Compile Data Set for Download or QSAR
Report error Found 229 Enz. Inhib. hit(s) with all data for entry = 50018700
TargetToll-like receptor 7(Human)
Panjab University

Curated by ChEMBL
LigandPNGBDBM50611739(CHEMBL5265854)
Affinity DataEC50:  1nMAssay Description:Agonist activity at human TLR7 in HEK-Blue hTLR7 cells incubated for 18 hrs by quanti-blue reagent based analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetToll-like receptor 7(Human)
Panjab University

Curated by ChEMBL
LigandPNGBDBM393035(US9962388, Compound Example 41 | 4-amino-2-butoxy-...)
Affinity DataEC50:  1nMAssay Description:Agonist activity at TLR7 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetToll-like receptor 7(Human)
Panjab University

Curated by ChEMBL
LigandPNGBDBM50320082(1-(4-Amino-2-butyl-1H-imidazo-[4,5-c]quinolin-1-yl...)
Affinity DataEC50:  2.5nMAssay Description:Agonist activity at human TLR7 expressed in HEK293 cells assessed as activation of NFkappaB incubated for 18 to 24 hrs by SEAP reporter gene based as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetToll-like receptor 7(Human)
Panjab University

Curated by ChEMBL
LigandPNGBDBM50330063(1-(4-(Aminomethyl)benzyl)-2-butyl-1H-imidazo[4,5-c...)
Affinity DataEC50:  4nMAssay Description:Agonist activity at human TLR7 expressed in HEK293 cells assessed as activation of NFkappaB incubated for 18 to 24 hrs by SEAP reporter gene based as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetToll-like receptor 7(Human)
Panjab University

Curated by ChEMBL
LigandPNGBDBM50611654(CHEMBL5273504)
Affinity DataEC50:  11nMAssay Description:Agonist activity at human TLR7 transfected in HEK293 cells assessed as induction of SEAP production incubated overnight by SEAP reporter gene based a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetToll-like receptor 7(Human)
Panjab University

Curated by ChEMBL
LigandPNGBDBM50611663(CHEMBL5290342)
Affinity DataEC50:  17nMAssay Description:Agonist activity at human TLR7 transfected in HEK293 cells assessed as induction of SEAP production incubated overnight by SEAP reporter gene based a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetToll-like receptor 8(Human)
Panjab University

Curated by ChEMBL
LigandPNGBDBM50320082(1-(4-Amino-2-butyl-1H-imidazo-[4,5-c]quinolin-1-yl...)
Affinity DataEC50:  19nMAssay Description:Agonist activity at human TLR8 expressed in HEK293 cells assessed as activation of NFkappaB incubated for 18 to 24 hrs by SEAP reporter gene based as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetToll-like receptor 7(Human)
Panjab University

Curated by ChEMBL
LigandPNGBDBM50611660(CHEMBL5273693)
Affinity DataEC50:  20nMAssay Description:Agonist activity at human TLR7 transfected in HEK293 cells assessed as induction of SEAP production incubated overnight by SEAP reporter gene based a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetToll-like receptor 7(Human)
Panjab University

Curated by ChEMBL
LigandPNGBDBM50611664(CHEMBL5280480)
Affinity DataEC50:  21nMAssay Description:Agonist activity at human TLR7 transfected in HEK293 cells assessed as induction of SEAP production incubated overnight by SEAP reporter gene based a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetToll-like receptor 7(Human)
Panjab University

Curated by ChEMBL
LigandPNGBDBM50611599(CHEMBL5266058)
Affinity DataEC50:  23nMAssay Description:Agonist activity at human TLR7 transfected in HEK293 cells assessed as induction of SEAP production incubated overnight by SEAP reporter gene based a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetToll-like receptor 7(Human)
Panjab University

Curated by ChEMBL
LigandPNGBDBM50611659(CHEMBL5266002)
Affinity DataEC50:  23nMAssay Description:Agonist activity at human TLR7 transfected in HEK293 cells assessed as induction of SEAP production incubated overnight by SEAP reporter gene based a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetToll-like receptor 7(Human)
Panjab University

Curated by ChEMBL
LigandPNGBDBM50611597(CHEMBL5279923)
Affinity DataEC50:  24nMAssay Description:Agonist activity at human TLR7 transfected in HEK293 cells assessed as induction of SEAP production incubated overnight by SEAP reporter gene based a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetToll-like receptor 7(Human)
Panjab University

Curated by ChEMBL
LigandPNGBDBM50611661(CHEMBL5280741)
Affinity DataEC50:  25nMAssay Description:Agonist activity at human TLR7 transfected in HEK293 cells assessed as induction of SEAP production incubated overnight by SEAP reporter gene based a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetToll-like receptor 7(Human)
Panjab University

Curated by ChEMBL
LigandPNGBDBM50611598(CHEMBL5273317)
Affinity DataEC50:  26nMAssay Description:Agonist activity at human TLR7 transfected in HEK293 cells assessed as induction of SEAP production incubated overnight by SEAP reporter gene based a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetToll-like receptor 7(Human)
Panjab University

Curated by ChEMBL
LigandPNGBDBM50611614(CHEMBL5284955)
Affinity DataEC50:  27nMAssay Description:Agonist activity at human TLR7 transfected in HEK293 cells assessed as induction of SEAP production incubated overnight by SEAP reporter gene based a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetToll-like receptor 7(Human)
Panjab University

Curated by ChEMBL
LigandPNGBDBM50611622(CHEMBL5279529)
Affinity DataEC50:  28nMAssay Description:Agonist activity at human TLR7 transfected in HEK293 cells assessed as induction of SEAP production incubated overnight by SEAP reporter gene based a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetToll-like receptor 7(Human)
Panjab University

Curated by ChEMBL
LigandPNGBDBM50330062(1-(3-(Aminomethyl)benzyl)-2-butyl-1H-imidazo[4,5-c...)
Affinity DataEC50:  29nMAssay Description:Agonist activity at human TLR7 expressed in HEK293 cells assessed as activation of NFkappaB incubated for 18 to 24 hrs by SEAP reporter gene based as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetToll-like receptor 7(Human)
Panjab University

Curated by ChEMBL
LigandPNGBDBM50608584(CHEMBL5275885)
Affinity DataEC50:  30nMAssay Description:Agonist activity at TLR7 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetToll-like receptor 7(Human)
Panjab University

Curated by ChEMBL
LigandPNGBDBM50611585(CHEMBL5289435)
Affinity DataEC50:  32nMAssay Description:Agonist activity at human TLR7 transfected in HEK293 cells assessed as induction of SEAP production incubated overnight by SEAP reporter gene based a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetToll-like receptor 7(Human)
Panjab University

Curated by ChEMBL
LigandPNGBDBM50611600(CHEMBL5283748)
Affinity DataEC50:  33nMAssay Description:Agonist activity at human TLR7 transfected in HEK293 cells assessed as induction of SEAP production incubated overnight by SEAP reporter gene based a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetToll-like receptor 8(Human)
Panjab University

Curated by ChEMBL
LigandPNGBDBM50330062(1-(3-(Aminomethyl)benzyl)-2-butyl-1H-imidazo[4,5-c...)
Affinity DataEC50:  33nMAssay Description:Agonist activity at human TLR8 expressed in HEK293 cells assessed as activation of NFkappaB incubated for 18 to 24 hrs by SEAP reporter gene based as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetToll-like receptor 7(Human)
Panjab University

Curated by ChEMBL
LigandPNGBDBM50611595(CHEMBL5267937)
Affinity DataEC50:  38nMAssay Description:Agonist activity at human TLR7 transfected in HEK293 cells assessed as induction of SEAP production incubated overnight by SEAP reporter gene based a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetToll-like receptor 7(Human)
Panjab University

Curated by ChEMBL
LigandPNGBDBM50611626(CHEMBL5275611)
Affinity DataEC50:  40nMAssay Description:Agonist activity at human TLR7 transfected in HEK293 cells assessed as induction of SEAP production incubated overnight by SEAP reporter gene based a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetToll-like receptor 7(Human)
Panjab University

Curated by ChEMBL
LigandPNGBDBM50611596(CHEMBL5280107)
Affinity DataEC50:  43nMAssay Description:Agonist activity at human TLR7 transfected in HEK293 cells assessed as induction of SEAP production incubated overnight by SEAP reporter gene based a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetToll-like receptor 7(Human)
Panjab University

