Compile Data Set for Download or QSAR
Report error Found 30 Enz. Inhib. hit(s) with all data for entry = 50018654
TargetHistone deacetylase 3(Human)
Xinyang Normal University

Curated by ChEMBL
LigandPNGBDBM50464790(CHEMBL4288953)
Affinity DataIC50: 0.75nMAssay Description:Inhibition of HDAC3 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetHistone deacetylase 6(Human)
Xinyang Normal University

Curated by ChEMBL
LigandPNGBDBM50464790(CHEMBL4288953)
Affinity DataIC50: 1.10nMAssay Description:Inhibition of HDAC6 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetHistone deacetylase 1(Human)
Xinyang Normal University

Curated by ChEMBL
LigandPNGBDBM50464790(CHEMBL4288953)
Affinity DataIC50: 2.80nMAssay Description:Inhibition of HDAC1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetHistone deacetylase 6(Human)
Xinyang Normal University

Curated by ChEMBL
LigandPNGBDBM50610754(CHEMBL5278415)
Affinity DataIC50: 7.60nMAssay Description:Inhibition of HDAC6 (unknown origin) using (Boc-Lys (Ac)-AMC substrate incubated for 30 mins by fluorescence plate reader analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetHistone deacetylase 1(Human)
Xinyang Normal University

Curated by ChEMBL
LigandPNGBDBM50610754(CHEMBL5278415)
Affinity DataIC50: 29nMAssay Description:Inhibition of HDAC1 (unknown origin) using (Boc-Lys (Ac)-AMC substrate incubated for 30 mins by fluorescence plate reader analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetSerine/threonine-protein kinase PLK1(Human)
Xinyang Normal University

Curated by ChEMBL
LigandPNGBDBM50610758(CHEMBL5280383)
Affinity DataIC50: 310nMAssay Description:Inhibition of PLK1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetSerine/threonine-protein kinase PLK1(Human)
Xinyang Normal University

Curated by ChEMBL
LigandPNGBDBM50395381(CHEMBL2164716 | US9168247, JR95)
Affinity DataIC50: 527nMAssay Description:Inhibition of PLK1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetSerine/threonine-protein kinase haspin(Human)
Xinyang Normal University

Curated by ChEMBL
LigandPNGBDBM100152(cid_5359389 | SMR001233259 | HARMINE | 7-methoxy-1...)
Affinity DataIC50: 590nMAssay Description:Inhibition of HASPIN (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetSerine/threonine-protein kinase PLK3(Human)
Xinyang Normal University

Curated by ChEMBL
LigandPNGBDBM50395381(CHEMBL2164716 | US9168247, JR95)
Affinity DataIC50: 607nMAssay Description:Inhibition of PLK3 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetSerine/threonine-protein kinase haspin(Human)
Xinyang Normal University

Curated by ChEMBL
LigandPNGBDBM50047009(CHEMBL1535235 | 1-methyl-9H-pyrido[3,4-b]indol-7-o...)
Affinity DataIC50: 770nMAssay Description:Inhibition of HASPIN (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetSerine/threonine-protein kinase PLK1(Human)
Xinyang Normal University

Curated by ChEMBL
LigandPNGBDBM50610757(CHEMBL5269742)
Affinity DataIC50: 854nMAssay Description:Inhibition of PLK1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetSerine/threonine-protein kinase PLK1(Human)
Xinyang Normal University

Curated by ChEMBL
LigandPNGBDBM50610756(CHEMBL5287676)
Affinity DataIC50: 897nMAssay Description:Inhibition of PLK1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetSerine/threonine-protein kinase PLK3(Human)
Xinyang Normal University

Curated by ChEMBL
LigandPNGBDBM50610757(CHEMBL5269742)
Affinity DataIC50: 1.11E+3nMAssay Description:Inhibition of PLK3 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetSerine/threonine-protein kinase PLK3(Human)
Xinyang Normal University

Curated by ChEMBL
LigandPNGBDBM50610758(CHEMBL5280383)
Affinity DataIC50: 1.81E+3nMAssay Description:Inhibition of PLK3 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetDNA topoisomerase 1(Human)
Xinyang Normal University

Curated by ChEMBL
LigandPNGBDBM50610761(CHEMBL5270699)
Affinity DataIC50: 2.50E+3nMAssay Description:Inhibition of Topoisomerase 1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetSerine/threonine-protein kinase PLK2(Human)
Xinyang Normal University

Curated by ChEMBL
LigandPNGBDBM50610757(CHEMBL5269742)
Affinity DataIC50: 3.82E+3nMAssay Description:Inhibition of PLK2 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetSerine/threonine-protein kinase PLK2(Human)
Xinyang Normal University

Curated by ChEMBL
LigandPNGBDBM50395381(CHEMBL2164716 | US9168247, JR95)
Affinity DataIC50: 4.30E+3nMAssay Description:Inhibition of PLK2 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
Xinyang Normal University

Curated by ChEMBL
LigandPNGBDBM50608893(CHEMBL5200447)
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of human CDK5/p25 nck5aMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetDNA topoisomerase 1(Human)
Xinyang Normal University

Curated by ChEMBL
LigandPNGBDBM50610759(CHEMBL5272233)
Affinity DataIC50: 5.80E+3nMAssay Description:Inhibition of Topoisomerase 1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
Xinyang Normal University

Curated by ChEMBL
LigandPNGBDBM50608893(CHEMBL5200447)
Affinity DataIC50: 6.00E+3nMAssay Description:Inhibition of human CDK2/Cyclin A in presence of gamma32P-ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetSerine/threonine-protein kinase PLK2(Human)
Xinyang Normal University

Curated by ChEMBL
LigandPNGBDBM50610758(CHEMBL5280383)
Affinity DataIC50: 6.45E+3nMAssay Description:Inhibition of PLK2 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetDNA topoisomerase 1(Human)
Xinyang Normal University

Curated by ChEMBL
LigandPNGBDBM50610760(CHEMBL5279607)
Affinity DataIC50: 7.80E+3nMAssay Description:Inhibition of Topoisomerase 1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetKinesin-like protein KIF11(Human)
Xinyang Normal University

Curated by ChEMBL
LigandPNGBDBM50610760(CHEMBL5279607)
Affinity DataIC50: 8.73E+3nMAssay Description:Inhibition of KSP (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetKinesin-like protein KIF11(Human)
Xinyang Normal University

Curated by ChEMBL
LigandPNGBDBM50610761(CHEMBL5270699)
Affinity DataIC50: 8.91E+3nMAssay Description:Inhibition of KSP (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetKinesin-like protein KIF11(Human)
Xinyang Normal University

Curated by ChEMBL
LigandPNGBDBM50610759(CHEMBL5272233)
Affinity DataIC50: 1.34E+4nMAssay Description:Inhibition of KSP (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
Xinyang Normal University

Curated by ChEMBL
LigandPNGBDBM100152(cid_5359389 | SMR001233259 | HARMINE | 7-methoxy-1...)
Affinity DataIC50: 1.70E+4nMAssay Description:Inhibition of cdk1/Cyclin B (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
Xinyang Normal University

Curated by ChEMBL
LigandPNGBDBM100152(cid_5359389 | SMR001233259 | HARMINE | 7-methoxy-1...)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of human CDK5/p25 nck5aMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
Xinyang Normal University

Curated by ChEMBL
LigandPNGBDBM50610755(CHEMBL5274823)
Affinity DataIC50: 2.70E+4nMAssay Description:Inhibition of CDK2/Cyclin A (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetDNA topoisomerase 1(Human)
Xinyang Normal University

Curated by ChEMBL
LigandPNGBDBM50013811(9H-pyrido[3,4-b]indole | Norharman | CHEMBL275224 ...)
Affinity DataIC50: 3.10E+4nMAssay Description:Inhibition of Topoisomerase 1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
Xinyang Normal University

Curated by ChEMBL
LigandPNGBDBM100152(cid_5359389 | SMR001233259 | HARMINE | 7-methoxy-1...)
Affinity DataIC50: 3.30E+4nMAssay Description:Inhibition of CDK2/Cyclin A (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed