Compile Data Set for Download or QSAR
Report error Found 49 Enz. Inhib. hit(s) with all data for entry = 50015021
TargetSodium channel protein type 8 subunit alpha(Mouse)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50582056(CHEMBL5091623)
Affinity DataEC50:  93nMAssay Description:Modulator activity at mouse Nav1.6 expressed in Xenopus laevis oocytes assessed as elicitation in sodium current measured after 1 to 4 days by two-el...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetSodium channel protein type 4 subunit alpha(Rat)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50582058(CHEMBL5093878)
Affinity DataEC50:  15nMAssay Description:Modulator activity at rat Nav1.4 expressed in Xenopus laevis oocytes assessed as elicitation in sodium current measured after 1 to 4 days by two-elec...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetSodium channel protein type 4 subunit alpha(Rat)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50582059(CHEMBL5082582)
Affinity DataEC50:  46nMAssay Description:Modulator activity at rat Nav1.4 expressed in Xenopus laevis oocytes assessed as elicitation in sodium current measured after 1 to 4 days by two-elec...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetSodium channel protein type 4 subunit alpha(Rat)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50582060(CHEMBL5084333)
Affinity DataEC50:  811nMAssay Description:Modulator activity at rat Nav1.4 expressed in Xenopus laevis oocytes assessed as elicitation in sodium current measured after 1 to 4 days by two-elec...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetSodium channel protein type 5 subunit alpha(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50582054(CHEMBL5091679)
Affinity DataEC50:  138nMAssay Description:Modulator activity at human Nav1.5 expressed in Xenopus laevis oocytes assessed as elicitation in sodium current measured after 1 to 4 days by two-el...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetSodium channel protein type 5 subunit alpha(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50582055(CHEMBL5083412)
Affinity DataEC50:  149nMAssay Description:Modulator activity at human Nav1.5 expressed in Xenopus laevis oocytes assessed as elicitation in sodium current measured after 1 to 4 days by two-el...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetSodium channel protein type 5 subunit alpha(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50582056(CHEMBL5091623)
Affinity DataEC50:  108nMAssay Description:Modulator activity at human Nav1.5 expressed in Xenopus laevis oocytes assessed as elicitation in sodium current measured after 1 to 4 days by two-el...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetSodium channel protein type 5 subunit alpha(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50582057(CHEMBL5077579)
Affinity DataEC50:  28nMAssay Description:Modulator activity at human Nav1.5 expressed in Xenopus laevis oocytes assessed as elicitation in sodium current measured after 1 to 4 days by two-el...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetSodium channel protein type 5 subunit alpha(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50582058(CHEMBL5093878)
Affinity DataEC50:  133nMAssay Description:Modulator activity at human Nav1.5 expressed in Xenopus laevis oocytes assessed as elicitation in sodium current measured after 1 to 4 days by two-el...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetSodium channel protein type 5 subunit alpha(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50582059(CHEMBL5082582)
Affinity DataEC50:  215nMAssay Description:Modulator activity at human Nav1.5 expressed in Xenopus laevis oocytes assessed as elicitation in sodium current measured after 1 to 4 days by two-el...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetSodium channel protein type 5 subunit alpha(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50582060(CHEMBL5084333)
Affinity DataEC50:  156nMAssay Description:Modulator activity at human Nav1.5 expressed in Xenopus laevis oocytes assessed as elicitation in sodium current measured after 1 to 4 days by two-el...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetSodium channel protein type 8 subunit alpha(Mouse)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50582054(CHEMBL5091679)
Affinity DataEC50:  240nMAssay Description:Modulator activity at mouse Nav1.6 expressed in Xenopus laevis oocytes assessed as elicitation in sodium current measured after 1 to 4 days by two-el...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetSodium channel protein type 8 subunit alpha(Mouse)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50582055(CHEMBL5083412)
Affinity DataEC50:  1.36E+3nMAssay Description:Modulator activity at mouse Nav1.6 expressed in Xenopus laevis oocytes assessed as elicitation in sodium current measured after 1 to 4 days by two-el...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetSodium channel protein type 4 subunit alpha(Rat)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50582057(CHEMBL5077579)
Affinity DataEC50:  15nMAssay Description:Modulator activity at rat Nav1.4 expressed in Xenopus laevis oocytes assessed as elicitation in sodium current measured after 1 to 4 days by two-elec...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetSodium channel protein type 8 subunit alpha(Mouse)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50582057(CHEMBL5077579)
Affinity DataEC50:  124nMAssay Description:Modulator activity at mouse Nav1.6 expressed in Xenopus laevis oocytes assessed as elicitation in sodium current measured after 1 to 4 days by two-el...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetSodium channel protein type 8 subunit alpha(Mouse)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50582058(CHEMBL5093878)
Affinity DataEC50:  67nMAssay Description:Modulator activity at mouse Nav1.6 expressed in Xenopus laevis oocytes assessed as elicitation in sodium current measured after 1 to 4 days by two-el...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetSodium channel protein type 8 subunit alpha(Mouse)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50582059(CHEMBL5082582)
