Compile Data Set for Download or QSAR
Report error Found 104 Enz. Inhib. hit(s) with all data for entry = 50017414
TargetFurin(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50601761(CHEMBL5203869 | US11773078, Example 263)
Affinity DataIC50: 0.158nMAssay Description:Inhibition of Tev-FLAG-His-tagged furin (108 to 574 residues) (unknown origin) using FAM-QRVRRAVGIDK-TAMRA as substrate and measured after 2 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetFurin(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50601763(CHEMBL5197625 | US11773078, Example 62)
Affinity DataIC50: 0.158nMAssay Description:Inhibition of Tev-FLAG-His-tagged furin (108 to 574 residues) (unknown origin) using FAM-QRVRRAVGIDK-TAMRA as substrate and measured after 2 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetFurin(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50601747(CHEMBL5175553 | US11773078, Example 11)
Affinity DataIC50: 0.251nMAssay Description:Inhibition of Tev-FLAG-His-tagged furin (108 to 574 residues) (unknown origin) using FAM-QRVRRAVGIDK-TAMRA as substrate and measured after 2 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetFurin(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50601762(CHEMBL5190891 | US11773078, Example 369)
Affinity DataIC50: 0.501nMAssay Description:Inhibition of Tev-FLAG-His-tagged furin (108 to 574 residues) (unknown origin) using FAM-QRVRRAVGIDK-TAMRA as substrate and measured after 2 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetFurin(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50601703(CHEMBL5202322)
Affinity DataIC50: 0.560nMAssay Description:Inhibition of furin (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetFurin(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50601704(CHEMBL5184039)
Affinity DataIC50: 0.560nMAssay Description:Inhibition of furin (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetFurin(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50601759(CHEMBL5175809 | US11773078, Example 298)
Affinity DataIC50: 0.631nMAssay Description:Inhibition of Tev-FLAG-His-tagged furin (108 to 574 residues) (unknown origin) using FAM-QRVRRAVGIDK-TAMRA as substrate and measured after 2 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetFurin(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50601749(CHEMBL5171461 | US11773078, Example 180)
Affinity DataIC50: 0.794nMAssay Description:Inhibition of Tev-FLAG-His-tagged furin (108 to 574 residues) (unknown origin) using FAM-QRVRRAVGIDK-TAMRA as substrate and measured after 2 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetFurin(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50601750(CHEMBL5182363 | US11773078, Example 41)
Affinity DataIC50: 0.794nMAssay Description:Inhibition of Tev-FLAG-His-tagged furin (108 to 574 residues) (unknown origin) using FAM-QRVRRAVGIDK-TAMRA as substrate and measured after 2 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetFurin(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50601754(CHEMBL5208861 | US11773078, Example 207)
Affinity DataIC50: 0.794nMAssay Description:Inhibition of Tev-FLAG-His-tagged furin (108 to 574 residues) (unknown origin) using FAM-QRVRRAVGIDK-TAMRA as substrate and measured after 2 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetFurin(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50601757(CHEMBL5206910 | US11773078, Example 131)
Affinity DataIC50: 0.794nMAssay Description:Inhibition of Tev-FLAG-His-tagged furin (108 to 574 residues) (unknown origin) using FAM-QRVRRAVGIDK-TAMRA as substrate and measured after 2 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetFurin(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50601755(CHEMBL5195577 | US11773078, Example 126)
Affinity DataIC50: 1nMAssay Description:Inhibition of Tev-FLAG-His-tagged furin (108 to 574 residues) (unknown origin) using FAM-QRVRRAVGIDK-TAMRA as substrate and measured after 2 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetFurin(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50601756(CHEMBL5196204 | US11773078, Example 334)
Affinity DataIC50: 1.30nMAssay Description:Inhibition of Tev-FLAG-His-tagged furin (108 to 574 residues) (unknown origin) using FAM-QRVRRAVGIDK-TAMRA as substrate and measured after 2 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetFurin(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50601760(CHEMBL5180159 | US11773078, Example 306)
Affinity DataIC50: 1.30nMAssay Description:Inhibition of Tev-FLAG-His-tagged furin (108 to 574 residues) (unknown origin) using FAM-QRVRRAVGIDK-TAMRA as substrate and measured after 2 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetFurin(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50601752(CHEMBL5172689 | US11773078, Example 340)
Affinity DataIC50: 1.60nMAssay Description:Inhibition of Tev-FLAG-His-tagged furin (108 to 574 residues) (unknown origin) using FAM-QRVRRAVGIDK-TAMRA as substrate and measured after 2 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetFurin(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50601746(CHEMBL5172764 | US11773078, Example 10)
Affinity DataIC50: 2nMAssay Description:Inhibition of Tev-FLAG-His-tagged furin (108 to 574 residues) (unknown origin) using FAM-QRVRRAVGIDK-TAMRA as substrate and measured after 2 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetFurin(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50601751(CHEMBL5200817 | US11773078, Example 339)
Affinity DataIC50: 2nMAssay Description:Inhibition of Tev-FLAG-His-tagged furin (108 to 574 residues) (unknown origin) using FAM-QRVRRAVGIDK-TAMRA as substrate and measured after 2 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetFurin(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50601753(CHEMBL5207406 | US11773078, Example 206)
Affinity DataIC50: 2.5nMAssay Description:Inhibition of Tev-FLAG-His-tagged furin (108 to 574 residues) (unknown origin) using FAM-QRVRRAVGIDK-TAMRA as substrate and measured after 2 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetFurin(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50601758(CHEMBL5170962 | US11773078, Example 242)
Affinity DataIC50: 2.5nMAssay Description:Inhibition of Tev-FLAG-His-tagged furin (108 to 574 residues) (unknown origin) using FAM-QRVRRAVGIDK-TAMRA as substrate and measured after 2 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetFurin(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50601702(CHEMBL5199257)
Affinity DataIC50: 3nMAssay Description:Inhibition of furin (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetFurin(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50601748(CHEMBL5169887 | US11773078, Example 12)
Affinity DataIC50: 5nMAssay Description:Inhibition of Tev-FLAG-His-tagged furin (108 to 574 residues) (unknown origin) using FAM-QRVRRAVGIDK-TAMRA as substrate and measured after 2 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetFurin(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50601701(CHEMBL5177253)
Affinity DataIC50: 9.5nMAssay Description:Inhibition of furin (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetFurin(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50399746(CHEMBL2179435)
Affinity DataIC50: 20nMAssay Description:Inhibition of furin (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetProprotein convertase subtilisin/kexin type 6(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50399746(CHEMBL2179435)
Affinity DataIC50: 30nMAssay Description:Inhibition of PACE4 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetFurin(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM29692(3-ethyl-2-[(E,3E)-3-(3-ethylthiazolidin-2-ylidene)...)
Affinity DataIC50: 3.15E+4nMAssay Description:Inhibition of furin (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetFurin(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM29692(3-ethyl-2-[(E,3E)-3-(3-ethylthiazolidin-2-ylidene)...)
Affinity DataIC50: 3.38E+4nMAssay Description:Inhibition of furin (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetFurin(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50552678(CHEMBL4759036)
Affinity DataKi:  0.00500nMAssay Description:Inhibition of human furin expressed in HEK293 cells using pGlu-Arg-Thr-LysArg-AMC as substrate and measured by fluorescence based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetFurin(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50601724(CHEMBL5190391)
Affinity DataKi:  0.00600nMAssay Description:Inhibition of recombinant human furin using Phac-Arg-Val-Arg-Arg-AMC as substrate incubated for 30 mins and measured by microplate reader methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetFurin(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50601696(CHEMBL5189844)
Affinity DataKi:  0.00800nMAssay Description:Inhibition of human furin expressed in HEK293 cells using pGlu-Arg-Thr-LysArg-AMC as substrate and measured by fluorescence based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetFurin(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50601705(CHEMBL5203612)
Affinity DataKi:  0.00900nMAssay Description:Inhibition of furin (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetFurin(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50601720(CHEMBL5188244)
Affinity DataKi:  0.0100nMAssay Description:Inhibition of recombinant human furin using Phac-Arg-Val-Arg-Arg-AMC as substrate incubated for 30 mins and measured by microplate reader methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetFurin(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50601719(CHEMBL5193701)
Affinity DataKi:  0.0130nMAssay Description:Inhibition of recombinant human furin using Phac-Arg-Val-Arg-Arg-AMC as substrate incubated for 30 mins and measured by microplate reader methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetFurin(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50601721(CHEMBL5205365)
Affinity DataKi:  0.0140nMAssay Description:Inhibition of recombinant human furin using Phac-Arg-Val-Arg-Arg-AMC as substrate incubated for 30 mins and measured by microplate reader methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetFurin(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50601698(CHEMBL5175269)
Affinity DataKi:  0.0160nMAssay Description:Inhibition of human furin expressed in HEK293 cells using pGlu-Arg-Thr-LysArg-AMC as substrate and measured by fluorescence based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetFurin(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50601700(CHEMBL5207872)
Affinity DataKi:  0.0220nMAssay Description:Inhibition of furin (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetFurin(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50601703(CHEMBL5202322)
Affinity DataKi:  0.0223nMAssay Description:Inhibition of furin (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetFurin(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50601723(CHEMBL5203853)
Affinity DataKi:  0.0280nMAssay Description:Inhibition of recombinant human furin using Phac-Arg-Val-Arg-Arg-AMC as substrate incubated for 30 mins and measured by microplate reader methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetFurin(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50601722(CHEMBL5176040)
Affinity DataKi:  0.0340nMAssay Description:Inhibition of recombinant human furin using Phac-Arg-Val-Arg-Arg-AMC as substrate incubated for 30 mins and measured by microplate reader methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetFurin(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50601716(CHEMBL5207759)
Affinity DataKi:  0.0538nMAssay Description:Inhibition of furin (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetFurin(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50601712(CHEMBL5207183)
Affinity DataKi:  0.110nMAssay Description:Inhibition of furin (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetFurin(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50601697(CHEMBL5179893)
Affinity DataKi:  0.170nMAssay Description:Inhibition of human furin expressed in HEK293 cells using pGlu-Arg-Thr-LysArg-AMC as substrate and measured by fluorescence based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetFurin(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50601699(CHEMBL5191544)
Affinity DataKi:  0.196nMAssay Description:Inhibition of human furin expressed in HEK293 cells using pGlu-Arg-Thr-LysArg-AMC as substrate and measured by fluorescence based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetFurin(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50601714(CHEMBL5202985)
Affinity DataKi:  0.491nMAssay Description:Inhibition of furin (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetFurin(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50601710(CHEMBL5175238)
Affinity DataKi:  0.504nMAssay Description:Inhibition of furin (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetFurin(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50601717(CHEMBL5174341)
Affinity DataKi:  0.618nMAssay Description:Inhibition of furin (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetFurin(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50303774(phenylacetyl-Arg-Val-Arg-4-amidinobenzylamide | CH...)
Affinity DataKi:  0.660nMAssay Description:Inhibition of human furin expressed in HEK293 cells using pGlu-Arg-Thr-LysArg-AMC as substrate and measured by fluorescence based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetFurin(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50601713(CHEMBL5179100)
Affinity DataKi:  0.680nMAssay Description:Inhibition of furin (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetFurin(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50601702(CHEMBL5199257)
Affinity DataKi:  0.800nMAssay Description:Inhibition of furin (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetFurin(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50601711(CHEMBL5207252)
Affinity DataKi:  1.10nMAssay Description:Inhibition of furin (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetFurin(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50601715(CHEMBL5189192)
Affinity DataKi:  1.20nMAssay Description:Inhibition of furin (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
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