Curated by ChEMBL
LigandPNGBDBM50611651(CHEMBL5272563)
Affinity DataEC50:  43nMAssay Description:Agonist activity at human TLR7 transfected in HEK293 cells assessed as induction of SEAP production incubated overnight by SEAP reporter gene based a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetToll-like receptor 7(Human)
Panjab University

Curated by ChEMBL
LigandPNGBDBM50611615(CHEMBL5281367)
Affinity DataEC50:  46nMAssay Description:Agonist activity at human TLR7 transfected in HEK293 cells assessed as induction of SEAP production incubated overnight by SEAP reporter gene based a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetToll-like receptor 7(Human)
Panjab University

Curated by ChEMBL
LigandPNGBDBM50611601(CHEMBL5269286)
Affinity DataEC50:  46nMAssay Description:Agonist activity at human TLR7 transfected in HEK293 cells assessed as induction of SEAP production incubated overnight by SEAP reporter gene based a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetToll-like receptor 7(Human)
Panjab University

Curated by ChEMBL
LigandPNGBDBM50611655(CHEMBL5271968)
Affinity DataEC50:  47nMAssay Description:Agonist activity at human TLR7 transfected in HEK293 cells assessed as induction of SEAP production incubated overnight by SEAP reporter gene based a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetToll-like receptor 7(Human)
Panjab University

Curated by ChEMBL
LigandPNGBDBM50611605(CHEMBL5270161)
Affinity DataEC50:  50nMAssay Description:Agonist activity at human TLR7 transfected in HEK293 cells assessed as induction of SEAP production incubated overnight by SEAP reporter gene based a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetToll-like receptor 7(Human)
Panjab University

Curated by ChEMBL
LigandPNGBDBM50611602(CHEMBL5281112)
Affinity DataEC50:  52nMAssay Description:Agonist activity at human TLR7 transfected in HEK293 cells assessed as induction of SEAP production incubated overnight by SEAP reporter gene based a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetToll-like receptor 7(Human)
Panjab University

Curated by ChEMBL
LigandPNGBDBM50611606(CHEMBL5274813)
Affinity DataEC50:  52nMAssay Description:Agonist activity at human TLR7 transfected in HEK293 cells assessed as induction of SEAP production incubated overnight by SEAP reporter gene based a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetToll-like receptor 7(Human)
Panjab University

Curated by ChEMBL
LigandPNGBDBM50611593(CHEMBL5272502)
Affinity DataEC50:  55nMAssay Description:Agonist activity at human TLR7 transfected in HEK293 cells assessed as induction of SEAP production incubated overnight by SEAP reporter gene based a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetToll-like receptor 7(Human)
Panjab University

Curated by ChEMBL
LigandPNGBDBM50611662(CHEMBL5272783)
Affinity DataEC50:  56nMAssay Description:Agonist activity at human TLR7 transfected in HEK293 cells assessed as induction of SEAP production incubated overnight by SEAP reporter gene based a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetToll-like receptor 7(Human)
Panjab University

Curated by ChEMBL
LigandPNGBDBM50611618(CHEMBL5283934)
Affinity DataEC50:  56nMAssay Description:Agonist activity at human TLR7 transfected in HEK293 cells assessed as induction of SEAP production incubated overnight by SEAP reporter gene based a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetToll-like receptor 7(Human)
Panjab University

Curated by ChEMBL
LigandPNGBDBM50611611(CHEMBL5269918)
Affinity DataEC50:  56nMAssay Description:Agonist activity at human TLR7 transfected in HEK293 cells assessed as induction of SEAP production incubated overnight by SEAP reporter gene based a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetToll-like receptor 7(Human)
Panjab University

Curated by ChEMBL
LigandPNGBDBM50611610(CHEMBL5269610)
Affinity DataEC50:  57nMAssay Description:Agonist activity at human TLR7 transfected in HEK293 cells assessed as induction of SEAP production incubated overnight by SEAP reporter gene based a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetToll-like receptor 7(Human)
Panjab University

Curated by ChEMBL
LigandPNGBDBM50611658(CHEMBL5290083)
Affinity DataEC50:  57nMAssay Description:Agonist activity at human TLR7 transfected in HEK293 cells assessed as induction of SEAP production incubated overnight by SEAP reporter gene based a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetToll-like receptor 7(Human)
Panjab University

Curated by ChEMBL
LigandPNGBDBM50611607(CHEMBL5278058)
Affinity DataEC50:  61nMAssay Description:Agonist activity at human TLR7 transfected in HEK293 cells assessed as induction of SEAP production incubated overnight by SEAP reporter gene based a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetToll-like receptor 7(Human)
Panjab University

