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Report error Found 28 Enz. Inhib. hit(s) with all data for entry = 50014152
TargetCannabinoid receptor 2(Human)
Therachem Research Medilab

Curated by ChEMBL
LigandPNGBDBM50573083(CHEMBL4845707)
Affinity DataEC50:  108nMAssay Description:Agonist activity at human CB2 receptor expressed in CHO-K1 cells assessed as increase in cAMP level incubated for 20 mins measured after 60 mins addi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2022
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Therachem Research Medilab

Curated by ChEMBL
LigandPNGBDBM50573096(CHEMBL4865119)
Affinity DataEC50: >5nMAssay Description:Agonist activity at human CB2 receptor expressed in CHO-K1 cells assessed as increase in cAMP level incubated for 20 mins measured after 60 mins addi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2022
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Therachem Research Medilab

Curated by ChEMBL
LigandPNGBDBM50573095(CHEMBL4857198)
Affinity DataEC50: >5nMAssay Description:Agonist activity at human CB2 receptor expressed in CHO-K1 cells assessed as increase in cAMP level incubated for 20 mins measured after 60 mins addi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2022
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Therachem Research Medilab

Curated by ChEMBL
LigandPNGBDBM50573094(CHEMBL4872695)
Affinity DataEC50:  0.700nMAssay Description:Agonist activity at human CB2 receptor expressed in CHO-K1 cells assessed as increase in cAMP level incubated for 20 mins measured after 60 mins addi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2022
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Therachem Research Medilab

Curated by ChEMBL
LigandPNGBDBM50573093(CHEMBL4875720)
Affinity DataEC50: >5nMAssay Description:Agonist activity at human CB2 receptor expressed in CHO-K1 cells assessed as increase in cAMP level incubated for 20 mins measured after 60 mins addi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2022
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Therachem Research Medilab

Curated by ChEMBL
LigandPNGBDBM50573092(CHEMBL4851858)
Affinity DataEC50: >5nMAssay Description:Agonist activity at human CB2 receptor expressed in CHO-K1 cells assessed as increase in cAMP level incubated for 20 mins measured after 60 mins addi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2022
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Therachem Research Medilab

Curated by ChEMBL
LigandPNGBDBM50573091(CHEMBL4865162)
Affinity DataEC50:  130nMAssay Description:Agonist activity at human CB2 receptor expressed in CHO-K1 cells assessed as increase in cAMP level incubated for 20 mins measured after 60 mins addi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2022
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Therachem Research Medilab

Curated by ChEMBL
LigandPNGBDBM50573090(CHEMBL4847866)
Affinity DataEC50:  49nMAssay Description:Agonist activity at human CB2 receptor expressed in CHO-K1 cells assessed as increase in cAMP level incubated for 20 mins measured after 60 mins addi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2022
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Therachem Research Medilab

Curated by ChEMBL
LigandPNGBDBM50573089(CHEMBL4846759)
Affinity DataEC50:  1.78E+3nMAssay Description:Agonist activity at human CB2 receptor expressed in CHO-K1 cells assessed as increase in cAMP level incubated for 20 mins measured after 60 mins addi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2022
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Therachem Research Medilab

Curated by ChEMBL
LigandPNGBDBM50573088(CHEMBL4873473)
Affinity DataEC50:  17nMAssay Description:Agonist activity at human CB2 receptor expressed in CHO-K1 cells assessed as increase in cAMP level incubated for 20 mins measured after 60 mins addi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2022
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Therachem Research Medilab

Curated by ChEMBL
LigandPNGBDBM50573087(CHEMBL4862304)
Affinity DataEC50:  571nMAssay Description:Agonist activity at human CB2 receptor expressed in CHO-K1 cells assessed as increase in cAMP level incubated for 20 mins measured after 60 mins addi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2022
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Therachem Research Medilab

Curated by ChEMBL
LigandPNGBDBM50573086(CHEMBL4871491)
Affinity DataEC50:  422nMAssay Description:Agonist activity at human CB2 receptor expressed in CHO-K1 cells assessed as increase in cAMP level incubated for 20 mins measured after 60 mins addi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2022
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Therachem Research Medilab

Curated by ChEMBL
LigandPNGBDBM50573085(CHEMBL4871528)
Affinity DataEC50: >5nMAssay Description:Agonist activity at human CB2 receptor expressed in CHO-K1 cells assessed as increase in cAMP level incubated for 20 mins measured after 60 mins addi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2022
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Therachem Research Medilab

Curated by ChEMBL
LigandPNGBDBM50573084(CHEMBL4870368)
Affinity DataEC50: >5nMAssay Description:Agonist activity at human CB2 receptor expressed in CHO-K1 cells assessed as increase in cAMP level incubated for 20 mins measured after 60 mins addi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2022
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Therachem Research Medilab

Curated by ChEMBL
LigandPNGBDBM50573083(CHEMBL4845707)
Affinity DataEC50:  1.20nMAssay Description:Agonist activity at human CB1 receptor expressed in CHO-K1 cells assessed as increase in cAMP level incubated for 20 mins measured after 60 mins addi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2022
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Therachem Research Medilab

Curated by ChEMBL
LigandPNGBDBM50573096(CHEMBL4865119)
Affinity DataEC50:  2.67E+3nMAssay Description:Agonist activity at human CB1 receptor expressed in CHO-K1 cells assessed as increase in cAMP level incubated for 20 mins measured after 60 mins addi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2022
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Therachem Research Medilab

Curated by ChEMBL
LigandPNGBDBM50573095(CHEMBL4857198)
Affinity DataEC50:  1.65E+3nMAssay Description:Agonist activity at human CB1 receptor expressed in CHO-K1 cells assessed as increase in cAMP level incubated for 20 mins measured after 60 mins addi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2022
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Therachem Research Medilab

Curated by ChEMBL
LigandPNGBDBM50573094(CHEMBL4872695)
Affinity DataEC50:  0.0800nMAssay Description:Agonist activity at human CB1 receptor expressed in CHO-K1 cells assessed as increase in cAMP level incubated for 20 mins measured after 60 mins addi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2022
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Therachem Research Medilab

Curated by ChEMBL
LigandPNGBDBM50573093(CHEMBL4875720)
Affinity DataEC50:  0.0400nMAssay Description:Agonist activity at human CB1 receptor expressed in CHO-K1 cells assessed as increase in cAMP level incubated for 20 mins measured after 60 mins addi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2022
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Therachem Research Medilab

Curated by ChEMBL
LigandPNGBDBM50573092(CHEMBL4851858)
Affinity DataEC50:  7.97E+3nMAssay Description:Agonist activity at human CB1 receptor expressed in CHO-K1 cells assessed as increase in cAMP level incubated for 20 mins measured after 60 mins addi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2022
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Therachem Research Medilab

Curated by ChEMBL
LigandPNGBDBM50573091(CHEMBL4865162)
Affinity DataEC50:  0.0600nMAssay Description:Agonist activity at human CB1 receptor expressed in CHO-K1 cells assessed as increase in cAMP level incubated for 20 mins measured after 60 mins addi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2022
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Therachem Research Medilab

Curated by ChEMBL
LigandPNGBDBM50573090(CHEMBL4847866)
Affinity DataEC50:  0.0200nMAssay Description:Agonist activity at human CB1 receptor expressed in CHO-K1 cells assessed as increase in cAMP level incubated for 20 mins measured after 60 mins addi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2022
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Therachem Research Medilab

Curated by ChEMBL
LigandPNGBDBM50573089(CHEMBL4846759)
Affinity DataEC50:  0.0500nMAssay Description:Agonist activity at human CB1 receptor expressed in CHO-K1 cells assessed as increase in cAMP level incubated for 20 mins measured after 60 mins addi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2022
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Therachem Research Medilab

Curated by ChEMBL
LigandPNGBDBM50573088(CHEMBL4873473)
Affinity DataEC50:  0.0200nMAssay Description:Agonist activity at human CB1 receptor expressed in CHO-K1 cells assessed as increase in cAMP level incubated for 20 mins measured after 60 mins addi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2022
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Therachem Research Medilab

Curated by ChEMBL
LigandPNGBDBM50573087(CHEMBL4862304)
Affinity DataEC50:  0.0400nMAssay Description:Agonist activity at human CB1 receptor expressed in CHO-K1 cells assessed as increase in cAMP level incubated for 20 mins measured after 60 mins addi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2022
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Therachem Research Medilab

Curated by ChEMBL
LigandPNGBDBM50573086(CHEMBL4871491)
Affinity DataEC50:  0.0900nMAssay Description:Agonist activity at human CB1 receptor expressed in CHO-K1 cells assessed as increase in cAMP level incubated for 20 mins measured after 60 mins addi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2022
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Therachem Research Medilab

Curated by ChEMBL
LigandPNGBDBM50573085(CHEMBL4871528)
Affinity DataEC50:  0.560nMAssay Description:Agonist activity at human CB1 receptor expressed in CHO-K1 cells assessed as increase in cAMP level incubated for 20 mins measured after 60 mins addi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2022
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Therachem Research Medilab

Curated by ChEMBL
LigandPNGBDBM50573084(CHEMBL4870368)
Affinity DataEC50:  2.98E+3nMAssay Description:Agonist activity at human CB1 receptor expressed in CHO-K1 cells assessed as increase in cAMP level incubated for 20 mins measured after 60 mins addi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2022
Entry Details Article
PubMed