis
Curated by ChEMBL
University of Health Sciences & Pharmacy At St. Louis
Curated by ChEMBL
Affinity DataEC50: 5.30nMAssay Description:Agonist activity at human MOR expressed in HEK293T cells assessed as inhibition of forskolin-stimulated cAMP accumulation incubated for 30 mins by Gl...More data for this Ligand-Target Pair
TargetMu-type opioid receptor(Human)
University of Health Sciences & Pharmacy At St. Louis
Curated by ChEMBL
University of Health Sciences & Pharmacy At St. Louis
Curated by ChEMBL
Affinity DataEC50: 0.490nMAssay Description:Agonist activity at human MOR expressed in HEK293T cells assessed as inhibition of forskolin-stimulated cAMP accumulation incubated for 30 mins by Gl...More data for this Ligand-Target Pair
TargetMu-type opioid receptor(Human)
University of Health Sciences & Pharmacy At St. Louis
Curated by ChEMBL
University of Health Sciences & Pharmacy At St. Louis
Curated by ChEMBL
Affinity DataEC50: 241nMAssay Description:Agonist activity at human MOR expressed in HEK293T cells assessed as inhibition of forskolin-stimulated cAMP accumulation incubated for 30 mins by Gl...More data for this Ligand-Target Pair
TargetMu-type opioid receptor(Human)
University of Health Sciences & Pharmacy At St. Louis
Curated by ChEMBL
University of Health Sciences & Pharmacy At St. Louis
Curated by ChEMBL
Affinity DataEC50: 1.92E+4nMAssay Description:Agonist activity at human MOR receptor expressed in HTLA cells co-expressing TEV-fused-beta-arrestin2 assessed as induction of beta-arrestin2 recruit...More data for this Ligand-Target Pair
TargetMu-type opioid receptor(Human)
University of Health Sciences & Pharmacy At St. Louis
Curated by ChEMBL
University of Health Sciences & Pharmacy At St. Louis
Curated by ChEMBL
Affinity DataEC50: 1.04E+4nMAssay Description:Agonist activity at human MOR receptor expressed in HTLA cells co-expressing TEV-fused-beta-arrestin2 assessed as induction of beta-arrestin2 recruit...More data for this Ligand-Target Pair
TargetMu-type opioid receptor(Human)
University of Health Sciences & Pharmacy At St. Louis
Curated by ChEMBL
University of Health Sciences & Pharmacy At St. Louis
Curated by ChEMBL
Affinity DataEC50: 1.10E+4nMAssay Description:Agonist activity at human MOR receptor expressed in HTLA cells co-expressing TEV-fused-beta-arrestin2 assessed as induction of beta-arrestin2 recruit...More data for this Ligand-Target Pair
TargetMu-type opioid receptor(Human)
University of Health Sciences & Pharmacy At St. Louis
Curated by ChEMBL
University of Health Sciences & Pharmacy At St. Louis
Curated by ChEMBL
Affinity DataEC50: 8.04E+3nMAssay Description:Agonist activity at human MOR receptor expressed in HTLA cells co-expressing TEV-fused-beta-arrestin2 assessed as induction of beta-arrestin2 recruit...More data for this Ligand-Target Pair
TargetMu-type opioid receptor(Human)
University of Health Sciences & Pharmacy At St. Louis
Curated by ChEMBL
University of Health Sciences & Pharmacy At St. Louis
Curated by ChEMBL
Affinity DataEC50: 182nMAssay Description:Agonist activity at human MOR receptor expressed in HTLA cells co-expressing TEV-fused-beta-arrestin2 assessed as induction of beta-arrestin2 recruit...More data for this Ligand-Target Pair
TargetMu-type opioid receptor(Human)
University of Health Sciences & Pharmacy At St. Louis
Curated by ChEMBL
University of Health Sciences & Pharmacy At St. Louis
Curated by ChEMBL
Affinity DataEC50: 1.91E+4nMAssay Description:Agonist activity at human MOR receptor expressed in HTLA cells co-expressing TEV-fused-beta-arrestin2 assessed as induction of beta-arrestin2 recruit...More data for this Ligand-Target Pair
TargetMu-type opioid receptor(Human)
University of Health Sciences & Pharmacy At St. Louis
Curated by ChEMBL
University of Health Sciences & Pharmacy At St. Louis
Curated by ChEMBL
Affinity DataEC50: 1.05E+4nMAssay Description:Agonist activity at human MOR receptor expressed in HTLA cells co-expressing TEV-fused-beta-arrestin2 assessed as induction of beta-arrestin2 recruit...More data for this Ligand-Target Pair
TargetMu-type opioid receptor(Human)
University of Health Sciences & Pharmacy At St. Louis
Curated by ChEMBL
University of Health Sciences & Pharmacy At St. Louis
Curated by ChEMBL
Affinity DataEC50: 8.13E+3nMAssay Description:Agonist activity at human MOR receptor expressed in HTLA cells co-expressing TEV-fused-beta-arrestin2 assessed as induction of beta-arrestin2 recruit...More data for this Ligand-Target Pair
TargetMu-type opioid receptor(Human)
University of Health Sciences & Pharmacy At St. Louis
Curated by ChEMBL
University of Health Sciences & Pharmacy At St. Louis
Curated by ChEMBL
Affinity DataEC50: 1.10E+4nMAssay Description:Agonist activity at human MOR receptor expressed in HTLA cells co-expressing TEV-fused-beta-arrestin2 assessed as induction of beta-arrestin2 recruit...More data for this Ligand-Target Pair
TargetMu-type opioid receptor(Human)
University of Health Sciences & Pharmacy At St. Louis
Curated by ChEMBL
University of Health Sciences & Pharmacy At St. Louis
Curated by ChEMBL
Affinity DataEC50: 182nMAssay Description:Agonist activity at human MOR receptor expressed in HTLA cells co-expressing TEV-fused-beta-arrestin2 assessed as induction of beta-arrestin2 recruit...More data for this Ligand-Target Pair
TargetMu-type opioid receptor(Human)
University of Health Sciences & Pharmacy At St. Louis
Curated by ChEMBL
University of Health Sciences & Pharmacy At St. Louis
Curated by ChEMBL
Affinity DataEC50: 83nMAssay Description:Agonist activity at human MOR expressed in HEK293T cells assessed as inhibition of forskolin-stimulated cAMP accumulation incubated for 30 mins by Gl...More data for this Ligand-Target Pair
TargetMu-type opioid receptor(Human)
University of Health Sciences & Pharmacy At St. Louis
Curated by ChEMBL
University of Health Sciences & Pharmacy At St. Louis
Curated by ChEMBL
Affinity DataEC50: 36nMAssay Description:Agonist activity at human MOR expressed in HEK293T cells assessed as inhibition of forskolin-stimulated cAMP accumulation incubated for 30 mins by Gl...More data for this Ligand-Target Pair
TargetMu-type opioid receptor(Human)
University of Health Sciences & Pharmacy At St. Louis
Curated by ChEMBL
University of Health Sciences & Pharmacy At St. Louis
Curated by ChEMBL
Affinity DataEC50: 7.30nMAssay Description:Agonist activity at human MOR expressed in HEK293T cells assessed as inhibition of forskolin-stimulated cAMP accumulation incubated for 30 mins by Gl...More data for this Ligand-Target Pair
TargetMu-type opioid receptor(Human)
University of Health Sciences & Pharmacy At St. Louis
Curated by ChEMBL
University of Health Sciences & Pharmacy At St. Louis
Curated by ChEMBL
Affinity DataEC50: 94nMAssay Description:Agonist activity at human MOR expressed in HEK293T cells assessed as inhibition of forskolin-stimulated cAMP accumulation incubated for 30 mins by Gl...More data for this Ligand-Target Pair
TargetMu-type opioid receptor(Human)
University of Health Sciences & Pharmacy At St. Louis
Curated by ChEMBL
University of Health Sciences & Pharmacy At St. Louis
Curated by ChEMBL
Affinity DataEC50: 83nMAssay Description:Agonist activity at human MOR expressed in HEK293T cells assessed as inhibition of forskolin-stimulated cAMP accumulation incubated for 30 mins by Gl...More data for this Ligand-Target Pair
TargetMu-type opioid receptor(Human)
University of Health Sciences & Pharmacy At St. Louis
Curated by ChEMBL
University of Health Sciences & Pharmacy At St. Louis
Curated by ChEMBL
Affinity DataEC50: 83nMAssay Description:Agonist activity at human MOR expressed in HEK293T cells assessed as inhibition of forskolin-stimulated cAMP accumulation incubated for 30 mins by Gl...More data for this Ligand-Target Pair
TargetMu-type opioid receptor(Human)
University of Health Sciences & Pharmacy At St. Louis
Curated by ChEMBL
University of Health Sciences & Pharmacy At St. Louis
Curated by ChEMBL
Affinity DataEC50: 3.76E+3nMAssay Description:Agonist activity at human MOR expressed in HEK293T cells assessed as inhibition of forskolin-stimulated cAMP accumulation incubated for 30 mins by Gl...More data for this Ligand-Target Pair
TargetMu-type opioid receptor(Human)
University of Health Sciences & Pharmacy At St. Louis
Curated by ChEMBL
University of Health Sciences & Pharmacy At St. Louis
Curated by ChEMBL
Affinity DataEC50: 86nMAssay Description:Agonist activity at human MOR expressed in HEK293T cells assessed as inhibition of forskolin-stimulated cAMP accumulation incubated for 30 mins by Gl...More data for this Ligand-Target Pair
TargetMu-type opioid receptor(Human)
University of Health Sciences & Pharmacy At St. Louis
Curated by ChEMBL
University of Health Sciences & Pharmacy At St. Louis
Curated by ChEMBL
Affinity DataEC50: 370nMAssay Description:Agonist activity at human MOR expressed in HEK293T cells assessed as inhibition of forskolin-stimulated cAMP accumulation incubated for 30 mins by Gl...More data for this Ligand-Target Pair
TargetMu-type opioid receptor(Human)
University of Health Sciences & Pharmacy At St. Louis
Curated by ChEMBL
University of Health Sciences & Pharmacy At St. Louis
Curated by ChEMBL
Affinity DataEC50: 104nMAssay Description:Agonist activity at human MOR expressed in HEK293T cells assessed as inhibition of forskolin-stimulated cAMP accumulation incubated for 30 mins by Gl...More data for this Ligand-Target Pair
TargetMu-type opioid receptor(Human)
University of Health Sciences & Pharmacy At St. Louis
Curated by ChEMBL
University of Health Sciences & Pharmacy At St. Louis
Curated by ChEMBL
Affinity DataEC50: 535nMAssay Description:Agonist activity at human MOR expressed in HEK293T cells assessed as inhibition of forskolin-stimulated cAMP accumulation incubated for 30 mins by Gl...More data for this Ligand-Target Pair
TargetMu-type opioid receptor(Human)
University of Health Sciences & Pharmacy At St. Louis
Curated by ChEMBL
University of Health Sciences & Pharmacy At St. Louis
Curated by ChEMBL
Affinity DataEC50: 30nMAssay Description:Agonist activity at human MOR expressed in HEK293T cells assessed as inhibition of forskolin-stimulated cAMP accumulation incubated for 30 mins by Gl...More data for this Ligand-Target Pair
TargetMu-type opioid receptor(Human)
University of Health Sciences & Pharmacy At St. Louis
Curated by ChEMBL
University of Health Sciences & Pharmacy At St. Louis
Curated by ChEMBL
Affinity DataEC50: 1.11E+3nMAssay Description:Agonist activity at human MOR expressed in HEK293T cells assessed as inhibition of forskolin-stimulated cAMP accumulation incubated for 30 mins by Gl...More data for this Ligand-Target Pair
TargetMu-type opioid receptor(Human)
University of Health Sciences & Pharmacy At St. Louis
Curated by ChEMBL
University of Health Sciences & Pharmacy At St. Louis
Curated by ChEMBL
Affinity DataEC50: 186nMAssay Description:Agonist activity at human MOR expressed in HEK293T cells assessed as inhibition of forskolin-stimulated cAMP accumulation incubated for 30 mins by Gl...More data for this Ligand-Target Pair
TargetMu-type opioid receptor(Human)
University of Health Sciences & Pharmacy At St. Louis
Curated by ChEMBL
University of Health Sciences & Pharmacy At St. Louis
Curated by ChEMBL
Affinity DataEC50: 71nMAssay Description:Agonist activity at human MOR expressed in HEK293T cells assessed as inhibition of forskolin-stimulated cAMP accumulation incubated for 30 mins by Gl...More data for this Ligand-Target Pair