Curated by ChEMBL
LigandPNGBDBM50611604(CHEMBL5268173)
Affinity DataEC50:  66nMAssay Description:Agonist activity at human TLR7 transfected in HEK293 cells assessed as induction of SEAP production incubated overnight by SEAP reporter gene based a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetToll-like receptor 7(Human)
Panjab University

Curated by ChEMBL
LigandPNGBDBM50241029(1-[4-amino-2-(ethoxymethyl)-1H-imidazo[4,5-c]quino...)
Affinity DataEC50:  67nMAssay Description:Agonist activity at human TLR7 expressed in HEK293 cells assessed as activation of NFkappaB incubated for 18 to 24 hrs by SEAP reporter gene based as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetToll-like receptor 7(Human)
Panjab University

Curated by ChEMBL
LigandPNGBDBM50611571(CHEMBL5284794)
Affinity DataEC50:  68nMAssay Description:Agonist activity at human TLR7 transfected in HEK293 cells assessed as induction of SEAP production incubated overnight by SEAP reporter gene based a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetToll-like receptor 7(Human)
Panjab University

Curated by ChEMBL
LigandPNGBDBM50611635(CHEMBL5273257)
Affinity DataEC50:  68nMAssay Description:Agonist activity at human TLR7 transfected in HEK293 cells assessed as induction of SEAP production incubated overnight by SEAP reporter gene based a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetToll-like receptor 8(Human)
Panjab University

Curated by ChEMBL
LigandPNGBDBM50330063(1-(4-(Aminomethyl)benzyl)-2-butyl-1H-imidazo[4,5-c...)
Affinity DataEC50:  68nMAssay Description:Agonist activity at human TLR8 expressed in HEK293 cells assessed as activation of NFkappaB incubated for 18 to 24 hrs by SEAP reporter gene based as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetToll-like receptor 7(Human)
Panjab University

Curated by ChEMBL
LigandPNGBDBM50611603(CHEMBL5288639)
Affinity DataEC50:  69nMAssay Description:Agonist activity at human TLR7 transfected in HEK293 cells assessed as induction of SEAP production incubated overnight by SEAP reporter gene based a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetToll-like receptor 7(Human)
Panjab University

Curated by ChEMBL
LigandPNGBDBM50611621(CHEMBL5284039)
Affinity DataEC50:  74nMAssay Description:Agonist activity at human TLR7 transfected in HEK293 cells assessed as induction of SEAP production incubated overnight by SEAP reporter gene based a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetToll-like receptor 7(Human)
Panjab University

Curated by ChEMBL
LigandPNGBDBM50611561(CHEMBL5273836)
Affinity DataEC50:  74nMAssay Description:Agonist activity at human TLR7 transfected in HEK293 cells assessed as induction of SEAP production incubated overnight by SEAP reporter gene based a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetToll-like receptor 7(Human)
Panjab University

Curated by ChEMBL
LigandPNGBDBM50611676(CHEMBL5272402)
Affinity DataEC50:  75nMAssay Description:Agonist activity at human TLR7 in HEK-Blue hTLR7 cells assessed as activation of NFkappaB by SEAP reporter gene based spectrophotometry assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetToll-like receptor 7(Human)
Panjab University

Curated by ChEMBL
LigandPNGBDBM50611684(CHEMBL5269245)
Affinity DataEC50:  75nMAssay Description:Agonist activity at human TLR7 in HEK-Blue hTLR7 cells assessed as activation of NFkappaB by SEAP reporter gene based spectrophotometry assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetToll-like receptor 7(Human)
Panjab University

Curated by ChEMBL
LigandPNGBDBM50611625(CHEMBL5267422)
Affinity DataEC50:  77nMAssay Description:Agonist activity at human TLR7 transfected in HEK293 cells assessed as induction of SEAP production incubated overnight by SEAP reporter gene based a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetToll-like receptor 7(Human)
Panjab University

Curated by ChEMBL
LigandPNGBDBM50611657(CHEMBL5281949)
Affinity DataEC50:  79nMAssay Description:Agonist activity at human TLR7 transfected in HEK293 cells assessed as induction of SEAP production incubated overnight by SEAP reporter gene based a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
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