Compile Data Set for Download or QSAR
Report error Found 4 Enz. Inhib. hit(s) with all data for entry = 50014818
TargetEstrogen receptor(Human)
University of North Carolina Wilmington

Curated by ChEMBL
LigandPNGBDBM17292([2,4,6,7-3H]-17beta-estradiol | [3H]-estradiol | 1...)
Affinity DataIC50: 0.580nMAssay Description:Binding affinity of ERalpha LBD (unknown origin) incubated for 2 hrs by LanthaScreen TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/4/2023
Entry Details Article
PubMed
TargetEstrogen receptor(Human)
University of North Carolina Wilmington

Curated by ChEMBL
LigandPNGBDBM50580157(CHEMBL5071091)
Affinity DataIC50: 0.990nMAssay Description:Binding affinity of ERalpha LBD (unknown origin) incubated for 2 hrs by LanthaScreen TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/4/2023
Entry Details Article
PubMed
TargetEstrogen receptor(Human)
University of North Carolina Wilmington

Curated by ChEMBL
LigandPNGBDBM50351197(CHEMBL1818254)
Affinity DataIC50: 1.10nMAssay Description:Binding affinity of ERalpha LBD (unknown origin) incubated for 2 hrs by LanthaScreen TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/4/2023
Entry Details Article
PubMed
TargetEstrogen receptor(Human)
University of North Carolina Wilmington

Curated by ChEMBL
LigandPNGBDBM50580158(CHEMBL5072592)
Affinity DataIC50: 1.5nMAssay Description:Binding affinity of ERalpha LBD (unknown origin) incubated for 2 hrs by LanthaScreen TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/4/2023
Entry Details Article
PubMed