Compile Data Set for Download or QSAR
Report error Found 8 Enz. Inhib. hit(s) with all data for entry = 50018102
TargetProstaglandin E2 receptor EP2 subtype(Human)
University of Tennessee Health Science Center

Curated by ChEMBL
LigandPNGBDBM50403532(CHEMBL5285583)
Affinity DataKi:  0.630nMAssay Description:Binding affinity to EP2 receptor in human mast cell assessed as inhibition constantMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2024
Entry Details
PubMed
TargetProstaglandin E2 receptor EP2 subtype(Human)
University of Tennessee Health Science Center

Curated by ChEMBL
LigandPNGBDBM50403531(PF-04418948 | Pf-04418948)
Affinity DataKi:  7.60nMAssay Description:Binding affinity to human EP2 receptor expressed in CHO cells assessed as inhibition constantMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2024
Entry Details
PubMed
TargetProstaglandin D2 receptor(Human)
University of Tennessee Health Science Center

Curated by ChEMBL
LigandPNGBDBM50403532(CHEMBL5285583)
Affinity DataKi:  1.20E+3nMAssay Description:Binding affinity to DP1 receptor in human mast cell assessed as inhibition constantMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2024
Entry Details
PubMed
TargetProstaglandin D2 receptor(Human)
University of Tennessee Health Science Center

Curated by ChEMBL
LigandPNGBDBM50403531(PF-04418948 | Pf-04418948)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity to human DP1 receptor expressed in CHO cells assessed as inhibition constantMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2024
Entry Details
PubMed
TargetProstaglandin E2 receptor EP1 subtype(Human)
University of Tennessee Health Science Center

Curated by ChEMBL
LigandPNGBDBM50403531(PF-04418948 | Pf-04418948)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity to EP1 receptor (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2024
Entry Details
PubMed
TargetProstaglandin E2 receptor EP3 subtype(Human)
University of Tennessee Health Science Center

Curated by ChEMBL
LigandPNGBDBM50403531(PF-04418948 | Pf-04418948)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity to EP3 receptor (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2024
Entry Details
PubMed
TargetProstaglandin E2 receptor EP4 subtype(Human)
University of Tennessee Health Science Center

Curated by ChEMBL
LigandPNGBDBM50403531(PF-04418948 | Pf-04418948)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity to human EP4 receptor expressed in CHO cells assessed as inhibition constantMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2024
Entry Details
PubMed
TargetProstaglandin E2 receptor EP4 subtype(Human)
University of Tennessee Health Science Center

Curated by ChEMBL
LigandPNGBDBM50403532(CHEMBL5285583)
Affinity DataKi:  1.63E+4nMAssay Description:Binding affinity to EP4 receptor in human mast cell assessed as inhibition constantMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2024
Entry Details
PubMed