Affinity DataEC50:  36nMAssay Description:Modulator activity at mouse Nav1.6 expressed in Xenopus laevis oocytes assessed as elicitation in sodium current measured after 1 to 4 days by two-el...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetSodium channel protein type 8 subunit alpha(Mouse)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50582060(CHEMBL5084333)
Affinity DataEC50:  148nMAssay Description:Modulator activity at mouse Nav1.6 expressed in Xenopus laevis oocytes assessed as elicitation in sodium current measured after 1 to 4 days by two-el...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetSodium channel protein type 9 subunit alpha(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50582054(CHEMBL5091679)
Affinity DataEC50:  77nMAssay Description:Modulator activity at human Nav1.7 expressed in Xenopus laevis oocytes assessed as elicitation in sodium current measured after 1 to 4 days by two-el...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetSodium channel protein type 9 subunit alpha(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50582055(CHEMBL5083412)
Affinity DataEC50:  1.30E+3nMAssay Description:Modulator activity at human Nav1.7 expressed in Xenopus laevis oocytes assessed as elicitation in sodium current measured after 1 to 4 days by two-el...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetSodium channel protein type 9 subunit alpha(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50582056(CHEMBL5091623)
Affinity DataEC50:  102nMAssay Description:Modulator activity at human Nav1.7 expressed in Xenopus laevis oocytes assessed as elicitation in sodium current measured after 1 to 4 days by two-el...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetSodium channel protein type 9 subunit alpha(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50582057(CHEMBL5077579)
Affinity DataEC50:  81nMAssay Description:Modulator activity at human Nav1.7 expressed in Xenopus laevis oocytes assessed as elicitation in sodium current measured after 1 to 4 days by two-el...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetSodium channel protein type 9 subunit alpha(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50582058(CHEMBL5093878)
Affinity DataEC50:  73nMAssay Description:Modulator activity at human Nav1.7 expressed in Xenopus laevis oocytes assessed as elicitation in sodium current measured after 1 to 4 days by two-el...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetSodium channel protein type 9 subunit alpha(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50582059(CHEMBL5082582)
Affinity DataEC50:  97nMAssay Description:Modulator activity at human Nav1.7 expressed in Xenopus laevis oocytes assessed as elicitation in sodium current measured after 1 to 4 days by two-el...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetSodium channel protein type 9 subunit alpha(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50582060(CHEMBL5084333)
Affinity DataEC50:  129nMAssay Description:Modulator activity at human Nav1.7 expressed in Xenopus laevis oocytes assessed as elicitation in sodium current measured after 1 to 4 days by two-el...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetSodium channel protein type 2 subunit alpha(Rat)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50582059(CHEMBL5082582)
Affinity DataEC50:  24nMAssay Description:Modulator activity at rat Nav1.2 expressed in Xenopus laevis oocytes assessed as elicitation in sodium current measured after 1 to 4 days by two-elec...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetSodium channel protein type 1 subunit alpha(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50582055(CHEMBL5083412)
Affinity DataEC50:  126nMAssay Description:Modulator activity at human Nav1.1 expressed in Xenopus laevis oocytes assessed as elicitation in sodium current measured after 1 to 4 days by two-el...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetSodium channel protein type 1 subunit alpha(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50582056(CHEMBL5091623)
Affinity DataEC50:  126nMAssay Description:Modulator activity at human Nav1.1 expressed in Xenopus laevis oocytes assessed as elicitation in sodium current measured after 1 to 4 days by two-el...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetSodium channel protein type 1 subunit alpha(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50582057(CHEMBL5077579)
Affinity DataEC50:  92nMAssay Description:Modulator activity at human Nav1.1 expressed in Xenopus laevis oocytes assessed as elicitation in sodium current measured after 1 to 4 days by two-el...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetSodium channel protein type 1 subunit alpha(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50582058(CHEMBL5093878)
Affinity DataEC50:  102nMAssay Description:Modulator activity at human Nav1.1 expressed in Xenopus laevis oocytes assessed as elicitation in sodium current measured after 1 to 4 days by two-el...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetSodium channel protein type 1 subunit alpha(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50582059(CHEMBL5082582)
Affinity DataEC50:  7.90nMAssay Description:Modulator activity at human Nav1.1 expressed in Xenopus laevis oocytes assessed as elicitation in sodium current measured after 1 to 4 days by two-el...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetSodium channel protein type 1 subunit alpha(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50582060(CHEMBL5084333)
Affinity DataEC50:  172nMAssay Description:Modulator activity at human Nav1.1 expressed in Xenopus laevis oocytes assessed as elicitation in sodium current measured after 1 to 4 days by two-el...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetSodium channel protein type 2 subunit alpha(Rat)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50582054(CHEMBL5091679)
Affinity DataEC50:  360nMAssay Description:Modulator activity at rat Nav1.2 expressed in Xenopus laevis oocytes assessed as elicitation in sodium current measured after 1 to 4 days by two-elec...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetSodium channel protein type 2 subunit alpha(Rat)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50582055(CHEMBL5083412)
Affinity DataEC50:  98nMAssay Description:Modulator activity at rat Nav1.2 expressed in Xenopus laevis oocytes assessed as elicitation in sodium current measured after 1 to 4 days by two-elec...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetSodium channel protein type 2 subunit alpha(Rat)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50582056(CHEMBL5091623)
Affinity DataEC50:  138nMAssay Description:Modulator activity at rat Nav1.2 expressed in Xenopus laevis oocytes assessed as elicitation in sodium current measured after 1 to 4 days by two-elec...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetSodium channel protein type 2 subunit alpha(Rat)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50582057(CHEMBL5077579)
Affinity DataEC50:  134nMAssay Description:Modulator activity at rat Nav1.2 expressed in Xenopus laevis oocytes assessed as elicitation in sodium current measured after 1 to 4 days by two-elec...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetSodium channel protein type 2 subunit alpha(Rat)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50582058(CHEMBL5093878)
Affinity DataEC50:  156nMAssay Description:Modulator activity at rat Nav1.2 expressed in Xenopus laevis oocytes assessed as elicitation in sodium current measured after 1 to 4 days by two-elec...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetSodium channel protein type 1 subunit alpha(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50582054(CHEMBL5091679)
Affinity DataEC50:  124nMAssay Description:Modulator activity at human Nav1.1 expressed in Xenopus laevis oocytes assessed as elicitation in sodium current measured after 1 to 4 days by two-el...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetSodium channel protein type 2 subunit alpha(Rat)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50582060(CHEMBL5084333)
Affinity DataEC50:  50nMAssay Description:Modulator activity at rat Nav1.2 expressed in Xenopus laevis oocytes assessed as elicitation in sodium current measured after 1 to 4 days by two-elec...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetSodium channel protein type 3 subunit alpha(Rat)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50582054(CHEMBL5091679)
Affinity DataEC50:  135nMAssay Description:Modulator activity at rat Nav1.3 expressed in Xenopus laevis oocytes assessed as elicitation in sodium current measured after 1 to 4 days by two-elec...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetSodium channel protein type 3 subunit alpha(Rat)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50582055(CHEMBL5083412)
Affinity DataEC50:  128nMAssay Description:Modulator activity at rat Nav1.3 expressed in Xenopus laevis oocytes assessed as elicitation in sodium current measured after 1 to 4 days by two-elec...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetSodium channel protein type 3 subunit alpha(Rat)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50582056(CHEMBL5091623)
Affinity DataEC50:  139nMAssay Description:Modulator activity at rat Nav1.3 expressed in Xenopus laevis oocytes assessed as elicitation in sodium current measured after 1 to 4 days by two-elec...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetSodium channel protein type 3 subunit alpha(Rat)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50582057(CHEMBL5077579)
Affinity DataEC50:  13nMAssay Description:Modulator activity at rat Nav1.3 expressed in Xenopus laevis oocytes assessed as elicitation in sodium current measured after 1 to 4 days by two-elec...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetSodium channel protein type 3 subunit alpha(Rat)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50582058(CHEMBL5093878)
Affinity DataEC50:  9.40nMAssay Description:Modulator activity at rat Nav1.3 expressed in Xenopus laevis oocytes assessed as elicitation in sodium current measured after 1 to 4 days by two-elec...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetSodium channel protein type 3 subunit alpha(Rat)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50582059(CHEMBL5082582)
Affinity DataEC50:  106nMAssay Description:Modulator activity at rat Nav1.3 expressed in Xenopus laevis oocytes assessed as elicitation in sodium current measured after 1 to 4 days by two-elec...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetSodium channel protein type 3 subunit alpha(Rat)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50582060(CHEMBL5084333)
Affinity DataEC50:  170nMAssay Description:Modulator activity at rat Nav1.3 expressed in Xenopus laevis oocytes assessed as elicitation in sodium current measured after 1 to 4 days by two-elec...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetSodium channel protein type 4 subunit alpha(Rat)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50582054(CHEMBL5091679)
Affinity DataEC50:  146nMAssay Description:Modulator activity at rat Nav1.4 expressed in Xenopus laevis oocytes assessed as elicitation in sodium current measured after 1 to 4 days by two-elec...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetSodium channel protein type 4 subunit alpha(Rat)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50582055(CHEMBL5083412)
Affinity DataEC50:  1.15E+3nMAssay Description:Modulator activity at rat Nav1.4 expressed in Xenopus laevis oocytes assessed as elicitation in sodium current measured after 1 to 4 days by two-elec...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetSodium channel protein type 4 subunit alpha(Rat)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50582056(CHEMBL5091623)
Affinity DataEC50:  150nMAssay Description:Modulator activity at rat Nav1.4 expressed in Xenopus laevis oocytes assessed as elicitation in sodium current measured after 1 to 4 days by two-elec...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed