Compile Data Set for Download or QSAR
Report error Found 39 Enz. Inhib. hit(s) with all data for entry = 50015430
TargetCannabinoid receptor 2(Human)
Shanghaitech University

Curated by ChEMBL
LigandPNGBDBM50586527(CHEMBL5091640)
Affinity DataIC50: 70nMAssay Description:Antagonist activity at human CB2 Receptor expressed in CHO cell membranes measured after 24 hrs by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Shanghaitech University

Curated by ChEMBL
LigandPNGBDBM50586530(CHEMBL5090191)
Affinity DataIC50: 360nMAssay Description:Antagonist activity at human CB2 Receptor expressed in CHO cell membranes measured after 24 hrs by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Shanghaitech University

Curated by ChEMBL
LigandPNGBDBM50586533(CHEMBL5090102)
Affinity DataIC50: 410nMAssay Description:Antagonist activity at human CB2 Receptor expressed in CHO cell membranes measured after 24 hrs by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Shanghaitech University

Curated by ChEMBL
LigandPNGBDBM50586532(CHEMBL5078575)
Affinity DataIC50: 620nMAssay Description:Antagonist activity at human CB2 Receptor expressed in CHO cell membranes measured after 24 hrs by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Shanghaitech University

Curated by ChEMBL
LigandPNGBDBM50586518(CHEMBL5075936)
Affinity DataIC50: 1.10E+3nMAssay Description:Antagonist activity at human CB2 Receptor expressed in CHO cell membranes measured after 24 hrs by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Shanghaitech University

Curated by ChEMBL
LigandPNGBDBM50586527(CHEMBL5091640)
Affinity DataIC50: 1.10E+3nMAssay Description:Antagonist activity at human CB1 Receptor expressed in CHO cell membranes measured after 24 hrs by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Shanghaitech University

Curated by ChEMBL
LigandPNGBDBM50586517(CHEMBL5093760)
Affinity DataIC50: 1.30E+3nMAssay Description:Antagonist activity at human CB2 Receptor expressed in CHO cell membranes measured after 24 hrs by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Shanghaitech University

Curated by ChEMBL
LigandPNGBDBM50586525(CHEMBL5094165)
Affinity DataIC50: 1.50E+3nMAssay Description:Antagonist activity at human CB2 Receptor expressed in CHO cell membranes measured after 24 hrs by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Shanghaitech University

Curated by ChEMBL
LigandPNGBDBM50586515(CHEMBL5092588)
Affinity DataIC50: 1.60E+3nMAssay Description:Antagonist activity at human CB2 Receptor expressed in CHO cell membranes measured after 24 hrs by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Shanghaitech University

Curated by ChEMBL
LigandPNGBDBM50586520(CHEMBL5085907)
Affinity DataIC50: 1.60E+3nMAssay Description:Antagonist activity at human CB1 Receptor expressed in CHO cell membranes measured after 24 hrs by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Shanghaitech University

Curated by ChEMBL
LigandPNGBDBM50586530(CHEMBL5090191)
Affinity DataIC50: 1.70E+3nMAssay Description:Antagonist activity at human CB1 Receptor expressed in CHO cell membranes measured after 24 hrs by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Shanghaitech University

Curated by ChEMBL
LigandPNGBDBM50586521(CHEMBL5083983)
Affinity DataIC50: 2.10E+3nMAssay Description:Antagonist activity at human CB2 Receptor expressed in CHO cell membranes measured after 24 hrs by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Shanghaitech University

Curated by ChEMBL
LigandPNGBDBM50586533(CHEMBL5090102)
Affinity DataIC50: 2.40E+3nMAssay Description:Antagonist activity at human CB1 Receptor expressed in CHO cell membranes measured after 24 hrs by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Shanghaitech University

Curated by ChEMBL
LigandPNGBDBM50586520(CHEMBL5085907)
Affinity DataIC50: 3.20E+3nMAssay Description:Antagonist activity at human CB2 Receptor expressed in CHO cell membranes measured after 24 hrs by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Shanghaitech University

Curated by ChEMBL
LigandPNGBDBM50586515(CHEMBL5092588)
Affinity DataIC50: 3.30E+3nMAssay Description:Antagonist activity at human CB1 Receptor expressed in CHO cell membranes measured after 24 hrs by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Shanghaitech University

Curated by ChEMBL
LigandPNGBDBM50586516(CHEMBL5082618)
Affinity DataIC50: 3.30E+3nMAssay Description:Antagonist activity at human CB1 Receptor expressed in CHO cell membranes measured after 24 hrs by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Shanghaitech University

Curated by ChEMBL
LigandPNGBDBM50586523(CHEMBL5082613)
Affinity DataIC50: 3.40E+3nMAssay Description:Antagonist activity at human CB2 Receptor expressed in CHO cell membranes measured after 24 hrs by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Shanghaitech University

Curated by ChEMBL
LigandPNGBDBM50586519(CHEMBL5070839)
Affinity DataIC50: 3.50E+3nMAssay Description:Antagonist activity at human CB2 Receptor expressed in CHO cell membranes measured after 24 hrs by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Shanghaitech University

Curated by ChEMBL
LigandPNGBDBM50586524(CHEMBL5081238)
Affinity DataIC50: 3.70E+3nMAssay Description:Antagonist activity at human CB2 Receptor expressed in CHO cell membranes measured after 24 hrs by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Shanghaitech University

Curated by ChEMBL
LigandPNGBDBM50586521(CHEMBL5083983)
Affinity DataIC50: 3.80E+3nMAssay Description:Antagonist activity at human CB1 Receptor expressed in CHO cell membranes measured after 24 hrs by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Shanghaitech University

Curated by ChEMBL
LigandPNGBDBM50586518(CHEMBL5075936)
Affinity DataIC50: 3.80E+3nMAssay Description:Antagonist activity at human CB1 Receptor expressed in CHO cell membranes measured after 24 hrs by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Shanghaitech University

Curated by ChEMBL
LigandPNGBDBM50586517(CHEMBL5093760)
Affinity DataIC50: 3.90E+3nMAssay Description:Antagonist activity at human CB1 Receptor expressed in CHO cell membranes measured after 24 hrs by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Shanghaitech University

Curated by ChEMBL
LigandPNGBDBM50586529(CHEMBL5091980)
Affinity DataIC50: 4.10E+3nMAssay Description:Antagonist activity at human CB1 Receptor expressed in CHO cell membranes measured after 24 hrs by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Shanghaitech University

Curated by ChEMBL
LigandPNGBDBM50586524(CHEMBL5081238)
Affinity DataIC50: 4.80E+3nMAssay Description:Antagonist activity at human CB1 Receptor expressed in CHO cell membranes measured after 24 hrs by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Shanghaitech University

Curated by ChEMBL
LigandPNGBDBM50586516(CHEMBL5082618)
Affinity DataIC50: 5.20E+3nMAssay Description:Antagonist activity at human CB2 Receptor expressed in CHO cell membranes measured after 24 hrs by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Shanghaitech University

Curated by ChEMBL
LigandPNGBDBM50586519(CHEMBL5070839)
Affinity DataIC50: 5.40E+3nMAssay Description:Antagonist activity at human CB1 Receptor expressed in CHO cell membranes measured after 24 hrs by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Shanghaitech University

Curated by ChEMBL
LigandPNGBDBM50586531(CHEMBL5082876)
Affinity DataIC50: 5.50E+3nMAssay Description:Antagonist activity at human CB2 Receptor expressed in CHO cell membranes measured after 24 hrs by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Shanghaitech University

Curated by ChEMBL
LigandPNGBDBM50586528(CHEMBL5075782)
Affinity DataIC50: 5.80E+3nMAssay Description:Antagonist activity at human CB1 Receptor expressed in CHO cell membranes measured after 24 hrs by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Shanghaitech University

Curated by ChEMBL
LigandPNGBDBM50586522(CHEMBL5080263)
Affinity DataIC50: 5.90E+3nMAssay Description:Antagonist activity at human CB1 Receptor expressed in CHO cell membranes measured after 24 hrs by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Shanghaitech University

Curated by ChEMBL
LigandPNGBDBM50586525(CHEMBL5094165)
Affinity DataIC50: 6.20E+3nMAssay Description:Antagonist activity at human CB1 Receptor expressed in CHO cell membranes measured after 24 hrs by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Shanghaitech University

Curated by ChEMBL
LigandPNGBDBM50586522(CHEMBL5080263)
Affinity DataIC50: 6.50E+3nMAssay Description:Antagonist activity at human CB2 Receptor expressed in CHO cell membranes measured after 24 hrs by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Shanghaitech University

Curated by ChEMBL
LigandPNGBDBM50586529(CHEMBL5091980)
Affinity DataIC50: 6.90E+3nMAssay Description:Antagonist activity at human CB2 Receptor expressed in CHO cell membranes measured after 24 hrs by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Shanghaitech University

Curated by ChEMBL
LigandPNGBDBM50586528(CHEMBL5075782)
Affinity DataIC50: 7.00E+3nMAssay Description:Antagonist activity at human CB2 Receptor expressed in CHO cell membranes measured after 24 hrs by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Shanghaitech University

Curated by ChEMBL
LigandPNGBDBM50586537(CHEMBL5087154)
Affinity DataIC50: 7.20E+3nMAssay Description:Antagonist activity at human CB1 Receptor expressed in CHO cell membranes measured after 24 hrs by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Shanghaitech University

Curated by ChEMBL
LigandPNGBDBM50586536(CHEMBL5087401)
Affinity DataIC50: 7.90E+3nMAssay Description:Antagonist activity at human CB1 Receptor expressed in CHO cell membranes measured after 24 hrs by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Shanghaitech University

Curated by ChEMBL
LigandPNGBDBM50586535(CHEMBL5089064)
Affinity DataIC50: 8.30E+3nMAssay Description:Antagonist activity at human CB1 Receptor expressed in CHO cell membranes measured after 24 hrs by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Shanghaitech University

Curated by ChEMBL
LigandPNGBDBM50586526(CHEMBL5092678)
Affinity DataIC50: 9.00E+3nMAssay Description:Antagonist activity at human CB2 Receptor expressed in CHO cell membranes measured after 24 hrs by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Shanghaitech University

Curated by ChEMBL
LigandPNGBDBM50586523(CHEMBL5082613)
Affinity DataIC50: 9.00E+3nMAssay Description:Antagonist activity at human CB1 Receptor expressed in CHO cell membranes measured after 24 hrs by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Shanghaitech University

Curated by ChEMBL
LigandPNGBDBM50586534(CHEMBL5094751)
Affinity DataIC50: 9.40E+3nMAssay Description:Antagonist activity at human CB1 Receptor expressed in CHO cell membranes measured after 24 hrs by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed