Report error Found 45 Enz. Inhib. hit(s) with all data for entry = 50018099
Affinity DataKd: 210nMAssay Description:Binding affinity to human MDM4 assessed as inhibition constantMore data for this Ligand-Target Pair
Affinity DataEC50: 2.30E+3nMAssay Description:Inhibition of human MDM4More data for this Ligand-Target Pair
Affinity DataKd: 43nMAssay Description:Binding affinity to human MDM4 assessed as dissociation constant by ITC assayMore data for this Ligand-Target Pair
Affinity DataKd: 25nMAssay Description:Binding affinity to human MDM4 assessed as dissociation constantMore data for this Ligand-Target Pair
TargetE3 ubiquitin-protein ligase Mdm2(Human)
University of Chinese Academy of Sciences
Curated by ChEMBL
University of Chinese Academy of Sciences
Curated by ChEMBL
Affinity DataEC50: 2.60E+4nMAssay Description:Inhibition of human MDM2More data for this Ligand-Target Pair
Affinity DataKd: 27nMAssay Description:Inhibition of human his-tagged MDM4 assessed as dissociation constant by ITC assayMore data for this Ligand-Target Pair
TargetE3 ubiquitin-protein ligase Mdm2(Human)
University of Chinese Academy of Sciences
Curated by ChEMBL
University of Chinese Academy of Sciences
Curated by ChEMBL
Affinity DataKd: 149nMAssay Description:Binding affinity to human MDM2 assessed as dissociation constantMore data for this Ligand-Target Pair
Affinity DataKd: 13nMAssay Description:Binding affinity to human MDM4 assessed as dissociation constant by FP assayMore data for this Ligand-Target Pair
Affinity DataKd: 229nMAssay Description:Binding affinity to human MDM4 assessed as dissociation constant by FP assayMore data for this Ligand-Target Pair
Affinity DataKd: <100nMAssay Description:Inhibition of MDM4 assessed as dissociation constantMore data for this Ligand-Target Pair
TargetE3 ubiquitin-protein ligase Mdm2(Human)
University of Chinese Academy of Sciences
Curated by ChEMBL
University of Chinese Academy of Sciences
Curated by ChEMBL
Affinity DataKd: 12nMAssay Description:Binding affinity to human MDM2 assessed as dissociation constant by FP assayMore data for this Ligand-Target Pair
TargetE3 ubiquitin-protein ligase Mdm2(Human)
University of Chinese Academy of Sciences
Curated by ChEMBL
University of Chinese Academy of Sciences
Curated by ChEMBL
Affinity DataKd: 216nMAssay Description:Binding affinity to human MDM2 assessed as dissociation constant by FP assayMore data for this Ligand-Target Pair
TargetE3 ubiquitin-protein ligase Mdm2(Human)
University of Chinese Academy of Sciences
Curated by ChEMBL
University of Chinese Academy of Sciences
Curated by ChEMBL
Affinity DataKd: 600nMAssay Description:Binding affinity to human MDM2 assessed as inhibition constantMore data for this Ligand-Target Pair
Affinity DataIC50: 0.210nMAssay Description:Inhibition of human MDM4 by SRP assayMore data for this Ligand-Target Pair
TargetE3 ubiquitin-protein ligase Mdm2(Human)
University of Chinese Academy of Sciences
Curated by ChEMBL
University of Chinese Academy of Sciences
Curated by ChEMBL
Affinity DataIC50: 0.210nMAssay Description:Binding affinity to human MDM2 assessed as inhibition constantMore data for this Ligand-Target Pair
TargetE3 ubiquitin-protein ligase Mdm2(Human)
University of Chinese Academy of Sciences
Curated by ChEMBL
University of Chinese Academy of Sciences
Curated by ChEMBL
Affinity DataIC50: 0.900nMAssay Description:Binding affinity to human MDM2 assessed as inhibition constantMore data for this Ligand-Target Pair
TargetE3 ubiquitin-protein ligase Mdm2(Human)
University of Chinese Academy of Sciences
Curated by ChEMBL
University of Chinese Academy of Sciences
Curated by ChEMBL
Affinity DataIC50: 17nMAssay Description:Inhibition of human MDM2More data for this Ligand-Target Pair
Affinity DataIC50: 17nMAssay Description:Inhibition of human MDM4 by TR-FRET assayMore data for this Ligand-Target Pair
TargetE3 ubiquitin-protein ligase Mdm2(Human)
University of Chinese Academy of Sciences
Curated by ChEMBL
University of Chinese Academy of Sciences
Curated by ChEMBL
Affinity DataIC50: 19nMAssay Description:Antagonist activity against human MDM2 by TR-FRET assayMore data for this Ligand-Target Pair
TargetE3 ubiquitin-protein ligase Mdm2(Human)
University of Chinese Academy of Sciences
Curated by ChEMBL
University of Chinese Academy of Sciences
Curated by ChEMBL
Affinity DataIC50: 20nMAssay Description:Inhibition of human MDM2 by ELISA assayMore data for this Ligand-Target Pair
Affinity DataIC50: 25nMAssay Description:Inhibition of human MDM4More data for this Ligand-Target Pair
TargetE3 ubiquitin-protein ligase Mdm2(Human)
University of Chinese Academy of Sciences
Curated by ChEMBL
University of Chinese Academy of Sciences
Curated by ChEMBL
Affinity DataIC50: 33nMAssay Description:Inhibition of human MDM2More data for this Ligand-Target Pair
Affinity DataIC50: 40nMAssay Description:Inhibition of human MDM4 by ELISA assayMore data for this Ligand-Target Pair
Affinity DataIC50: 41nMAssay Description:Inhibition of human MDM4More data for this Ligand-Target Pair
TargetE3 ubiquitin-protein ligase Mdm2(Human)
University of Chinese Academy of Sciences
Curated by ChEMBL
University of Chinese Academy of Sciences
Curated by ChEMBL
Affinity DataIC50: 44nMAssay Description:Inhibition of human MDM2 by ELISA assayMore data for this Ligand-Target Pair
Affinity DataIC50: 110nMAssay Description:Inhibition of human MDM4 by ELISA assayMore data for this Ligand-Target Pair
Affinity DataIC50: 145nMAssay Description:Inhibition of human MDM4 by TR-FRET assayMore data for this Ligand-Target Pair
Affinity DataIC50: 550nMAssay Description:Inhibition of human MDM4 by ELISA assayMore data for this Ligand-Target Pair
Affinity DataIC50: 3.00E+3nMAssay Description:Binding affinity to human MDM4 assessed as inhibition constantMore data for this Ligand-Target Pair
Affinity DataIC50: 3.70E+3nMAssay Description:Inhibition of human MDM4 by TR-FRET assayMore data for this Ligand-Target Pair
TargetE3 ubiquitin-protein ligase Mdm2(Human)
University of Chinese Academy of Sciences
Curated by ChEMBL
University of Chinese Academy of Sciences
Curated by ChEMBL
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of human MDM2 by TR-FRET assayMore data for this Ligand-Target Pair
Affinity DataKi: 6.80nMAssay Description:Binding affinity to human MDM4 assessed as inhibition constantMore data for this Ligand-Target Pair
TargetE3 ubiquitin-protein ligase Mdm2(Human)
University of Chinese Academy of Sciences
Curated by ChEMBL
University of Chinese Academy of Sciences
Curated by ChEMBL
Affinity DataKi: 7.70nMAssay Description:Binding affinity to human MDM2 assessed as inhibition constant by fluorescence based assayMore data for this Ligand-Target Pair
Affinity DataKi: 25nMAssay Description:Binding affinity to human MDM4 assessed as inhibition constant by fluorescence based assayMore data for this Ligand-Target Pair
TargetE3 ubiquitin-protein ligase Mdm2(Human)
University of Chinese Academy of Sciences
Curated by ChEMBL
University of Chinese Academy of Sciences
Curated by ChEMBL
Affinity DataKi: 109nMAssay Description:Binding affinity to human MDM2 assessed as inhibition constant by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataKi: 620nMAssay Description:Binding affinity to human MDM4 assessed as dissociation constantMore data for this Ligand-Target Pair
TargetE3 ubiquitin-protein ligase Mdm2(Human)
University of Chinese Academy of Sciences
Curated by ChEMBL
University of Chinese Academy of Sciences
Curated by ChEMBL
Affinity DataKi: 620nMAssay Description:Binding affinity to human MDM2 assessed as dissociation constantMore data for this Ligand-Target Pair
TargetE3 ubiquitin-protein ligase Mdm2(Human)
University of Chinese Academy of Sciences
Curated by ChEMBL
University of Chinese Academy of Sciences
Curated by ChEMBL
Affinity DataKi: 916nMAssay Description:Binding affinity to human MDM2 assessed as dissociation constant by FP assayMore data for this Ligand-Target Pair
TargetE3 ubiquitin-protein ligase Mdm2(Human)
University of Chinese Academy of Sciences
Curated by ChEMBL
University of Chinese Academy of Sciences
Curated by ChEMBL
Affinity DataKi: 5.50E+3nMAssay Description:Binding affinity to human MDM2 assessed as dissociation constantMore data for this Ligand-Target Pair
Affinity DataKi: 1.10E+4nMAssay Description:Binding affinity to human MDM4 assessed as inhibition constant by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataKi: 3.60E+4nMAssay Description:Binding affinity to human MDM4 assessed as dissociation constant by FP assayMore data for this Ligand-Target Pair
TargetE3 ubiquitin-protein ligase Mdm2(Human)
University of Chinese Academy of Sciences
Curated by ChEMBL
University of Chinese Academy of Sciences
Curated by ChEMBL
Affinity DataKi: 5.40E+4nMAssay Description:Binding affinity to human MDM2 assessed as dissociation constantMore data for this Ligand-Target Pair
TargetE3 ubiquitin-protein ligase Mdm2(Human)
University of Chinese Academy of Sciences
Curated by ChEMBL
University of Chinese Academy of Sciences
Curated by ChEMBL
Affinity DataKi: 5.40E+4nMAssay Description:Binding affinity to human MDM2 assessed as dissociation constantMore data for this Ligand-Target Pair
Affinity DataKi: 6.90E+4nMAssay Description:Binding affinity to human MDM4 assessed as dissociation constant by FP assayMore data for this Ligand-Target Pair
TargetE3 ubiquitin-protein ligase Mdm2(Human)
University of Chinese Academy of Sciences
Curated by ChEMBL
University of Chinese Academy of Sciences
Curated by ChEMBL
Affinity DataKi: 7.00E+4nMAssay Description:Binding affinity to human MDM2 assessed as dissociation constant by FP assayMore data for this Ligand-Target Pair
