Compile Data Set for Download or QSAR
Report error Found 6 Enz. Inhib. hit(s) with all data for entry = 50018653
TargetCollagenase 3(Human)
Sichuan University-University of Oxford Huaxi Joint Centre For Gastrointestinal Cancer

Curated by ChEMBL
LigandPNGBDBM50610752(CHEMBL5268707)
Affinity DataIC50: 6nMAssay Description:Inhibition of MMP-13 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetStromelysin-2(Human)
Sichuan University-University of Oxford Huaxi Joint Centre For Gastrointestinal Cancer

Curated by ChEMBL
LigandPNGBDBM50610751(CHEMBL5278446)
Affinity DataIC50: 24nMAssay Description:Inhibition of MMP-10 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetCollagenase 3(Human)
Sichuan University-University of Oxford Huaxi Joint Centre For Gastrointestinal Cancer

Curated by ChEMBL
LigandPNGBDBM50610751(CHEMBL5278446)
Affinity DataIC50: 460nMAssay Description:Inhibition of MMP-13 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetStromelysin-2(Human)
Sichuan University-University of Oxford Huaxi Joint Centre For Gastrointestinal Cancer

Curated by ChEMBL
LigandPNGBDBM50610753(CHEMBL5280150)
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibition of MMP10 (unknown origin) using FRET peptideMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetMatrilysin(Human)
Sichuan University-University of Oxford Huaxi Joint Centre For Gastrointestinal Cancer

Curated by ChEMBL
LigandPNGBDBM50610753(CHEMBL5280150)
Affinity DataIC50: 2.20E+3nMAssay Description:Inhibition of MMP7 (unknown origin) using FRET peptideMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetCollagenase 3(Human)
Sichuan University-University of Oxford Huaxi Joint Centre For Gastrointestinal Cancer

Curated by ChEMBL
LigandPNGBDBM50361639(CHEMBL1371684)
Affinity DataIC50: 2.40E+3nMAssay Description:Inhibition of MMP-13 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMedPDB3D3D Structure (crystal)