TargetMu-type opioid receptor(Human)
University of Health Sciences & Pharmacy At St. Louis
Curated by ChEMBL
University of Health Sciences & Pharmacy At St. Louis
Curated by ChEMBL
Affinity DataEC50: 1.75E+4nMAssay Description:Agonist activity at human MOR expressed in HEK293T cells assessed as inhibition of forskolin-stimulated cAMP accumulation incubated for 30 mins by Gl...More data for this Ligand-Target Pair
TargetMu-type opioid receptor(Human)
University of Health Sciences & Pharmacy At St. Louis
Curated by ChEMBL
University of Health Sciences & Pharmacy At St. Louis
Curated by ChEMBL
Affinity DataEC50: 1.56E+3nMAssay Description:Agonist activity at human MOR expressed in HEK293T cells assessed as inhibition of forskolin-stimulated cAMP accumulation incubated for 30 mins by Gl...More data for this Ligand-Target Pair
TargetMu-type opioid receptor(Human)
University of Health Sciences & Pharmacy At St. Louis
Curated by ChEMBL
University of Health Sciences & Pharmacy At St. Louis
Curated by ChEMBL
Affinity DataEC50: 11nMAssay Description:Agonist activity at human MOR expressed in HEK293T cells assessed as inhibition of forskolin-stimulated cAMP accumulation incubated for 30 mins by Gl...More data for this Ligand-Target Pair
TargetMu-type opioid receptor(Human)
University of Health Sciences & Pharmacy At St. Louis
Curated by ChEMBL
University of Health Sciences & Pharmacy At St. Louis
Curated by ChEMBL
Affinity DataEC50: 241nMAssay Description:Agonist activity at human MOR expressed in HEK293T cells assessed as inhibition of forskolin-stimulated cAMP accumulation incubated for 30 mins by Gl...More data for this Ligand-Target Pair
TargetMu-type opioid receptor(Human)
University of Health Sciences & Pharmacy At St. Louis
Curated by ChEMBL
University of Health Sciences & Pharmacy At St. Louis
Curated by ChEMBL
Affinity DataEC50: 5.90nMAssay Description:Agonist activity at human MOR expressed in HEK293T cells assessed as inhibition of forskolin-stimulated cAMP accumulation incubated for 30 mins by Gl...More data for this Ligand-Target Pair
TargetMu-type opioid receptor(Human)
University of Health Sciences & Pharmacy At St. Louis
Curated by ChEMBL
University of Health Sciences & Pharmacy At St. Louis
Curated by ChEMBL
Affinity DataEC50: 0.490nMAssay Description:Agonist activity at human MOR expressed in HEK293T cells assessed as inhibition of forskolin-stimulated cAMP accumulation incubated for 30 mins by Gl...More data for this Ligand-Target Pair
TargetMu-type opioid receptor(Human)
University of Health Sciences & Pharmacy At St. Louis
Curated by ChEMBL
University of Health Sciences & Pharmacy At St. Louis
Curated by ChEMBL
Affinity DataEC50: 36nMAssay Description:Agonist activity at human MOR expressed in HEK293T cells assessed as inhibition of forskolin-stimulated cAMP accumulation incubated for 30 mins by Gl...More data for this Ligand-Target Pair
TargetMu-type opioid receptor(Human)
University of Health Sciences & Pharmacy At St. Louis
Curated by ChEMBL
University of Health Sciences & Pharmacy At St. Louis
Curated by ChEMBL
Affinity DataEC50: 5.20nMAssay Description:Agonist activity at human MOR expressed in HEK293T cells assessed as inhibition of forskolin-stimulated cAMP accumulation incubated for 30 mins by Gl...More data for this Ligand-Target Pair
TargetMu-type opioid receptor(Human)
University of Health Sciences & Pharmacy At St. Louis
Curated by ChEMBL
University of Health Sciences & Pharmacy At St. Louis
Curated by ChEMBL
Affinity DataEC50: 93nMAssay Description:Agonist activity at human MOR expressed in HEK293T cells assessed as inhibition of forskolin-stimulated cAMP accumulation incubated for 30 mins by Gl...More data for this Ligand-Target Pair
