Compile Data Set for Download or QSAR
Report error Found 6 Enz. Inhib. hit(s) with all data for entry = 50018513
TargetDipeptidyl peptidase 1(Human)
Fuyang Normal University

Curated by ChEMBL
LigandPNGBDBM50270029(2-Amino-N-[(S)-3-diazo-1-(4-iodo-benzyl)-2-oxo-pro...)
Affinity DataIC50: 1nMAssay Description:Inhibition of human Cathepsin C using Ala-4-[ 125 I]Phe-DMK as substrate preincubated for 30 mins followed by substrate addition measured after 6 to ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/20/2024
Entry Details
PubMed
TargetDipeptidyl peptidase 1(Human)
Fuyang Normal University

Curated by ChEMBL
LigandPNGBDBM50609008(CHEMBL5269225)
Affinity DataIC50: 1nMAssay Description:Inhibition of Cathepsin C (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/20/2024
Entry Details
PubMed
TargetDipeptidyl peptidase 1(Human)
Fuyang Normal University

Curated by ChEMBL
LigandPNGBDBM50270030(2-Amino-N-((S)-1-benzyl-3-diazo-2-oxo-propyl)-acet...)
Affinity DataIC50: 50nMAssay Description:Inhibition of human Cathepsin C using Ala-4-[ 125 I]Phe-DMK as substrate preincubated for 30 mins followed by substrate addition measured after 6 to ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/20/2024
Entry Details
PubMed
TargetDipeptidyl peptidase 1(Human)
Fuyang Normal University

Curated by ChEMBL
LigandPNGBDBM4779(cid_156414 | PD0183805 | CHEMBL545315 | CHEMBL3196...)
Affinity DataIC50: 120nMAssay Description:Inhibition of Cathepsin C (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/20/2024
Entry Details
PubMed
TargetDipeptidyl peptidase 1(Human)
Fuyang Normal University

Curated by ChEMBL
LigandPNGBDBM50609007(CHEMBL5290773)
Affinity DataIC50: 4.90E+3nMAssay Description:Inhibition of human Cathepsin C using Z-Arg-Arg-AM as substrate at 3 microM relative to controlMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/20/2024
Entry Details
PubMed
TargetDipeptidyl peptidase 1(Human)
Fuyang Normal University

Curated by ChEMBL
LigandPNGBDBM50147181(3-{[1-(2-Amino-acetylamino)-3-methyl-butyl]-hydrox...)
Affinity DataIC50: 3.90E+4nMAssay Description:Inhibition of human Cathepsin C using Gly- L -Phe-p-nitroanilide.HCl as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/20/2024
Entry Details
PubMed